Synthesis, Table of Contents PAPER © Georg Thieme Verlag Stuttgart · New York New Synthetic Route to 2-(Diethylphosphono)-2H-Azirines Valery K. Brel*Institute of Physiologically Active Compounds of Russian Academy of Science, Chernogolovka, Moscow region, 142432, RussiaFax: +7(95)7857024; e-Mail: brel@ipac.ac.ru; Recommend Article Abstract Buy Article All articles of this category Abstract Synthesis of new 2-substituted-2-(diethylphosphono)-3-isopropenyl-2H-azirines is described by aconvenient and efficient procedure starting from phosphorylated allenes. Key words cyclizations - azides - allenes - phosphorus - heterocycles. Full Text References References 1a Pearson WH. Lian BW. Bergmeier SC. Padwa A. Comprehensive Heterocyclic Chemistry II Pergamon Press; Oxford: 1996. Chap. 1. 1b Backes J. In Methoden der Organische Chemie (Houben-Weyl) Vol. E16c: Klamann D. Thieme; Stuttgart: 1992. p.317 1c Heimgartner H. Angew. Chem., Int. Ed. Engl. 1991, 30: 238 2a Pinho e Melo TMVD. Lopes CSJ. Rocha Gonsalves AMd’A. Beja AM. Paixão JA. Silva MR. Alte da Veiga L. J. Org. Chem. 2002, 67: 66 2b Palacios F. Ochoa de Retana AM. Gil JI. Ezpeleta JM. J. Org. Chem. 2000, 65: 3213 3 Bucher CB. Heimgartner H. Helv. Chim. Acta. 1996, 79: 1903 4 Russell GA. Yao CF. J. Org. Chem. 1992, 57: 6508 5 Pinho e Melo TMVD. Lopes CSJ. Rocha Gonsalves AMd’A. Storr RC. Synthesis 2002, 605 6 Drögemüller M. Jautelat R. Winterfeldt E. Angew. Chem., Int. Ed. Engl. 1996, 35: 1572 7a Davis FA. Wu Y. Yan H. Prasad KR. McCoull W. Org. Lett. 2002, 4: 655 7b Davis FA. McCoull W. Tetrahedron Lett. 1999, 40: 249 8 Alabugin IV. Brel VK. Usp. Khim. 1997, 66: 225 ; Chem. Abstr. 1998, 128, 114977r 9 Brel VK. Synthesis 1999, 463 10 Brel VK. Synthesis 2001, 1539 11 Mark V. In Mechanism of Molecular Migrations Vol. 3: Thyagajaran BS. Wiley; New York: 1969. p.320 12 Perrin DD. Armarego WLF. Perin DR. Purification of Laboratory Chemicals Pergamon Press Ltd; New York: 1980. 13 Brandsma L. Preparative Acetylenic Chemistry Elsevier; Amsterdam: 1988. p.265 14 Brel VK. Synth. Commun. 1999, 29: 3869