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© Georg Thieme Verlag Stuttgart ˙ New York

Efficient and Scalable Synthesis of 3,5,7-Trisubstituted 1H-Indazoles as Potent IKK2 Inhibitors

Xichen Lin*a, Jakob Busch-Petersena, Jianghe Denga, Christine Edwardsb, Zhaoguo Zhangc, Jeffrey K. Kernsa
a Respiratory Center of Excellent Drug Discovery, GlaxoSmithKline, 709 Swedeland Road, King of Prussia, PA 19406, USA
Fax: +1(610)2704451; e-Mail: Xichen.2.Lin@gsk.com;
b Argenta Discovery Ltd. , 8/9 Spire Green Centre, Flex Meadow, Harlow, Essex CM19 5TR, UK
c School of Chemistry and Chemical Engineering, Shanghai Jiaotong University, 800 Dongchuan Road, Shanghai 200240, P. R. of China