Synthesis 2023; 55(07): 1123-1129
DOI: 10.1055/a-1983-3890
paper

Samarium-Promoted Homocoupling of Benzaldehydes and In Situ Condensation with Esters Under the Catalysis of Cuprous Iodide

Hongping Chen
,
Bin Song
,
Mingzhong Mi
,
Yan Qi
,
Yongjun Liu
The project was sponsored by the Shandong Provincial Key Research and Development Program (SPKR&DP) (2019GGXI02036), and the Open Project of Faculty of Chemistry of Qingdao University of Science and Technology (QUSTHX201902).


Abstract

A novel C–H functionalization method was successfully explored by a reductive three molecule coupling of benzaldehydes and esters mediated by samarium and cuprous iodide; thus, the diarylmethanol skeletons were afforded readily via an in situ esterification in one-pot. Substrates including a variety of esters and different benzaldehydes were investigated, and the desired products were readily obtained in moderate to good yields under mild conditions.

Supporting Information



Publication History

Received: 03 September 2022

Accepted after revision: 21 November 2022

Accepted Manuscript online:
21 November 2022

Article published online:
14 December 2022

© 2022. Thieme. All rights reserved

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Rüdigerstraße 14, 70469 Stuttgart, Germany

 
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