Synthesis 2016; 48(23): 4295-4299
DOI: 10.1055/s-0035-1562789
paper
© Georg Thieme Verlag Stuttgart · New York

An Improved Synthesis of Multi-Substituted Pyrazines under Catalyst- and Solvent-Free Conditions

Fatemeh Tamaddon*
Yazd University, University Blvd, Safayich, Yazd 89195-741, Iran   eMail: ftamaddon@yazd.ac.ir
,
Arefeh Dehghani Tafti
Yazd University, University Blvd, Safayich, Yazd 89195-741, Iran   eMail: ftamaddon@yazd.ac.ir
,
Farzaneh Pooramini
Yazd University, University Blvd, Safayich, Yazd 89195-741, Iran   eMail: ftamaddon@yazd.ac.ir
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Publikationsverlauf

Received: 03. Mai 2016

Accepted after revision: 27. Juni 2016

Publikationsdatum:
25. August 2016 (online)


Abstract

A one-pot pseudo four-component reaction between a variety of 2-hydroxy-1,2-diarylethanone derivatives and ammonium acetate or amines has been developed to synthesize substituted pyrazines under catalyst-free and solvent-free conditions. This procedure provides a synthetic method to access pyrazine derivatives in excellent yields under green conditions.

 
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