Synthesis

Issue 01/2024

Takebe, Hiyori; Matsubara, Seijiro: Decoration on Cubane with an Awareness of Chirality: Development of Substituted Cubane Syntheses

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Bera, Satabdi; Jana, Subhenira; Samanta, Rajarshi: Recent Progress on Copper-Catalyzed C–C Bond Formation via C(sp²)–H Insertions Using Diazo and Related Compounds

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Issue 02/2024

Hattori, Hiroyuki; Ishida, Kento; Sakai, Norio: Synthetic Strategies for Accessing Dibenzophosphole Scaffolds

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Saito, Fumito: Recent Developments on the Synthesis of Sulfoxides via Sulfenate Anions

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Morrison, Kathleen M.; Stradiotto, Mark: Advances in Nickel-Catalyzed O-Arylation of Aliphatic Alcohols and Phenols with (Hetero)aryl Electrophiles

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Issue 02/2025

Kotha, Sambasivarao; Khedkar, Priti: Design of Synthetic Strategies towards Sulfur Containing Scaffolds

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Kant, Kamal; Naik, Priyadarshini; Patel, Chandresh Kumar; Some, Sanjukta; Banerjee, Sourav; Aljaar, Nayyef; Atta, Ananta K.; Malakar, Chandi C.: Organocatalytic Approaches Towards the Synthesis of Asymmetric Tetrahydroquinoline (THQ) Derivatives

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Knieb, Alexander; Prakash, G. K. Surya: Recent Advances in Fluoroalkylation Strategies: Exploring Novel Reactivities and Synthetic Applications of Sulfone- and Sulfinate-Based Reagents for Mono-, Di-, and Trifluoromethylations

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Issue 03/2024

Jeanmart, Stephane; Edmunds, Andrew J. F.; Lamberth, Clemens; Pouliot, Martin; Morris, James A.: Synthetic Approaches to the 2019–2020 New Agrochemicals

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Issue 02/2025

Pandit, Soumen; Majumdar, Nilanjana: Catalytic Intermolecular [4+2]-Cycloaddition toward the Stereo­selective C2–C3 Annulation of Indoles

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Issue 03/2024

Yang, Liangliang; Wang, Haiyang; Lang, Ming; Peng, Shiyong: Recent Advances on High-Order Dipolar Annulations of Donor–Acceptor Cyclopropanes/Cyclobutanes

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Issue 03/2025

Zheng, Cameron H. M.; Schafer, Laurel L.: Recent Advances in Saturated N-Heterocycle C–H Bond Functionalization for Alkylated N-Heterocycle Synthesis

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Li, Fei; Song, Jia-Wei; Han, Xue; Zhang, Cheng-Pan: Progress in Photocatalyzed Trifluoromethylthiolation and Trifluoromethylselenolation Reactions

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Issue 05/2024

Komijani, Samira; Orellana, Arturo: The Electrocyclization of Heptatrienyl Anions

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Issue 04/2025

Martos, Mario; Bosque, Irene; Gonzalez-Gomez, Jose C.: Advances in Photoinduced Minisci-like Reactions

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Issue 05/2024

Van Hoof, Max; Force, Guillaume; Lebœuf, David: Modern Macrolactonization Techniques

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Li, Tao; Chan, Albert S. C.; Meng, Shan-Shui: Direct Reductive Coupling of Nitro Compounds for the Synthesis of Advanced Amines

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Issue 06/2024

Arora, Aditi; Kumar, Sumit; Khatri, Vinod; Prasad, Ashok K.; Chhatwal, Rajni Johar; Kumar, Sandeep: Recent Advances in the Synthesis and Application of C-2-Formyl Glycals

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Issue 05/2025

Sajjad, Farrukh; Zhang, Shuyue; Xu, Ming-Hua: Advances in Transition-Metal Catalysis and Organocatalysis Approaches towards Asymmetric Synthesis of β-Amino Acid Derivatives

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Horwitz, Matthew A.: Discovery Process Chemistry: An Innovation Hub at the Interface of Academia, the Pharmaceutical Industry, and Contract Research Organizations

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Issue 07/2024

Das, Ramanand; Das, Malati; Mukherjee, Debaraj; Kundu, Taraknath: Recent Advances on the Synthesis of C-Glycosides from 1,2-Glycals

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Kumar, Sumit; Khan, Yousuf; Arora, Aditi; Kumar, Manish; Rungta, Pallavi; Singh, Brajendra K.; Sharma, Vivek K.; Singh, Sunil K.: Advances in the Synthesis of Spirocyclic Nucleosides

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Issue 06/2025

Gerlach, Tabea; Turner, Nicholas J.: Biocatalytic Dearomatisation Reactions

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Miguélez, Rubén; Arto, Omar; Rodríguez-Arias, Carlos; Barrio, Pablo: Gold(I)-Catalyzed Intramolecular C(sp3)–H Bond Functionalization

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Issue 08/2024

Mamedov, Vakhid A.; Zhukova, Nataliya A.: Recent Advances in the Synthesis of Indoles with Partially Hydrogenated Benzene Ring (Tetrahydroindoles)

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Zhao, Xian; Liu, Wei: Recent Advances in Transition-Metal-Catalyzed Sonogashira Cross-Coupling Reactions of Alkyl Electrophiles

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Issue 07/2025

Li, Xiang; Tu, Yong-Liang; Chen, Xiang-Yu: Recent Advances in Combining Photo- and N-Heterocycle Nitrenium Catalysis

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Issue 08/2024

Wang, Zi-Lu; Xu, Yun-He: Progress on the Enantioselective Synthesis of Axially Chiral Cycloalkylidenes

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Issue 09/2024

Ito, Hideto; Kawahara, Kou P.; Itami, Kenichiro: Heteroatom-Embedding Annulative π-Extension (Hetero-APEX) Reactions: An Overview

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Li, Mengran; Chen, Peng; Liu, Haoqi; Huang, Jian; Chen, Yang: Review of the Total Synthesis of the Aromatic Abietane Diterpenoid Ferruginol

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Bellemin-Laponnaz, Stéphane; Achard, Thierry: Recent Progress in Developing Thioether-Containing Ligands for Catalysis Applications

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Issue 08/2025

Burianova, Valeria K.; McErlain, Holly; Sutherland, Andrew: Transition-Metal-Mediated Radiohalogenation using Aryl Boron Reagents

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Takebe, Hiyori; Matsubara, Seijiro: Cuneanes as Potential Benzene Bioisosteres Having Chirality

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Issue 10/2024

Kang, Eunsu; Joo, Jung Min: Pyrazolopyridine Ligands in Transition-Metal-Catalyzed C–C and C–Heteroatom Bond-Forming Reactions

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Issue 11/2024

Xu, Wei; Kumagai, Naoya: Recent Advances in Quinoline-Based Macrocycles: Synthesis, Properties, and Applications in Catalytic Reactions

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Hussain, Waseem A.; Parasram, Marvin: Recent Advances in Photoinduced Oxidative Cleavage of Alkenes

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Issue 12/2024

Gope, Biplab; Mishra, Anupam; Awasthi, Satish K.: Rhodium(III)-Catalyzed C–H Activation in Indole: A Comprehensive Report (2017–2022)

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Croll, Elizabeth A.; Kwon, Ohyun: Mechanism of the Mitsunobu Reaction: An Ongoing Mystery

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Zou, Jia-Yu; Xu, Wan-Yi; Wang, Jie; Liu, Qi; He, Ying: Atroposelective Construction of Tetrasubstituted Axially Chiral Alkene Frameworks

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Issue 13/2024

Li, Xin; Song, Qiuling: Recent Progress on the Zweifel Olefination: An Update

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Issue 14/2024

Maheshwari, Mittali; Hussain, Nazar: Chemical Synthesis of Substituted Naphthalene Derivatives: A Review

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Dai, Peng-Fei; Li, Qiang-Qiang; Qu, Jian-Ping; Kang, Yan-Biao: Recent Developments on the Earth-Abundant-Metal-Catalyzed α,β-Dehydrogenation of Carbonyl Compounds

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Healy, Alan R.: Stereodivergent Carbon–Carbon Bond-Forming Reactions

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Issue 16/2024

Javahershenas, Ramin; Mei, Haibo; Koley, Manankar; Soloshonok, Vadim A.; Makarem, Ata: Recent Advances in the Multicomponent Synthesis of Heterocycles Using 5-Aminotetrazole

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Issue 21/2024

Sumino, Shuhei; Ryu, Ilhyong; Robert, Frédéric; Landais, Yannick: 1,2-Bis(phenylsulfonyl)ethylene (BPSE): A Potent Radical C2 Synthon Available in the Radical and Electron-Transfer-Based Organic Synthesis

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Issue 22/2024

Sakuraba, Mahiro; Hoshimoto, Yoichi: Recent Trends in Triarylborane Chemistry: Diversification of Structures and Reactivity via meta-Substitution of the Aryl Groups

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Issue 23/2024

Khorasani, Fereshteh; Ranjbar-Karimi, Reza; Marra, Alberto: Recent Advances in the Synthesis and Applications of Ionic Liquids Derived from Natural Products

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Sen, Abhijit; Yamada, Yoichi M. A.: Latest Developments on Palladium- and Nickel-Catalyzed Cross-Couplings Using Aryl Chlorides: Suzuki–Miyaura and Buchwald–Hartwig Reactions

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Issue 24/2024

Ullah, Saif; Hussain, Zulfiqar; Peng, Yungui: Recent Advances in Diazophosphonate Chemistry: Reactions and Transformations

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Bernardo, Olaya; García-Martínez, Patricia; Santamaría, Javier; López, Luis A.: Recent Advances in Gold-Catalyzed Transformations of Vinyldiazo Reagents

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Issue eFirst

Li, Heyin; Wang, Yi: Progress in Radical Fluorosulfonyl Reagents

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Chen, Xu; Zhou, Xuesi; He, Jiawei; Liu, Xiang: Recent Advances in Photoinduced Borylation via N-Heterocyclic Carbene Boryl Radicals

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Issue 03/2024

Singh, Sanjay; Hazra, Chinmoy K.: Recent Advancements in Typical Friedel–Crafts Alkylation Reactions Focused on Targeting Arene Nucleophiles

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Issue 01/2024

Kang, Taeho; Apolinar, Omar; Engle, Keary M.: Ni- and Pd-Catalyzed Enantioselective 1,2-Dicarbofunctionalization of Alkenes

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Issue 18/2023

Wang, Qian; Liu, Han-Fu; Ren, Sai-Yan; He, Mu-Xue; Pan, Ying-Ming: Research Advances in Electrochemical Synthesis of Spirocyclic Skeleton Compounds

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