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Joule, J. A. et al.: 2017 Science of Synthesis, 2017/1: Knowledge Updates 2017/1 DOI: 10.1055/sos-SD-110-01022
Knowledge Updates 2017/1

10.22.4 Product Subclass 4: 1,2-Dihydroazaindol-3-ones

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Editors: Joule, J. A.; Krause, N.; Oestreich, M.; Rademann, J.; Schaumann, E.; Wirth, T.

Authors: Albericio, F.; Atodiresei, I.; Baba, A.; Baker, A.; Braun, M.; Cherkupally, P.; Delvos, L.; Govender, T.; Hardman-Baldwin, A. M.; Joseph, B.; Kleeberg, C.; Kruger, H. G.; Mattson, A. E.; Mérour, J.-Y.; Nishimoto, Y.; Oestreich, M.; Qian, D.; Ramesh, S.; Rueping, M.; Singh, F. V.; de la Torre, B. G.; Wirth, T.; Yasuda, M.; Zhang, J.

Title: Knowledge Updates 2017/1

Print ISBN: 9783132414105; Online ISBN: 9783132414136; Book DOI: 10.1055/b-004-140261

1st edition © 2017 Thieme. All rights reserved.
Georg Thieme Verlag KG, Stuttgart

Subjects: Organic Chemistry

Science of Synthesis Knowledge Updates



Parent publication

Title: Science of Synthesis

DOI: 10.1055/b-00000101

Series Editors: Carreira, E. M.; Decicco, C. P.; Fürstner, A.; Koch, G.; Molander, G.; Schaumann, E.; Shibasaki, M.; Thomas, E. J.; Trost, B. M.

Type: Multivolume Edition

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Abstract

This chapter reviews the synthesis and reactivity of 1,2-dihydroazaindol-3-ones (azaindoxyls) and related 1,2-dihydroazaindol-3-yl acetates. Synthetic preparations are reviewed for all isomers except for 1,2-dihydro-3H-pyrrolo[2,3-c]pyridin-3-ones.

Key words

1,2-dihydroazaindol-3-ones - azaindoxyls - 1,2-dihydroazaindol-3-yl acetates - cyclization - C2-aldolization
 
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