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Synthesis 2007(12): 1765-1767
DOI: 10.1055/s-2007-983710
DOI: 10.1055/s-2007-983710
SHORTPAPER
© Georg Thieme Verlag Stuttgart · New York
An Approach to Amino Ester Subunits of Tamiflu
Further Information
Received
30 March 2007
Publication Date:
08 June 2007 (online)
Publication History
Publication Date:
08 June 2007 (online)
Abstract
A two-step synthesis of amino cyclohexene carboxylic acid esters has been achieved in good overall yield from nitro phosphonate and unsaturated aldehydes.
Key words
Tamiflu - Michael addition - ring closure
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