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Synfacts 2011(2): 0178-0178
DOI: 10.1055/s-0030-1259335
DOI: 10.1055/s-0030-1259335
Metal-Catalyzed Asymmetric Synthesis and Stereoselective Reactions
© Georg Thieme Verlag
Stuttgart ˙ New York
Copper-Catalyzed Synthesis of 3-Aminoindoles and Pyrroloindolines
T. Benkovics, I. A. Guzei, T. P. Yoon*
University of Wisconsin-Madison, USA
Further Information
Publication History
Publication Date:
19 January 2011 (online)
Significance
Indoles and pyrroloindolines are common motifs found in natural products and pharmaceuticals. The authors present an oxyamination of indoles using Davis oxaziridines to produce complex oxazolidine products, which can be readily transformed into 3-aminopyrroloindolines.