Synthesis

Issue 01/2020

Periasamy, Mariappan; Venkanna, Boda; Nagaraju, Miriyala; Mohan, Lakavathu: Methods for the Synthesis of Piperazine Derivatives Containing a Chiral Bi-2-naphthyl Moiety

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Issue 03/2021

Pharande, Shrikant G.: Synthesis of Lactams via Isocyanide-Based Multicomponent Reactions

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Issue 03/2020

Karmakar, Ananta; Ramalingam, Sridharan; Basha, Mushkin; Indasi, Gopi Kumar; Belema, Makonen; Meanwell, Nicholas A.; Dhar, T. G. Murali; Rampulla, Richard; Mathur, Arvind; Gupta, Anuradha; Gupta, Arun Kumar: Facile Access to 1,4-Disubstituted Pyrrolo[1,2-a]pyrazines from α-Aminoacetonitriles

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Issue 03/2021

Dibdalli, Yuvaraja; Faúndez, Rodrigo; Preite, Marcelo; Molins, Elies; Chávez, Ivonne; Amshumali, Mungalimane K.; Morales-Verdejo, Cesar; Manriquez, Juan M.: An Improved Synthesis of 3,6-Dihydro-as-indacene

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Issue 04/2020

Mittal, Rupali; Mishra, Anupam; Awasthi, Satish K.: A Greener Approach for the Chemoselective Boc Protection of Amines Using Sulfonated Reduced Graphene Oxide as a Catalyst in Metal- and Solvent-Free Conditions

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Issue 05/2020

Tripathi, Krishna N.; Bansode, Avinash H.; Singh, Ravi P.: Palladium-Catalyzed Oxidative Annulation of Pyrrolylalkyl-1H-azoles: Towards the Synthesis of Polyheterocyclic Arenes

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Reddy, Julakanti Satyanarayana; Gangababu, Marri; Manimala, Patel; Rammohan, Aluru; Yadav, Jillu Singh: Studies towards the Total Synthesis of Kadcotrione B

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Issue 05/2021

Vijayan, Ajesh; Rao, Desaboini Nageswara; Radhakrishnan, K. V.; Lam, Patrick Y. S.; Das, Parthasarathi: Advances in Carbon–Element Bond Construction under Chan–Lam Cross-Coupling Conditions: A Second Decade

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Issue 06/2021

Raji Reddy, Chada; Bodasu, Srinivas; Mallesh, Kathe; Prapurna, Y. Lakshmi: Synthesis of Fused Pyrimido[1,6-a]indolones via Rhodium(III)-Catalyzed Cascade Annulations

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Issue 09/2020

Devi, Ngangbam Renubala; Shit, Sudip; Behera, Bipin Kumar; Saikia, Anil K.: Synthesis of 4-Vinyl-1,2,3,4-tetrahydroisoquinoline from N-Tethered Benzyl-Alkenol Catalyzed by Indium(III) Chloride: Formal Synthesis of (±)-Isocyclocelabenzine

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Kiran, Kuppalli R.; Swaroop, Toreshettahally R.; Rajeev, Narasimhamurthy; Anil, Seegehalli M.; Rangappa, Kanchugarakoppal S.; Sadashiva, Maralinganadoddi P.: Cyclization of Active Methylene Isocyanides with α-Oxodithioesters Induced by Base: An Expedient Synthesis of 4-Methylthio/Ethoxycarbonyl-5-acylthiazoles

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Issue 10/2020

Gucchait, Arin; Ghosh, Sritin; Misra, Anup Kumar: Synthesis of Novel Glycosyl Carbamo(dithioperoxo)thioate Derivatives

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Issue 08/2021

Chaubey, Narendra R.; Kapdi, Anant R.; Maity, Biswanath: Organophotoredox-Catalyzed C–H Alkylation of Imidazoheterocycles with Malonates: Total Synthesis of Zolpidem

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Issue 09/2021

Singh, Pushpinder; Batra, Aanchal; Singh, Kamal Nain; Mritunjay, Mritunjay: Transition-Metal-Free Strategies for the Synthesis of C-1 Aryl-Substituted Tetrahydroisoquinolines

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Issue 10/2020

Hussain, Mulla Althafh; Khan, Faiz Ahmed: Total Synthesis of (±)-Cassumunins A–C and Curcumin Analogues

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Issue 11/2020

Keerthana, Meledath Sudhakaran; Manoharan, Ramasamy; Jeganmohan, Masilamani: Cobalt(III)-Catalyzed Redox-Neutral Coupling of Acrylamides with Activated Alkenes via C–H Bond Activation

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Issue 13/2020

Teixeira, Wystan K. O.; de Albuquerque, Danilo Yano; Narayanaperumal, Senthil; Schwab, Ricardo S.: Recent Advances in the Synthesis of Enantiomerically Enriched Diaryl, Aryl Heteroaryl, and Diheteroaryl Alcohols through Addition of Organometallic Reagents to Carbonyl Compounds

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Issue 11/2021

Gairola, Deepti; Peddinti, Rama Krishna: Methanesulfonic Acid Catalyzed Friedel–Crafts Reaction of Electron-Rich Arenes with N-Arylmaleimides: A Highly Efficient Metal-Free Route To Access 3-Arylsuccinimides

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Kotha, Sambasivarao; Pulletikurti, Sunil; Fatma, Ambareen; Dhangar, Gopal; Naidu, Gonna Somu: Synthesis of Polycycles and Oxacycles via Tandem Metathesis of endo-Norbornene Derivatives

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Issue 14/2020

Sharathna, Puthiyaparambath; Meenu, Murugan Thulasi; Dhanya, Bhandara Purayil; Gopalan, Greeshma; Sasikumar, Parameswaran; Krishnan, Radhakrishnan Syam; Radhakrishnan, Kokkuvayil Vasu: Accessing Polycyclic Terpenoids from Zerumbone via Lewis Acid Catalyzed Synthetic Strategies

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Issue 12/2021

Schefzig, Luise; Kurzawa, Timon; Rancan, Giaime; Linder, Igor; Leisering, Stefan; Bera, Mrinal K.; Gart, Max; Zimmer, Reinhold; Reissig, Hans-Ulrich: Access to Highly Substituted Pyrimidine N-Oxides and 4-Acetoxymethyl-Substituted Pyrimidines via the LANCA Three-Component Reaction–Cyclocondensation Sequence

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Issue 13/2021

Hsu, Ming-Hua; Kapoor, Mohit; Pradhan, Tapan Kumar; Tse, Man-Him; Chen, Hsin-Ya; Yan, Man-Jun; Cheng, Yu-Tsen; Lin, Yu-Cheng; Hsieh, Cheng-Ying; Liu, Ker-Yin; Han, Chien-Chung: Mild and Efficient Copper-Catalyzed Synthesis of Trisubstituted Pyrroles

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Issue 15/2020

R., Chandran; Tiwari, Keshri Nath: Krapcho Dealkoxycarbonylation Strategy of Ethyl Cyanoacetate for the Synthesis of 3-Hydroxy-3-cyanomethyl-2-oxindoles and 3,3′-Dicyanomethyl-2-oxindoles in a Reaction with Isatin

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Issue 13/2021

Pramanik, Sayan; Ray, Suman; Maity, Suvendu; Ghosh, Prasanta; Mukhopadhyay, Chhanda: Diastereoselective trans Cyclopropanation of 3-Alkylidene Oxindoles with In Situ Generated α-Diazo Carbonyls or α,β-Unsaturated Diazo Compounds

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Issue 15/2020

Kumari, Anupama; Fernandes, Rodney A.: BX₃-Mediated Intermolecular Formation of Functionalized 3-Halo-1H-indenes via Cascade Halo-Nazarov-Type Cyclization

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Issue 13/2021

Yadav, Mamta; Jat, Ram Singh; Sarma, Bibek; Bhanuchandra, M.: 2-Pyridyl Sulfoxide Directed Pd(II)-Catalyzed C–H Olefination of Arenes with Molecular Oxygen as the Sole Oxidant

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Saravanan, Velu; Mohanakrishnan, Arasambattu K.: Synthesis of Annulated Carbazoles via FeCl₃/SnCl₄‑Mediated Domino Reaction of Vinyl Ketone Tethered Bromomethylindoles with Arenes and Heteroarenes

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Issue 14/2021

Yadav, Mangal S.; Singh, Sumt K.; Agrahari, Anand K.; Singh, Anoop S.; Tiwari, Vinod K.: N-Acylbenzotriazoles as Proficient Substrates for an Easy Access to Ureas, Acylureas, Carbamates, and Thiocarbamates via Curtius Rearrangement Using Diphenylphosphoryl Azide (DPPA) as Azide Donor

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Issue 17/2020

Rao, V. U. Bhaskara; Singh, Shashank; Tripathi, Krishna N.; Singh, Ravi P.: Stereoselective Synthesis of Spiro-α-methylene-γ-lactams via Chiral Quaternary 3-Aminooxindole Adducts Accessed by Zn-Mediated Allylation of Sulfinyl Ketimines

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Issue 15/2021

Inani, Heena; Singh, Avtar; Bhati, Meeta; Kumari, Kiran; Kucherenko, Alexander S.; Zlotin, Sergei G.; Easwar, Srinivasan: Proline-Histidine Dipeptide: A Suitable Template for Generating Ion-Tagged Organocatalysts for the Asymmetric Aldol Reaction

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Issue 16/2021

Kumari, Arram Haritha; Kumar, Jangam Jagadesh; Krishna, Gamidi Rama; Reddy, Raju Jannapu: Nickel-Catalyzed Difunctionalization of Alkynyl Bromides with Thiosulfonates and N-Arylthio Succinimides: A Convenient Synthesis of 1,2-Thiosulfonylethenes and 1,1-Dithioethenes

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Mandadapu, Raghuramaiah; Dehade, Amol Satish; Shete, Shrikant Abhiman; Montgomery, Mark; Sikervar, Vikas; Sonawane, Ravindra: Lewis Acid Mediated [3+2] and [3+3] Annulations of an Azomethine Imine with Donor–Acceptor Cyclopropanes

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Issue 19/2020

Patil, Mahendra: Mechanism of the t-BuOM (M = K, Na, Li)/DMEDA-Mediated Direct C–H Arylation of Benzene: A Computational Study

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Issue 16/2021

Shelar, Santosh V.; Argade, Narshinha P.: Wittig Reactions of Maleimide-Derived Stabilized Ylides with Alkyl Pyruvates: Concise Approach to Methyl Ester of (±)-Chaetogline A

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Senapati, Sibadatta; Unmesh, Nivedya A.; Shet, Manoj N.; Ahmad, Iram; Ajikumar, Nandu; Ramana, Chepuri V.: Unified Approach for the Total Synthesis of Bis-THF C₁₅ Acetogenins: A Chloroenyne from Laurencia majuscula, Laurendecumenyne B and Laurefurenynes A/B

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Issue 17/2021

Vijaykumar, Muniyappa; Punji, Benudhar: Advances in Transition-Metal-Catalyzed C–H Bond Oxygenation of Amides

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Issue 18/2021

Basak, Sumon; Biswas, Jyoti Prasad; Maiti, Debabrata: Transition-Metal-Catalyzed C–H Arylation Using Organoboron Reagents

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Issue 21/2020

Kadari, Lingaswamy; Roisnel, Thierry; Erb, William; Krishna, Palakodety Radha; Mongin, Florence: Remote Deprotometalation-Iodolysis of N,N-Diisopropyl-2-trimethylsilylferrocenecarboxamide: A New Route Toward 1,1′-Disubstituted Ferrocenes

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Issue 18/2021

Sihag, Pinki; Jeganmohan, Masilamani: Recent Advances in Transition-Metal-Catalyzed C–H Functionalization Reactions Involving Aza/Oxabicyclic Alkenes

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Issue 21/2020

Verma, Saumya; Kumar, Puneet; Khatana, Anil K.; Chandra, Dinesh; Yadav, Ajay K.; Tiwari, Bhoopendra; Jat, Jawahar L.: Zinc(II)-Catalyzed Synthesis of Secondary Amides from Ketones via Beckmann Rearrangement Using Hydroxylamine-O-sulfonic Acid in Aqueous Media

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Issue 18/2021

Dalal, Arup; Babu, Srinivasarao Arulananda: Pd(II)-Catalyzed Directing-Group-Aided C–H Arylation and Alkylation of Pyrene Core: Synthesis of C1,C2- and C1,C10-Disubstituted Pyrene Motifs

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Hassan, Mirja Md Mahamudul; Hoque, Md Emdadul; Dey, Sayan; Guria, Saikat; Roy, Brindaban; Chattopadhyay, Buddhadeb: Iridium-Catalyzed Site-Selective Borylation of 8-Arylquinolines

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Issue 19/2021

Tadiparthi, Krishnaji; Anand, Pragya: A Review on Synthetic Approaches towards Kavalactones

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Issue 22/2020

Chavan, Subhash P.; Pawar, Ambaji A.; Patil, Niteen B.; Kadam, Appasaheb L.; Shinde, Shrikrishna S.: Scalable Synthesis of 3-Ethyl-4-methyl-1,5-dihydro-2H-pyrrol-2-one: An Important Building Block of the Antidiabetic Drug Glimepiride

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Issue 23/2020

Khandelwal, Manisha; Ray, Sumit Kumar; Khangarot, Rama Kanwar: Syntheses and Applications of Singh’s Catalyst

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Bhilare, Shatrughn; Kori, Santosh; Shet, Harshita; Balaram, Gundapally; Mahendar, Koosam; Sanghvi, Yogesh S.; Kapdi, Anant R.: Scale-Up of a Heck Alkenylation Reaction: Application to the Synthesis of an Amino-Modifier Nucleoside ‘Ruth Linker’

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Issue 19/2021

Gucchait, Arin; Kundu, Monalisa; Misra, Anup Kumar: Synthesis of Pentasaccharide Repeating Unit Corresponding to the Cell Wall O-Polysaccharide of Salmonella enterica O55 Strain Containing a Rare Sugar 3-Acetamido-3-deoxy-d-fucose

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Issue 24/2020

Talukdar, Ranadeep: Synthetically Important Ring-Opening Acylations of Alkoxybenzenes

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Yu, Jie; Singh, Anoop S.; Yan, Guobing; Yu, Jian; Tiwari, Vinod K.: Recent Developments on Denitrogenative Functionalization of Benzotriazoles

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Issue 21/2021

Dhiman, Ankit Kumar; Kumar, Rohit; Sharma, Upendra: Catalyst- and Additive-Free Synthesis of Fluoroalkoxyquinolines

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