Synthesis 1992; 1992(9): 884-887
DOI: 10.1055/s-1992-26252
paper
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Regiospecific Synthesis of Dihydropyrroles

Denis Jacoby* , Jean Pierre Celerier, Gjergi Haviari, Huguette Petit, Gérard Lhommet
  • *Laboratoire de Chimie des Hétérocycles, U.R.A. 455, Université Pierre et Marie Curie, 4 Place Jussieu, F-75252 Paris Cedex 05, France
Further Information

Publication History

Publication Date:
17 September 2002 (online)

A regiospecific synthesis of substituted dihydropyrroles is reported via nucleophilic homoallylic addition of activated cyclopropanes, followed by intramolecular ß-enamino ester formation.