Synlett 2016; 27(19): 2685-2688
DOI: 10.1055/s-0036-1588300
letter
© Georg Thieme Verlag Stuttgart · New York

Synthesis of a Novel Rhizobitoxine-Like Triazole-Containing Amino Acid

Thibaut Boibessot
a   Université de Nîmes, EA7352 CHROME, Rue du Dr G. Salan, 30021 Nîmes Cedex 1, France   eMail: patrick.meffre@unimes.fr
,
David Bénimèlis
a   Université de Nîmes, EA7352 CHROME, Rue du Dr G. Salan, 30021 Nîmes Cedex 1, France   eMail: patrick.meffre@unimes.fr
,
Marion Jean
b   Aix Marseille Univ, CNRS, Centrale Marseille, iSm2, Marseille, France
,
Zohra Benfodda
a   Université de Nîmes, EA7352 CHROME, Rue du Dr G. Salan, 30021 Nîmes Cedex 1, France   eMail: patrick.meffre@unimes.fr
,
Patrick Meffre*
a   Université de Nîmes, EA7352 CHROME, Rue du Dr G. Salan, 30021 Nîmes Cedex 1, France   eMail: patrick.meffre@unimes.fr
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Publikationsverlauf

Received: 10. Juni 2016

Accepted after revision: 05. August 2016

Publikationsdatum:
18. August 2016 (online)


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Abstract

The synthesis of the four stereoisomers of a new 1,2,3-triazole analogue of rhizobitoxine from serine is described. The key step is a Huisgen 1,3-dipolar cycloaddition on an ethynylglycine synthon.

Supporting Information