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Synthesis 2011(16): 2595-2599
DOI: 10.1055/s-0030-1260603
DOI: 10.1055/s-0030-1260603
SPECIALTOPIC
© Georg Thieme Verlag
Stuttgart ˙ New York
Palladium-Catalyzed Domino Heck/C-H Activation/Intermolecular Direct Arylation Reactions
Weitere Informationen
Received
8 March 2011
Publikationsdatum:
26. Mai 2011 (online)
Publikationsverlauf
Publikationsdatum:
26. Mai 2011 (online)
![](https://www.thieme-connect.de/media/synthesis/201116/lookinside/thumbnails/10.1055-s-0030-1260603-1.jpg)
Abstract
A regioselective, palladium-catalyzed domino Heck/C-H activation/intermolecular direct arylation reaction has been developed, providing rapid access to diverse biaryl heterocycles.
Key words
palladium - domino reaction - C-H activation - arylation
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