DOI: 10.1055/s-00000083

Synlett

Issue 02 · Volume 37 · January 2026 DOI: 10.1055/s-015-62798

Table of Contents

  • V

    Table of Contents

    • Synpacts

  • 141
    Liu, Chang; Zhang, Mingyu; Dai, Mingji:

    Total Synthesis of (±)-Phaeocaulisin A Enabled Chemistry Innovation and Biological Discovery

    Image for article: Total Synthesis of (±)-Phaeocaulisin A Enabled Chemistry Innovation and Biological Discovery
  • 145
    Ban, Xu; Jiang, Zhiyong:

    Boron-Migration-Mediated Photochemical Enantioselective Protonation/Deuteration via Chiral Hydrogen-Bonding Catalysis

    Image for article: Boron-Migration-Mediated Photochemical Enantioselective Protonation/Deuteration via Chiral Hydrogen-Bonding Catalysis
  • 151
    Wang, Yi-Bo; Xin, Nie; Long, Li:

    New Advances in Atroposelective Synthesis of Axial Chirality via Asymmetric Gold(I)-Catalyzed Annulation of Diazo-Alkynes

    Image for article: New Advances in Atroposelective Synthesis of Axial Chirality via Asymmetric Gold(I)-Catalyzed Annulation of Diazo-Alkynes
  • 155
    Wang, Zi-Chao; Wang, Peng; Shi, Shi-Liang:

    Ni-Catalyzed Addition of Arylborons to Alkenes for the Synthesis of Quaternary Carbon Centers

    Image for article: Ni-Catalyzed Addition of Arylborons to Alkenes for the Synthesis of Quaternary Carbon Centers

    • Account

  • 160
    Dhayalan, Vasudevan:

    Recent Advances in Strain-Release Functionalization of [1.1.1]Propellanes Using Organometallic Reagents

    Image for article: Recent Advances in Strain-Release Functionalization of [1.1.1]Propellanes Using Organometallic Reagents
  • 167
    Garg, Sneha; Kumar, Ankush; Yash; Chaubey, Suruchi; Harnoor; Kumari, Pratima; Bhatia, Rohit; Singh, Ravinder:

    Recent Development of Metallopharmaceuticals in Cancer Therapy: Ruthenium Complexes and Their Analogues

    Image for article: Recent Development of Metallopharmaceuticals in Cancer Therapy: Ruthenium Complexes and Their Analogues

    • Published as part of the Cluster Alkynes in Organic Synthesis

  • 183
    Große, Michel; Wegner, Hermann A.:

    Cyclooctynes as Building Blocks for the Synthesis of Arene-Annulated Eight-Membered Ring Systems

    Image for article: Cyclooctynes as Building Blocks for the Synthesis of Arene-Annulated Eight-Membered Ring Systems

    • Published as part of the Special Issue dedicated to Prof. S. Chandrasekaran on his 80th birthday

  • 191
    Kotha, Sambasivarao; Solanke, Balaji U.:

    Diversity-Oriented Approach to Furan Building Blocks and Their Relevance in Organic Synthesis, Materials Science, and Medicinal Chemistry

    Image for article: Diversity-Oriented Approach to Furan Building Blocks and Their Relevance in Organic Synthesis, Materials Science, and Medicinal Chemistry

    • New Tools

  • 208
    Wang, Fei; Wu, Yadong; Yang, Shiwei:

    Research on the Synthetic Methodology for Lurasidone Hydrochloride

    Image for article: Research on the Synthetic Methodology for Lurasidone Hydrochloride
    Supplementary Material (PDF)

    • Letter

  • 212
    Ghosh, Sumit; Ghosh, Asim Kumar; Mahato, Frenki; Taher, Abu; Sinha, Subrata; Hajra, Alakananda:

    Visible-Light-Induced Ru-Catalyzed Ortho C−H Diarylation of 2-Phenyl-2H-Indazoles and 1-Phenyl-1H-Pyrazoles

    Image for article: Visible-Light-Induced Ru-Catalyzed <i>Ortho</i> C−H Diarylation of 2-Phenyl-2<i>H</i>-Indazoles and 1-Phenyl-1<i>H</i>-Pyrazoles
    Supplementary Material (PDF)
  • 217
    Kumar, Mahesh; Sharma, Anup Kumar; Kishor, Kaushal; Singh, Krishna Nand:

    A Catalyst-Free Transamination of (E)-N,N-Dimethyl Enaminones to β-Amino-α,β-Unsaturated Carbonyl Compounds by Using Isothiocyanates as Amines Proxy

    Image for article: A Catalyst-Free Transamination of (<i>E</i>)-<i>N,N</i>-Dimethyl Enaminones to β-Amino-α<i>,</i>β-Unsaturated Carbonyl Compounds by Using Isothiocyanates as Amines Proxy
    Supplementary Material (PDF)
  • 221
    Liu, Han; Yang, Zhiyong; Yan, Jiaqi; Guo, Jing:

    Photoinduced and N-Bromosuccinimide-Initiated Esterification of Aromatic acids and Terminal Alkynes with Alcohols

    Image for article: Photoinduced and <i>N</i>-Bromosuccinimide-Initiated Esterification of Aromatic acids and Terminal Alkynes with Alcohols
    Supplementary Material (PDF)

    • Published as part of the Special Issue dedicated to Prof. S. Chandrasekaran on his 80th birthday

  • 225
    Pandavadara, Atul R.; Khanvilkar, Aditya N.; Bedekar, Ashutosh V.; Butcher, Raymond; Abraham, Alex:

    Applications of Optically Pure Biphenyloxycyclohexanols in Deracemization of α-Substituted Aryloxypropanoic Acids by Dynamic Kinetic Resolution

    Image for article: Applications of Optically Pure Biphenyloxycyclohexanols in Deracemization of α-Substituted Aryloxypropanoic Acids by Dynamic Kinetic Resolution

    • Published as part of the Special Topic Alkynes in Organic Synthesis

  • 232
    Kies, Wolfgang; Misselwitz, Erik; Borstelmann, Jan; Berger, Georg; Rominger, Frank; Kivala, Milan:

    Synthesis and Chiroptical Characterization of a Negatively Curved Helicene with a Central Tropone Unit

    Image for article: Synthesis and Chiroptical Characterization of a Negatively Curved Helicene with a Central Tropone Unit
    Supplementary Material (PDF)
  • 237
    Yuan, Xinxin; Zeng, Qian-Ding; Yao, Hongmiao; Jin, Wenjun; Ren, Jiangmeng; Zeng, Bu-Bing:

    Rapid Deprotection of O-Allyoxycarbonyl(alloc) Alcohols by NiCl2•6H2O and NaBH4

    Image for article: Rapid Deprotection of <i>O</i>-Allyoxycarbonyl(alloc) Alcohols by NiCl<sub>2</sub>•6H<sub>2</sub>O and NaBH<sub>4</sub>
    Supplementary Material (PDF)

    • Published as part of the Special Topic Alkynes in Organic Synthesis

  • 241
    Liu, Zhi-Chao; Wang, Tao; Yang, Shengchao; Zhou, Jian; Yu, Jin-Sheng:

    A Tandem Aldol/Desilylation/CuAAC Sequence of Difluoroenoxysilanes and Silyl-α-ketoalkynes to α-Fluoroketone α-1,2,3 Triazole Tertiary Alcohol

    Image for article: A Tandem Aldol/Desilylation/CuAAC Sequence of Difluoroenoxysilanes and Silyl-α-ketoalkynes to α-Fluoroketone α-1,2,3 Triazole Tertiary Alcohol
    Supplementary Material (PDF)

    • Published as part of the Special Issue dedicated to Prof. S. Chandrasekaran on his 80th birthday

  • 246
    Choudhuri, Tathagata; Sikdar, Papiya; Paul, Suvam; Das, Sourav; Bagdi, Avik Kumar:

    I2-Catalyzed Access to Bis(pyrazolo[1,5-a]pyrimidinyl)sulfanes and Sulfenylated Pyrazolo[1,5-a]pyrimidines via C–H Functionalization

    Image for article: I<sub>2</sub>-Catalyzed Access to Bis(pyrazolo[1,5-<i>a</i>]pyrimidinyl)sulfanes and Sulfenylated Pyrazolo[1,5-<i>a</i>]pyrimidines via C–H Functionalization
    Supplementary Material (PDF)
  • 251
    Chatragadda, Kranthi; Nagarajan, Rajagopal:

    Facile Synthesis of 11H-Indolo[3,2-c]quinolines Through Pictet–Spengler Cyclization and Aromatization by Oxygen

    Image for article: Facile Synthesis of 11<i>H</i>-Indolo[3,2-<i>c</i>]quinolines Through Pictet–Spengler Cyclization and Aromatization by Oxygen
    Supplementary Material (PDF)
  • 255
    Wang, Hai-Yang; Liu, Fu-Sheng:

    Three-Component Reaction of N-(Sulfonyl)acrylamides, Tert-Butyl nitrite, and Acetone: Preparation of Isoxazole Compounds

    Image for article: Three-Component Reaction of <i>N</i>-(Sulfonyl)acrylamides, <i>Tert</i>-Butyl nitrite, and Acetone: Preparation of Isoxazole Compounds
    Supplementary Material (PDF) Supplementary Material (PDF)
  • 265
    Ando, Sosuke; Anada, Masahiro; Sueki, Shunsuke; Makino, Kosho; Kawasaki-Takasuka, Tomoko; Mori, Keiji:

    Intramolecular Hydride Shift-Mediated Double C(sp3)–H Bond Functionalization of Conformationally Flexible Aliphatic Alkenylidene Malonates

    Image for article: Intramolecular Hydride Shift-Mediated Double C(sp<sup>3</sup>)–H Bond Functionalization of Conformationally Flexible Aliphatic Alkenylidene Malonates
    Supplementary Material (PDF)
  • 269
    Shi, Houguang; Song, Yanhong; Gong, Hegui:

    Facile Preparation of Chiral 1,2-Amino Alcohols Containing Unsymmetrical N-α-Secondary Alkyl Substituents

    Image for article: Facile Preparation of Chiral 1,2-Amino Alcohols Containing Unsymmetrical <i>N</i>-α-Secondary Alkyl Substituents
  • 275
    Patel, Shweta A.:

    ADME-Based Drug Development of 2H-Pyran Derivatives with Enhanced Antimicrobial Efficacy

    Image for article: ADME-Based Drug Development of 2<i>H</i>-Pyran Derivatives with Enhanced Antimicrobial Efficacy