One-Pot Synthesis of Functionalized Arylboronic Acids

doi:10.1055/s-0031-1289204

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Synfacts 2011(11): 1225-1225
DOI: 10.1055/s-0031-1289204

Metal-Mediated Synthesis

One-Pot Synthesis of Functionalized Arylboronic Acids

Contributor(s): Paul Knochel, Nadja M. Barl
T. Leermann, F. R. Leroux*, F. Colobert*
Université de Strasbourg, France

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Publication History

Publication Date:
19 October 2011 (online)

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Significance

The authors report a simple one-pot synthesis of various functionalized arylboronic acids via electrophilic borylation of Grignard reagents, which are prepared either by direct magnesium insertion in the presence of LiCl or by a bro-mine-magnesium exchange using i-PrMgCl˙LiCl.