Synthesis 1988; 1988(7): 529-533
DOI: 10.1055/s-1988-27625
paper
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A Simple Method for N-Amination of Peptide Derivatives

F. Szurdoki* , S. Andreae, E. Baitz-Gács, J. Tamás, K. Valkó, E. Schmitz, Cs. Szántay
  • *Central Research Institute for Chemistry of the Hungarian Academy of Sciences, H-1525 Budapest, P. O. Box 17, Hungary
Further Information

Publication History

Publication Date:
18 September 2002 (online)

A smooth and mild procedure is reported for the N-amination of α-amino acid and peptide derivatives with cyclohexanespiro-3′-oxaziridine; the chiral integrity is preserved throughout.