Synfacts

Issue 12 · December 2012

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A122
SYNFORM ISSUE 2012/12 FREE ACCESS

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Synthesis of Natural Products and Potential Drugs
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1279
Synthesis of the CGRP Receptor Antagonist BMS-846372

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1280
Formal Total Syntheses of Didehydrostemofoline and Isodidehydrostemofoline

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1281
Synthesis of (−)-205B

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1282
Synthesis of Piragliatin

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1283
Synthesis of Bixafen

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1284
Total Synthesis of (+)-Ibophyllidine

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1285
Total Synthesis of (±)-Gracilamine

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1286
Formal Synthesis of Ezetimibe

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1287
Total Syntheses of Incarviditone and Incarvilleatone

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1288
Synthesis of AM-1638

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1289
Synthesis of DS-8108b

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1290
Synthesis of (–)-Huperzine A

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1291
Enantioselective Synthesis of (+)-Cubitene

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1292
Enantioselective Total Synthesis of Prostaglandin PGF_2αin Seven Steps

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1293
Synthesis of LY411575

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Synthesis of Heterocycles
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1295
Palladium-Catalyzed Cyclization of Electron-Deficient Enynes

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1296
A Palladium-Catalyzed Multicomponent Heteroannulation Route to Indoles

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1297
A Pd-Catalyzed C–H Activation Route to Benzisoxazolones

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1298
Rhodium-Catalyzed Synthesis of 3-Aryl Indoles from 1-Sulfonyl 1,2,3-Triazoles

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1299
Synthesis of Sultams via Rh(III)-Catalyzed Directed C–H Activation

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1300
Synthesis of Imidazopyridines by Cu(II)/Fe(III) Co-catalyzed C–N Coupling

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1301
Synthesis of 5-Acyl-2-amino-1,3,4-thiadiazoles From Acid Chlorides

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1302
Synthesis of Functionalized Azaindolines and Azatetrahydroquinolines

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1303
Stereoselective Access to Quaternary Carbon Atoms via S_N2 Cleavage of Azetidinium Ions

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1304
Ru-Catalyzed Synthesis of Polysubstituted Pyrazoles

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1305
Copper–Silver Cocatalyzed Synthesis of Pyrazoloisoquinolines

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1306
Synthesis of 3-Aminoindolizines Enabled by Flow Technology

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1307
Synthesis of Cyclic Azomethine Imines as Precursors to β-Aminocarbonyl Scaffolds

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1308
Copper-Catalyzed Synthesis of 1,4-Dihydroazete Derivatives

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1309
Cu- and Ni-Catalyzed Regioselective Synthesis of Disubstituted Pyrroles

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Synthesis of Materials and Unnatural Products
z1311
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1311
Breaking the B≡N Bond for 1,4-Azaborines

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1312
A Two-Step Procedure to Brominated 2-Alkoxythiophenes

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1313
Radical Dearomatization and Two-Electron Reduction of a Redox-Active Ligand

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1314
A Stable Phosphinonitrene

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1315
Triphenylene-Based Electron-Deficient Discotic Liquid Crystals

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1316
A Tetrabenzoporphyrin Precursor in Four Steps

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1317
From Carboxylic Acids to Alkyl Bromides by Reductive Bromination

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1318
Extending Porphyrinoids with Fused Anthracenes

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1319
A FRET Donor–Acceptor Copolymer with Spatially Alternating Transition Dipoles

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1320
Regioselective Synthesis of Fused Anthracenes

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1321
Synthesis of Photocleavable Star Polymers by the ‘Brush-First’ Method

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1322
Mild Gold-Catalyzed Biaryl Synthesis

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Metal-Catalyzed Asymmetric Synthesis and Stereoselective Reactions
z1323
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1323
Counteranion-Directed Tsuji–Trost Reaction

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1324
Solvent- or Temperature-Controlled Diastereoselective Aldol Reaction

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1325
Nickel-Catalyzed Intermolecular [2+2] Cycloaddition

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1326
Palladium-Catalyzed Cycloisomerization of 1,n-Dienes via a Chain-Walking Mechanism

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1327
Ru–NHC Catalyzed Asymmetric Hydrogenation of Benzothiophenes

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1328
Ru(CO)-salen Catalyzed Aziridination of Vinyl Ketones

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1329
Copper–NHC Catalyzed Conjugate Addition of Grignard Reagents

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1330
Iridium-Catalyzed Asymmetric Hydrogenation of N-Benzyl Pyridinium Bromides

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1331
Palladium-Mediated Asymmetric Synthesis of 3-Amino-2-oxindoles

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1332
Gold Catalyzed Ene–Yne Cyclization for the Formation of Benzo[b]oxepines

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1333
Copper–NHC Catalyzed Hydroboration of Propargylic Substrates

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1334
Axially Chiral Carbene Gold Complex Catalyzed [4+2] Cycloadditions

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1335
Copper-Catalyzed Asymmetric Henry Reaction

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1336
Iridium-Catalyzed Asymmetric Allylation of Trimethylsiloxy Furans

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1337
Iridium-Catalyzed Asymmetric Transfer Hydrogenation in Water

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1338
Allylation of Cyclopropanols via Zinc–Copper Homoenolates

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1339
Palladium-Catalyzed Asymmetric Alkene Carboamination

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1340
Palladium-Catalyzed Stereospecific Suzuki–Miyaura Cross-Coupling

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1341
Asymmetric Synthesis of β-Aryl-β-Boronyl Enoates

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1342
Rh-catalyzed Asymmetric Conjugate Addition to Dihydronitronaphthalenes

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1343
Chiral Quaternary Carbons from Organolithiums and Organocuprates

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1344
Ruthenium-Catalyzed Formal Arylformylation of E-β-Bromostyrenes with Aldehydes

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1345
Ruthenium-Catalyzed C–C Coupling of Dienes to α‑Hydroxy Esters

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1346
Silver-Catalyzed Enantioselective Conjugate Addition and Cycloaddition

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1347
Merged Au–Enamine Catalysis for Enantioselective α-Allylic Alkylation

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1348
Cyclobutenamides by Rhodium-Mediated Formal [2+2] Cycloaddition

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1349
Rhodium-Catalyzed Asymmetric Coupling Reactions of Allylic Ethers

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1350
Copper-Catalyzed [6+3] Cycloadditions of Azomethine Ylides with Fulvenes

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1351
2,6-cis-Tetrahydropyranes via an Asymmetric Tandem Sequence

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1352
Kinetic Resolution of N-Acylaziridines

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Metal-Mediated Synthesis
z1353
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1353
Ruthenium-Catalyzed Hydroboration of Terminal Alkynes

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1354
Synthesis of Secondary Aminomethylated Arenes via Cross-Coupling

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1355
Stereoselective Cu-Mediated Oxyamination to Yield Morpholines

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1356
Difluoromethylation of Lithium Enolates by Umpolung of Fluoroform

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1357
Cu-Mediated Trifluoromethylation of Boronic Acids using NaSO₂CF₃ and TBHP

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1358
Cross-Coupling of Benzyl Alcohols with Grignard Reagents

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1359
Catalytic Boracarboxylation of Alkynes using B₂(pin)₂ and CO₂

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1360
Ruthenium-Catalyzed Transformation of Aryl and Alkenyl Triflates into Halides

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1361
Copper-Mediated Trifluoromethylation of α-Diazo Esters with TMSCF₃

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1362
Iron- and Zink-Mediated Synthesis of Oxazolines and Oxazoles

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1363
Boron-to-Zinc Exchange of Allyl Organometallic reagents

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1364
Cobalt-Catalyzed Migratory Arylzincation of Alkynes

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1365
Ni-Catalyzed Kumada Reaction of Tosylalkanes and Aryltosylethanones

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1366
Trifluoromethylation of α-Haloketones with Fluoroform-Derived CuCF₃

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1367
Electrophilic Trifluoromethanesulfanylation of Organometallic Species

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Organo- and Biocatalysis
z1369
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1369
Medium Ring Size Bromolactonization

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1370
Enantioselective Brønsted Acid Catalyzed Route to Pyrroloindolines

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1371
Thiourea-Catalyzed Ring Opening of Episulfonium Ions with Indole Derivatives

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1372
Amidine Catalyzed Kinetic Resolution of Lactams and Thiolactams

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1373
A Supported Squaramide as a Recyclable Catalyst for Michael Additions

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1374
Light-Driven Organocatalytic Synthesis of Benzothiophenes

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1375
Organocatalytic Activation of Anthracenes in Asymmetric Diels–Alder Reactions

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1376
Cinchona Alkaloid Derivatives Catalyzed Asymmetric [4+2] Cycloaddition

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Polymer-Supported Synthesis
z1377
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1377
Green LED Responding Photocatalytic Oxidation of Alcohols with Au/CeO₂

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1378
Preparation of Benzimidazoles via Hydrogen Transfer with Pd/C

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1379
Suzuki Coupling With a Supported Pd–Glucosamine Phosphine Complex

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1380
Oxidative Esterification and Imination of Alcohols Using Au/Mg_xAl-HT

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1381
Polystyrene-Supported Pd(II) for Heck and Sonogashira Reactions

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1382
Au-Nanoparticle-Catalyzed Hydrosilylation of Alkynes

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1383
α-Hydroxylation of 1,3-Dicarbonyl Compounds Using PI/CB-Au

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1384
A Cooperative Catalytic System for the Aerobic Oxidation of Amines

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1385
Asymmetric Henry–Michael Reaction with Bifunctional Catalysts

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1386
Controlled Hydrogenation of Nitroarenes Using Ruthenium NPs/Charcoal

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1387
Aerobic Oxidation of Alcohols with Pd Nanoparticles on AmP-MCF

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1388
Reduction of Nitroarenes and Carbonyl Compounds with Ni–Fe₃O₄ MNPs

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1389
Synthesis of Aryloxypyridines via Pd/C-Catalyzed Suzuki–Miyaura Cross-Coupling

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