Synthesis 2017; 49(18): 4372-4382
DOI: 10.1055/s-0036-1589058
paper
© Georg Thieme Verlag Stuttgart · New York

Pd/Indanone-Based Ligands: An Efficient Catalyst System for Ullmann­-Type, Suzuki–Miyaura, and Mizoroki–Heck Cross-Coupling Reactions with Aryl Tosylates and Aryl Halides

Department of Chemistry, Indian Institute of Technology Roorkee, Roorkee 247 667, India   Email: nasemfcy@iitr.ac.in
,
Naseem Ahmed*
Department of Chemistry, Indian Institute of Technology Roorkee, Roorkee 247 667, India   Email: nasemfcy@iitr.ac.in
› Author Affiliations
Further Information

Publication History

Received: 24 March 2017

Accepted after revision: 22 May 2017

Publication Date:
31 July 2017 (online)


Abstract

2-Hydroxyindan-1-ones have been efficiently synthesized and successfully applied as ligands in Pd-catalyzed Ullmann type, Suzuki–Miyaura, and Mizoroki–Heck cross-coupling reactions with aryl tosylates and aryl halides. The ligands are air- and moisture-stable and have shown high catalytic activity with Pd(OAc)2 in these cross-coupling reactions. The system tolerates a variety of functional groups in the product and can be re-used at least three times with maximum efficiency.

Supporting Information