DOI: 10.1055/s-00000131

Synfacts

Issue 09 · Volume 10 · September 2014 DOI: 10.1055/s-004-27536

Synform

A114
Zanda, Matteo: SYNFORM ISSUE 2014/09

Synthesis of Natural Products and Potential Drugs

z893
All PDFs of this category
0893
Synthesis of the Antifungal Agent ASP9726
0894
Synthesis of γ-Secretase Modulator SPI-1865
0895
Total Synthesis of Sespenine
0896
Synthesis of Taiwaniadducts B, C, and D
0897
Synthesis of a Saxagliptin Fragment
0898
Synthesis of (±)-Penifulvin A
0899
Total Synthesis of Sculponeatin N
0900
Synthesis of Both Enantiomers of Mequitazine
0901
Synthesis of ALK Inhibitor PF-06463922
0902
Total Synthesis of (–)-Nitidasin
0903
Total Synthesis of Coccinellid Alkaloids
0904
Syntheses of (+)-Psoracorylifol B and (+)-Psoracorylifol C

Synthesis of Heterocycles

z905
All PDFs of this category
0905
Synthesis of Bioactive Nucleoside Analogues
0906
2,3-Dihydro-1H-indazoles by Rhodium Catalysis
0907
C–H Fluorination and Nucleophilic Aromatic Substitution of Nitrogen Heterocycles
0908
2H‑Indazoles by Condensation−Cadogan Reductive Cyclization
0909
Pd/C-Catalyzed Synthesis of 2-Substituted Benzothiazoles
0910
Diastereoselective Preparation of Enantioenriched Polycyclic Oxoquinolines
0911
Intramolecular Aryl–Aryl Coupling of 2-Substituted N-Phenylbenzamides
0912
Synthesis of 1,3-Oxathiolan-2-ylidenes from α-Enolic Dithioesters and Epoxides
0913
Synthesis of Oxepines by Cycloisomerization of 1,7-Oxadienes
0914
Biomimetic Synthesis of Symmetrical Tetrasubstituted Pyrroles
0915
Three-Component Synthesis of Fully Substituted Triazoles
0916
Synthesis of Pyrroles by Photocatalyzed Cycloaddition of Alkynes to Azirines
0917
C(sp2)–C(sp3) Bonds by Intramolecular Reductive Cross-Coupling
0918
Fused Heterocycles via C–H Activation and Cyclization of Indoles and Pyrroles

Synthesis of Materials and Unnatural Products

z919
All PDFs of this category
0919
SET Sets the Stage: Photochemical Synthesis of Aminomethylfullerenes
0920
Activate Twice, Then Annulate
0921
Get Your Biotin Kicks on Route 6+6
0922
Stabilization of Hexacenes by Dioxolane Functionalization
0923
Heterobenzene Club Welcomes First Aluminum Member
0924
Highly Fluorinated Luminescent Subporphyrins
0925
Light the Way: Phenanthro[9,10-c]thiophenes by Photocyclization
0926
[2+2+2] to Twist: Synthesis of [9]- and [11]Helicene-Like Molecules
0927
Reduce, Rearrange, Reoxidize: Thermal Route to a Ladder Diborole
0928
Better Building of Benzo[b]phosphole Derivatives
0929
Intramolecular Acylation of Biarylcarboxylic Acids to Fluorenones
0930
We All Scream for Selenophenes

Metal-Catalyzed Asymmetric Synthesis and Stereoselective Reactions

z931
All PDFs of this category
0931
Diastereo- and Enantioselective Iridium-Catalyzed Annulation of Salicylimines
0932
Intramolecular Heck Reaction of Secondary Benzylic Ethers
0933
Dearomative Cycloadditions Catalyzed by Palladium
0934
Iridium-Catalyzed Hydrogenation of Pyrrolo[1,2-a]pyrazinium Salts
0935
Asymmetric Hydrogenation of Quinolin-3-amines
0936
Enantioselective Synthesis of 2-Arylchromenes via Palladium Catalysis
0937
Allylic Substitution of Enolates Derived from α,β-Unsaturated Ketones
0938
Cyclopropanation of Allenes Catalyzed by Ruthenium
0939
Enantioselective Copper-Catalyzed 1,4-Addition and Enolate Trapping
0940
Titanium-Promoted Asymmetric Cyclo-propanation of N-Alkenyl Thioamides
0941
Isoindolines via Enantioselective C−H Insertion of Diazo Compounds
0942
Enantioselective β-Lactam Synthesis via Pd-Catalyzed C(sp3)–H Alkylation
0943
Enantioselective Rhodium-Catalyzed Primary C–H Bonds
0944
Hetero-Diels–Alder Reaction of Danishefsky’s Diene with Keto Esters
0945
Direct syn-Selective Asymmetric Mannich-Type Reaction
0946
Copper-Catalyzed Asymmetric 1,4-Additions to α,β-Unsaturated Lactones
0947
Allylic Sulfonamides via a Palladium-Catalyzed Rearrangement of Allylic Carbonates
0948
Selective Synthesis of Secondary Alkyl Fluorides
0949
Asymmetric Hydrogenation of Disubstituted Furans
0950
Enantioselective Rh-Catalyzed Additions to Cyclic N-Sulfamidate Ketimines
0951
Enantioselective Copper-Catalyzed Decarboxylative Propargylic Alkylation
0952
Diastereoselective Gold-Catalyzed Cycloisomerization of Enediynes
0953
Carboetherification–Intermolecular Heck-Type Coupling
0954
Asymmetric Friedel–Crafts Alkylation Catalyzed by Copper
0955
Enantioselective Alkylative Ring Opening Catalyzed by Rhodium
0956
Enantioselective Aminolactonization by Means of Copper Catalysis
0957
Scandium-Catalyzed Enantioselective Epoxidation of 2-Arylidene-1,3-diketones
0958
Polyenes via Palladium- and Chromium-Catalyzed Allylic C–H Olefination
0959
Synthesis of Chiral Cyclic Allylic Amines via Rhodium-Catalyzed Hydrogenation

Metal-Mediated Synthesis

z961
All PDFs of this category
0961
Copper-Catalyzed Trifluoromethylthiolation
0962
Copper-Mediated Three-Component Reaction
0963
Stereospecific Coupling of Aromatics with Secondary and Tertiary Boronates
0964
Arylboration by Cooperative Pd/Cu Catalysis
0965
Gold-Catalyzed Cross-Coupling of Aryl Boronic Acids
0966
Cobalt-Catalyzed Migratory Arylzincation
0967
trans-Diborylation of Propargylic Alcohols
0968
Cyclotrimerization of Alkynes Mediated by n-BuLi–Ti(Oi-Pr)4
0969
Synthesis of Allenyl Boronates by Pd/Cu Catalysis
0970
Amide-Directed C–NMe2 Bond Activation and C–C Coupling Reactions
0971
Lead-Mediated Arylation Using Aryl Azides for the Synthesis of 3H-Indoles
0972
SmI2-Induced Umpolung of Glycals
0973
Nickel-Catalyzed Regioselective 1,4-Addition of Organoboronic Acid to Dienones
0974
Zinc-Mediated C–H Activation of THF
0975
Tandem Divergent Catalysis using Nitriles

Organo- and Biocatalysis

z977
All PDFs of this category
0977
Catalytic Enantioselective [2+2] Intermolecular Photocycloaddition
0978
Desymmetrization of Cyclohexadienones via Dienamine Catalysis
0979
Metal-Free Arylation via a [3,3]-Sigmatropic Rearrangement
0980
Stereoselective 1,2-Dibromination of Olefins Catalyzed by Ph3PO
0981
Lewis Base Catalyzed Enantioselective Sulfenoamination of Olefins
0982
(+)-trans-Dyhydrolycoricidine via an Organocatalytic Michael–Aldol Sequence
0983
Diastereodivergent Synthesis of Tetrasubstituted Cyclohexanes
0984
Cooperative N-Heterocyclic Carbene–Chiral Phosphate Organocatalysis
0985
Highly Enantioselective Route to Chromenes
0986
Organocatalytic Asymmetric Hydrolysis of Epoxides
0987
Preparation of (S)-CHBE by Bioreduction–Optimization and Scale-up
0988
Esterase-Catalyzed Desymmetrization of a meso-Diester

Polymer-Supported Synthesis

z989
All PDFs of this category
0989
An Immobilized Cobalt Complex for Alkyne-Tagged Peptide Enrichment
0990
Cyanation of Aryl Halides with K4[Fe(CN)6] Using ZnO-Pd Nanoparticles
0991
Core–Shell Palladium Nanocatalysts for the Oxidation of Alcohols
0992
Palladium-Catalyzed Hydrogenation Using a Continuous Flow System
0993
Cycloaddition of CO2 to Epoxides Using Polymer-Supported NHC–Zn
0995
Immobilized Rhodium Catalysts for Asymmetric Hydroformylation of Alkenes
0996
Synthesis of Benzoxazoles and Benzimidazoles Using Au/TiO2
0997
Amide Condensation with MCF-Supported Boronic Acids
0998
N-Methylation of Secondary Amines with CO2 and H2 Using Pt-MoOx/TiO2
0999
Preparation of Indoles and Indolines via Pd/C-Mediated Cross-Couplings
1000
Synthesis of 5-Substituted 1H-Tetrazoles Using Ln(OTf)3–SiO2
1001
Oxidative Dimerization of Thioamides Using Phosphovanadomolybdic Acid
1002
C3-Formylation of Indoles Using CAN-SiO2