Studies on the Synthesis of the 1-Hydroxynortropane System; Part II.1 Synthesis of Calystegine A3 and Physoperuvine

François-Didier Boyer; Paul-Henri Ducrot; Vivien Henryon; Josette Soulié; Jean-Yves Lallemand

doi:10.1055/s-1992-22014

RSS-Feed abonnieren

Bitte kopieren Sie die angezeigte URL und fügen sie dann in Ihren RSS-Reader ein.

https://www.thieme-connect.de/rss/thieme/de/10.1055-s-00000083.xml

Teilen / Bookmarken

Facebook X Linkedin Weibo

PDF herunterladen

Synlett 1992; 1992(4): 357-359
DOI: 10.1055/s-1992-22014

letter

© Georg Thieme Verlag, Rüdigerstr. 14, 70469 Stuttgart, Germany. All rights reserved. This journal, including all individual contributions and illustrations published therein, is legally protected by copyright for the duration of the copyright period. Any use, exploitation or commercialization outside the narrow limits set by copyright legislation, without the publisher's consent, is illegal and liable to criminal prosecution. This applies in particular to photostat reproduction, copying, cyclostyling, mimeographing or duplication of any kind, translating, preparation of microfilms, and electronic data processing and storage.

Studies on the Synthesis of the 1-Hydroxynortropane System; Part II.¹ Synthesis of Calystegine A₃ and Physoperuvine

François-Didier Boyer^* , Paul-Henri Ducrot, Vivien Henryon, Josette Soulié, Jean-Yves Lallemand

^*Laboratoire de Synthèse Organique, Ecole Polytechnique, F-01128 Palaiseau Cedex, France

Weitere Informationen

Publikationsverlauf

Publikationsdatum:
08. März 2002 (online)

als PDF herunterladen Lizenzen und Reprints Alle Artikel dieser Rubrik

Total syntheses of racemic calystegine A₃ {8-azabicyclo-[3.2.1)octane-1,2,3-triol (3)} and physoperuvine {8-methyl-8-azabicyclo[3.2.1]octan-1-ol (4)} are described using intramolecular cyclisation of 4-aminocycloheptanones 7,8. Influence of the substituents on the stability of the cyclisation products is investigated.