DOI: 10.1055/s-00000131

Synfacts

Issue 08 · Volume 9 · August 2013 DOI: 10.1055/s-003-25362

Synform

A92
Zanda, Matteo: SYNFORM ISSUE 2013/08

Synthesis of Natural Products and Potential Drugs

z805
All PDFs of this category
0805
Synthesis of Dictyostatin
0806
Synthesis of IDX320
0807
Total Synthesis of BE-43472B
0808
Total Synthesis of (+)-Schisanwilsonene A
0809
Total Synthesis of Caribenol A
0810
Synthesis of Combretastatin A-4
0811
Synthesis of a TORC 1/2 Inhibitor
0812
Synthesis of (+)-Bionectin A and C
0813
Synthesis of (+)-Armillarivin
0814
Synthesis of (±)-Gelsemoxonine
0815
Synthesis of Eravacycline

Synthesis of Heterocycles

z817
All PDFs of this category
0817
SNAr Route to Pyrazolo[3,4-d]pyrimidines
0818
Regioselective C–H Activated Alkylation of Pyrroles
0819
Furoxan Synthesis From Styrenes Under Non-Acidic Conditions
0820
18F-Labeled Heterocycles by Huisgen 1,3-Dipolar Cycloaddition
0821
Synthesis of [1,2]Oxazino[5,4-b]indoles by Intermolecular [3+3] Cycloaddition
0822
Synthesis of Quinazolinones via Radical Skeletal Rearrangement
0823
Synthesis of Fluorinated Azabicycles
0824
Efficient Chelation-Controlled Synthesis of Aza-Sugars from Aziridines
0825
Pd/In-Catalyzed Synthesis of Furans from β-Methoxystyrene and Dicarbonyls
0826
Au(I)/Ag(I)-Heteroannulation Approach to Heterocycles with a Very Long Name
0827
Synthesis of Benzo and Fused Heterocyclic Imidazoles from Nitroaminoaryls
0828
Rhodium(III)-Catalyzed C–H Activation Route to Azepinones
0829
C(sp3)–N Bond Formation for the Synthesis of Five- to Seven-Membered Azacycles
0830
Synthesis of Spiro[indoline]oxindoles from Isatin Ketonitrones and Alkynes
0831
Heteroannulative C–H Activation Route to Pyrazoles and Indazoles

Synthesis of Materials and Unnatural Products

z833
All PDFs of this category
0833
Dibenzo[a,e]pentalenes by ortho C–H Activation
0834
Pyrrole-Fused Azacoronene
0835
trans-Substituted Cyclobutanes by Electron Relay
0836
Surprise Synthesis of Azulenophenanthrenes
0837
Aromatic Trifluoromethylation
0838
A Pyrrole-Free Porphyrin: Synthesis of Azacalixphyrin
0839
Star- and Figure-Eight-Shaped Polyethers via Ring-Opening Polymerization
0840
Cleaving Carbon–Carbon Triple Bonds –A New Route to Nitriles
0841
Synthesis of a Series of Armchair SWCNT Segments
0842
Lewis Acid Catalyzed Formation of Dibenzopentalenes
0843
A New, Strongly Electron-Donating Building Block for Low-Bandgap Polymers
0844
Polymer Semiconductors Based on a New Electron-Accepting Building Block

Metal-Catalyzed Asymmetric Synthesis and Stereoselective Reactions

z833
All PDFs of this category
0845
Palladium-Catalyzed Asymmetric Allylation of Cyclobutene Derivatives
0846
Enantioselective Aziridination Catalyzed by a Cobalt(II)–Porphyrin Complex
0847
Highly Enantioenriched Allylsilanes via Copper-Catalyzed Allylic Substitution
0848
Spirocyclic Diketones via Asymmetric Redox-Pinacol–Mannich Cascade
0849
Diastereo- and Enantioselective Addition of Allylcopper to Carbonyls
0850
Vinylidenecyclopentane Synthesis by Palladium-Catalyzed [3+2] Cycloaddition
0851
Ruthenium-Catalyzed Dynamic Kinetic Resolution of β-Amino-α-Hydroxy Esters
0852
Dynamic Kinetic Friedel–Crafts Alkylation of Indoles with Cyclopropanes
0853
Silver-Catalyzed Asymmetric [3+2] Cycloaddition of Azomethine Ylides
0854
Synthesis of 2,3-Diaminosuccinic Acid Derivatives by Rhodium Catalysis
0855
Nickel-Catalyzed Asymmetric Direct Reductive Acyl Cross-Coupling Reaction
0856
Synthesis of Planar-Chiral Carba-Paracyclophanes by Rhodium Catalysis
0857
Rhodium-Catalyzed One-Pot Cyclo-isomerization/Hetero-Diels–Alder Reaction
0858
Rhodium-Catalyzed Enantioselective [2+2+2] Cycloaddition
0859
Asymmetric [2+2+2] Cycloaddition of Alkenyl Isocyanates with Alkynes
0860
Synthesis of Enantioenriched β-Bromo Oxazolidinones
0861
Enantioselective Hydrogenation of Tetra-substituted Olefins
0862
A Regioselective Palladium-Catalyzed Allylic Alkylation Cascade with Dihydropyrans
0863
Copper-Catalyzed Cyclopentannulation of Indoles
0864
Four-Step Sequence Involving an Electrophilic Trapping Reaction
0865
Self-Assembling Ligand/Rhodium-Catalyzed Alkyne Hydroformylation
0866
Diastereoselective Synthesis of Butyro-lactones via Palladium-Catalyzed Allylation
0867
[8+2] Cycloaddition of Azaheptafulvenes with Alkylidene Malonates
0868
Amide–Copper(II)-Catalyzed Asymmetric Vinylogous Mannich Reaction
0869
Enantioselective Cyclopropanation of α,β-Unsaturated Carbonyl Compounds
0870
Palladium-Catalyzed Decarboxylative Allylation of Glycal Derivatives
0871
Silver-Catalyzed Enantioselective Desymmetrization of Spirolactones
0872
Bimetallic Enantioselective Synthesis of Axially Chiral Allenes
0873
Ammonium Salt Accelerated Asymmetric Additions of Diethylzinc
0874
Iridium-Catalyzed Synthesis of Polycyclic Indoles and Pyrroles

Metal-Mediated Synthesis

z875
All PDFs of this category
0875
Asymmetric Strecker-Type Reaction of Nitrones Using Cyanohydrin
0876
Highly Enantioselective Fluorocyclopropanation of Allylic Alcohols
0877
Carbocupration of Cyclopropene Carboxylic Acid Esters
0878
Palladium-Catalyzed ortho-Selective C–F Activation with Triethylsilane
0879
Transition-Metal-Free Direct Arylation with Grignard Reagents
0880
Hydrosilane-Directed Borylation of Secondary Benzylic C−H Bonds
0881
Directed Amination of Non-Acidic Arene C–H Bonds
0882
Samarium-Mediated Synthesis of Indolizidines, Quinolizidines, and Piperidines
0883
Photoinduced, Copper-Catalyzed N-Alkylation of Carbazoles
0884
Synthesis of Phenanthrenes via Induction by Silicon
0885
Palladium-Catalyzed Olefination and Arylation of 2-Substituted 1,2,3-Triazole N-Oxides
0886
Copper-Mediated Electrophilic Imination of Alkenyl Zirconocenes
0887
Copper-Catalyzed Reaction of Internal Alkynes and Diaryliodonium Salts
0888
SET-Induced Cross-Couplings of Alkenyl Halides with Aryl Grignard Reagents
0889
Synthesis and Pauson–Khand Reaction of Trifluoromethylated Alkynes
0890
Stereoselective Titanium-Mediated Aldol Reactions

Organo- and Biocatalysis

z891
All PDFs of this category
0891
Another Stereochemical Model for Cinchona-Derived Primary Amine Catalysts
0892
C–C Coupling Catalyzed by a Protonated Diamine
0893
Enantio- and Diastereodivergent Dual Catalysis
0894
Kinetic Resolution of Unsaturated Carboxylic Acids via Protolactonization
0895
Regio- and Enantioselective Organocatalyzed 1,6-Additions
0896
Catalytic Asymmetric Remote Aziridination
0897
Catalytic Enantioselective Synthesis of Hindered Cyclic Ethers
0898
Stereoselective Synthesis and Functionalization of Tetrahydroquinolines
0899
Neutral Multidentate Halogen-Bond Donors as Organocatalysts
0900
Phase-Transfer-Catalyzed Asymmetric Alkylation of 2‑Arylcyclohexanones
0901
Desymmetrization of Oxetanes with Sulfur Nucleophiles

Polymer-Supported Synthesis

z903
All PDFs of this category
0903
Copper-Impregnated Magnetite for Glaser–Hay Reaction
0904
PdONPs-Catalyzed Synthesis of Dibenzyls and 3-Arylpropionic Acids
0905
Co3O4–Nitrogen Complex for Hydrogenation of Nitroarenes
0906
Cross-Coupling of Terminal Alkynes with Hydrosilanes Using Au/OMS-2
0907
Dehydrative N-Acylation of Amines with Nano-CeO2
0908
C3-Selective Direct Arylation of Benzo[b]thiophenes with Aryl Chlorides
0909
Suzuki Coupling and Reduction of Nitrobenzenes with Pd- and Rh-Fe3O4
0910
Meerwein Arylation of Benzoquinone with Anilines Using CuONPs/Gr
0911
DNA-MMT Hybrid-Supported Metal Nanoparticle Catalysts
0912
Preparation of Quinolines and Pyridocoumarins with Au/TiO2
0913
Sequential Azasulfenylation and Huisgen Cycloaddition Using CuNPs/C
0914
Silica-Supported Molybdenum Nitride for Alkyne Metathesis