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Synlett 1995; 1995(11): 1141-1142
DOI: 10.1055/s-1995-5219
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A Mild Preparation of Amino Acid N-Acylsulfonamides

Jeffrey C. Pelletier* , David P. Hesson
  • *Department of Chemistry, Symphony Pharmaceuticals, 76 Great Valley Pkwy, Malvern, PA 19355
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Publication Date:
31 December 2000 (online)

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A mild preparation of acylsulfonamide amino acids has been devised which is an improvement over existing methods. In particular, γ-substituted glutamic acid acylsulfonamide derivatives have been prepared without the competitive formation of pyroglutamates.

Aspartic Acid - Glutamic Acid - Acylsulfonamides