Synlett

Issue 03 · February 2013

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A15
Zanda, Matteo: SYNFORM ISSUE 2013/2 FREE ACCESS

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synpacts
269
Lalic, Gojko; Rucker, Richard P.: Copper-Catalyzed Electrophilic Amination of Organoboron Compounds

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276
Streuff, Jan: An Update on Catalytic Strategies for the Synthesis of α-Hydroxyketones

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account
281
Gualandi, Andrea; Cozzi, Pier Giorgio: Stereoselective Organocatalytic Alkylations with Carbenium Ions

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cluster
297
Cluster Cover Page FREE ACCESS

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298
Yasuda, Nobuyoshi: Cluster Preface: Process Chemistry

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301
Chen, Ying; Crockett, Richard D.; Wang, Xin; Larsen, Robert D.; Cui, Sheng; Faul, Margaret M.: Development of a Scalable Synthesis of a VEGFR Inhibitor

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305
Mudryk, Boguslaw; Joshi, Amit; Ortiz, Adrian; Young, Ian S.; Sawyer, James R.; Zheng, Bin; Sugiyama, Masano; Shi, Zhongping; Müslehiddinoğlu, Jale; Corbett, R. Michael; Kronenthal, David R.; Conlon, David A.: Evolution of the Process for the Preparation of a Selective ErbB VEGF Receptor Inhibitor

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313
Houpis, Ioannis N.; Lemaire, Sebastien; Farina, Vittorio; Xiao, Tingting; Liu, Renmao; Nettekoven, Ulrike; Wang, Youchu: New Synthesis of 2′,4′-Functionalized Nucleotides via Stereospecific Hydrogenation and Azidation Reactions

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317
Lu, Bruce Z.; Li, Guisheng; Rodriguez, Sonia; Liu, Jianxu; Eriksson, Magnus C.; Tan, Zhulin; Song, Jinhua J.; Yee, Nathan K.; Farina, Vittorio; Senanayake, Chris H.: Development of a Practical Synthesis of 4-[6-(Morpholinomethyl)-pyridin-3-yl]naphthalen-1-amine, a Key Intermediate for the Synthesis of BIRB 1017, a Potent p38 MAP Kinase Inhibitor

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323
Chase, Charles E.; Fang, Francis G.; Lewis, Bryan M.; Wilkie, Gordon D.; Schnaderbeck, Matthew J.; Zhu, Xiaojie: Process Development of Halaven^®: Synthesis of the C1–C13 Fragment from d-(–)-Gulono-1,4-lactone

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327
Austad, Brian C.; Benayoud, Farid; Calkins, Trevor L.; Campagna, Silvio; Chase, Charles E.; Choi, Hyeong-wook; Christ, William; Costanzo, Robert; Cutter, James; Endo, Atsushi; Fang, Francis G.; Hu, Yongbo; Lewis, Bryan M.; Lewis, Michael D.; McKenna, Shawn; Noland, Thomas A.; Orr, John D.; Pesant, Marc; Schnaderbeck, Matthew J.; Wilkie, Gordon D.; Abe, Taichi; Asai, Naoki; Asai, Yumi; Kayano, Akio; Kimoto, Yuichi; Komatsu, Yuki; Kubota, Manabu; Kuroda, Hirofumi; Mizuno, Masanori; Nakamura, Taiju; Omae, Takao; Ozeki, Naoki; Suzuki, Taeko; Takigawa, Teiji; Watanabe, Tomohiro; Yoshizawa, Kazuhiro: Process Development of Halaven^®: Synthesis of the C14–C35 Fragment via Iterative Nozaki–Hiyama–Kishi Reaction–Williamson Ether Cyclization

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333
Austad, Brian C.; Calkins, Trevor L.; Chase, Charles E.; Fang, Francis G.; Horstmann, Thomas E.; Hu, Yongbo; Lewis, Bryan M.; Niu, Xiang; Noland, Thomas A.; Orr, John D.; Schnaderbeck, Matthew J.; Zhang, Huiming; Asakawa, Naoki; Asai, Naoki; Chiba, Hiroyuki; Hasebe, Takashi; Hoshino, Yorihisa; Ishizuka, Hiroyuki; Kajima, Takashi; Kayano, Akio; Komatsu, Yuki; Kubota, Manabu; Kuroda, Hirofumi; Miyazawa, Mamoru; Tagami, Katsuya; Watanabe, Tomohiro: Commercial Manufacture of Halaven^®: Chemoselective Transformations En Route to Structurally Complex Macrocyclic Ketones

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338
Mayer, Marilyn Graziano; Nador, Fabiana; Volpe, María Alicia; Radivoy, Gabriel: High Surface Area CeO₂ Promoted Suzuki–Miyaura Cross-Coupling of Arylboronic Acids and Aryl Iodides

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343
Spork, Anatol P.; Ducho, Christian: Stereocontrolled Synthesis of 5′- and 6′-Epimeric Analogues of Muraymycin Nucleoside Antibiotics

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347
Dighe, Mahesh G.; Lonkar, Sachin L.; Degani, Mariam S.: Mechanistic Insights into Palladium Leaching in Novel Pd/C-Catalyzed Boron-Heck Reaction of Arylboronic Acid

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351
Pereshivko, Olga P.; Peshkov, Vsevolod A.; Ermolat’ev, Denis S.; Van der Eycken, Erik V.: Fast Assembly of 1H-Imidazo[1,2-a]imidazol-5-amines via Groebke–Blackburn–Bienaymé Reaction with 2-Aminoimidazoles

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355
Titanyuk, Igor D.; Beletskaya, Irina P.: Palladium-Catalyzed Hydroarylation of Diazoacetic Ester

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359
Ehlers, Peter; Petrosyan, Andranik; Ghochikyan, Tariel V.; Saghyan, Ashot S.; Neubauer, Antje; Lochbrunner, Stefan; Langer, Peter: Suzuki–Miyaura Reactions of 2,7-Dichloro-1,8-naphthyridine

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363
Craven, Philip G. E.; Taylor, Richard J. K.: Stereocontrolled Routes to 4-Methoxypentadienoates for Use in Natural Product Synthesis

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369
Varghese, Vimal; Hudlicky, Tomas: Total Synthesis of Dihydrocodeine and Hydrocodone via a Double Claisen Rearrangement and C-10/C-11 Closure Strategy

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375
Narayama, Akira; Shibatomi, Kazutaka; Soga, Yoshinori; Muto, Tsubasa; Iwasa, Seiji: Copper(II)-Catalyzed Enantioselective Fluorination of β-Keto Esters Using Chiral Spiro Oxazoline Ligands

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379
Choi, Juhee; Kim, Hyunseok; Park, Sangyun; Tae, Jinsung: Asymmetric Total Synthesis of (–)-Galanthamine via Intramolecular Heck Reaction of Conjugated Diene

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383
Xu, Xiangsheng; Li, Tao; Li, Xiaoqing; Shao, Jiangbin: Synthesis of Substituted Fluorenes by Cascade Allenylation, Electrocyclization and Intramolecular Friedel–Crafts Reaction of 1,3-Diene-Substituted Propargylic Alcohols

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389
Gao, Detian; Back, Thomas G.: Synthesis of the Reverse Transcriptase Inhibitor L-737,126 and the CB₂ Cannabinoid Receptor Agonist Pravadoline by a Copper-Catalyzed Intramolecular Cross-Coupling

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394
Voltrova, Svatava; Srogl, Jiri: Expedient Method for Samarium(II) Iodide Preparation Utilizing a Flow Approach

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spotlight
397
Fintelman Dias, Flaviana Rodrigues: Ethyl 2-Diazoacetoacetate FREE ACCESS

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399
Gigant, Nicolas: Triflic Acid FREE ACCESS

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erratum
e1
Chase, Charles E.; Fang, Francis G.; Lewis, Bryan M.; Wilkie, Gordon D.; Schnaderbeck, Matthew J.; Zhu, Xiaojie: Process Development of Halaven^®: Synthesis of the C1–C13 Fragment from d-(–)-Gulono-1,4-lactone

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e2
Austad, Brian C.; Benayoud, Farid; Calkins, Trevor L.; Campagna, Silvio; Chase, Charles E.; Choi, Hyeong-wook; Christ, William; Costanzo, Robert; Cutter, James; Endo, Atsushi; Fang, Francis G.; Hu, Yongbo; Lewis, Bryan M.; Lewis, Michael D.; McKenna, Shawn; Noland, Thomas A.; Orr, John D.; Pesant, Marc; Schnaderbeck, Matthew J.; Wilkie, Gordon D.; Abe, Taichi; Asai, Naoki; Asai, Yumi; Kayano, Akio; Kimoto, Yuichi; Komatsu, Yuki; Kubota, Manabu; Kuroda, Hirofumi; Mizuno, Masanori; Nakamura, Taiju; Omae, Takao; Ozeki, Naoki; Suzuki, Taeko; Takigawa, Teiji; Watanabe, Tomohiro; Yoshizawa, Kazuhiro: Process Development of Halaven^®: Synthesis of the C14–C35 Fragment via Iterative Nozaki–Hiyama–Kishi Reaction–Williamson Ether Cyclization

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e3
Austad, Brian C.; Calkins, Trevor L.; Chase, Charles E.; Fang, Francis G.; Horstmann, Thomas E.; Hu, Yongbo; Lewis, Bryan M.; Niu, Xiang; Noland, Thomas A.; Orr, John D.; Schnaderbeck, Matthew J.; Zhang, Huiming; Asakawa, Naoki; Asai, Naoki; Chiba, Hiroyuki; Hasebe, Takashi; Hoshino, Yorihisa; Ishizuka, Hiroyuki; Kajima, Takashi; Kayano, Akio; Komatsu, Yuki; Kubota, Manabu; Kuroda, Hirofumi; Miyazawa, Mamoru; Tagami, Katsuya; Watanabe, Tomohiro: Commercial Manufacture of Halaven^®: Chemoselective Transformations En Route to Structurally Complex Macrocyclic Ketones

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