Synthesis 2014; 46(14): 1954-1956
DOI: 10.1055/s-0033-1341158
paper
© Georg Thieme Verlag Stuttgart · New York

Facile Synthesis of the Isoquinoline Alkaloids Doryanine and Oxyhydrastinine

Ravi Jangir
Division of Organic Chemistry, National Chemical Laboratory (CSIR), Pune 411 008, India   Email: np.argade@ncl.res.in
,
Smita R. Gadre
Division of Organic Chemistry, National Chemical Laboratory (CSIR), Pune 411 008, India   Email: np.argade@ncl.res.in
,
Narshinha P. Argade*
Division of Organic Chemistry, National Chemical Laboratory (CSIR), Pune 411 008, India   Email: np.argade@ncl.res.in
› Author Affiliations
Further Information

Publication History

Received: 06 February 2014

Accepted after revision: 20 March 2014

Publication Date:
10 April 2014 (online)


Abstract

Starting from 4,5-(methylenedioxy)homophthalic acid, a concise and efficient synthesis of the isoquinoline alkaloids doryanine and oxyhydrastinine is described via the corresponding homophthalimide utilizing a one-pot regioselective reductive dehydration and catalytic hydrogenation pathway.

Supporting Information

 
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