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Synthesis 2003(15): 2325-2330
DOI: 10.1055/s-2003-41072
DOI: 10.1055/s-2003-41072
PAPER
© Georg Thieme Verlag Stuttgart · New York
Facile Baylis-Hillman Reaction of Substituted 3-Isoxazolecarbaldehydes: The Impact of a Proximal Heteroatom Within a Heterocycle on the Acceleration of the Reaction [1]
Further Information
Received
4 July 2003
Publication Date:
23 September 2003 (online)
Publication History
Publication Date:
23 September 2003 (online)
Abstract
The fast and facile Baylis-Hillman reaction in substituted 3-isoxazolecarbaldehydes confirms the impact of the proximal heteroatom within a heterocycle towards enhanced reactivity of the formyl group for this reaction.
Key words
Baylis-Hillman reaction - aldehydes - heterocycles - isoxazoles - alkenation
CDRI Communication No. 6430.
- 2
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References
CDRI Communication No. 6430.