16.12.5 Pyrimidines (Update 2020)

Abstract

This chapter is an update to the earlier Science of Synthesis contributions (Section 16.12 and 16.12.5) covering the synthesis and substituent modification of pyrimidines. It focuses on the literature published in the period 2012–2019, gathering all the methods reported in this period, but with a particular emphasis on transition-metal-catalyzed synthetic processes.

Key words

pyrimidines - heterocycles - transition-metal catalysis - cyclization - cycloadditions - metalation - substitution

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