DOI: 10.1055/s-00000131

Synfacts

Issue 04 · Volume 12 · April 2016 DOI: 10.1055/s-006-31372

Synform

A48
Zanda, Matteo: SYNFORM ISSUE 2016/04

Synthesis of Natural Products and Potential Drugs

z329
All PDFs of this category
0329
Synthesis of Ileabethoxazole, Pseudo-pteroxazole, and seco-Pseudopteroxazole
0330
Synthesis of (±)-Alstoscholarisine A
0331
Synthesis of MK-8831
0332
Synthesis of rac-Jungermannenones B and C
0333
Synthesis of (+)- and (–)-Perhexiline
0334
Synthesis of (+)-Asperazine, (+)-Pestalazine A, and (+)-iso-Pestalazine A
0335
Syntheses of (+)-Strictamine, (–)-2(S)-Cathafoline, and (–)-Aspidophylline A
0336
Synthesis of seco-Prezizaane Sesquiterpenes
0337
Synthesis of (+)-Lycopalhine A
0338
Synthesis of (+)-BMS-820836
0339
Synthesis of (+)-Asenapine
0340
Synthesis of Talazoparib

Synthesis of Heterocycles

z341
All PDFs of this category
0341
Copper-Catalyzed Synthesis of Substituted 1,4-Oxathianes
0342
Piperazines by Palladium-Catalyzed Reactions of Propargylic Alcohols
0343
Tetrafluoroimidazopyridines by Radical-Mediated Annulation
0344
Synthesis of Pyridinyl and Quinolinyl Triflates or Tosylates by Diazotization
0345
Biomimetic Photocatalytic C–H Activation Route to Coumarins
0346
γ-Lactams by Palladium-Catalyzed Intramolecular C(sp3)−H Alkenylation
0347
Iodine-Mediated Synthesis of Pyrido[1,2-a]benzimidazoles
0348
Synthesis of (Aminoalkyl)boronates from Cyclic Sulfamidates
0349
Spiropyrazolones by Sequential Michael and Conia–ene Reactions
0350
Isoquinolinium, Cinnolinium, and Quinolizinium Salts by Oxidative Annulation
0351
Synthesis of 3-Fluoropyrroles by Ring-Closing Metathesis
0352
Synthesis of Propellane, Azetidine, and Cyclobutane Amines
0353
Synthesis of Indolines by an Iron-Catalyzed (4+1) Cycloaddition
0354
Fluorinated 4H-1,4-Thiazine 1,1-Dioxides

Synthesis of Materials and Unnatural Products

z355
All PDFs of this category
0355
Synthesis of Novel Extended Tetrathiafulvalene Donors for OFETs
0356
N-Heteroarenes: 13 Rings in a Row
0357
A Super Electron Deficient Polymer
0358
Synthesis of Sulfur-Substituted Phosphangulenes
0359
Beyond Six Spiroketal-Linkages With Thioketals
0360
Stabilized Z-Shaped Acenes
0361
Molecularly Woven Organic Polymer Chains
0362
A Radical Idea for Stabilization
0363
It’s Elemental! S8 in Poly(benzoxazine) Copolymerizations
0364
The Meso–Meso Linked Antiaromatic Tetraoxa Isophlorin Dimer
0365
Protect and Serve: Boron in Conjugated Polymers
0366
A Molecular Pickup

Metal-Catalyzed Asymmetric Synthesis and Stereoselective Reactions

z367
All PDFs of this category
0367
Aliphatic Amines Formed by Asymmetric Copper-Catalyzed Hydroamination
0368
Nickel-Catalyzed Asymmetric Allylic Alkylation
0369
Asymmetric Allylic Alkylation of Toluene-Chromium Complexes
0370
Palladium-Catalyzed Dehydrogenation Reaction
0371
Iridium-Catalyzed Borylative C–H Activation
0372
Nickel(II)-Catalyzed Synthesis of Chiral Tetrahydrofurans
0373
Asymmetric 1,3-Dipolar Cycloaddition with Inverse Electron Demand
0374
Asymmetric Hydrosilylation Catalyzed by Frustrated Lewis Pairs
0375
Nickel-Catalyzed Borylation of Benzylic Ammonium Salts
0376
Enantioselective Rhodium/Phosphoric Acid Catalyzed Assembly of Chromans
0377
Synthesis of α-Amino Ketones by Rhodium-Catalyzed Hydrogenation
0378
Rhodium-Catalyzed Asymmetric Hydrogenation of β-Amino Nitroolefins
0379
Diastereoselective Copper-Catalyzed Construction of Homoallylic Amines
0380
Iron-Catalyzed Diastereoselective Diazidation of Alkenes
0381
Kinetic Resolution of Phenylacetic Acids by Palladium-Catalyzed C–H Olefination
0382
Asymmetric Henry Reaction Catalyzed by Manganese Complexes
0383
Synthesis of Chiral Diarylmethanes by Copper-Catalyzed Allylic Arylation
0384
Rhodium-Catalyzed Asymmetric Ring Opening of Oxabenzonorbornadienes
0385
Rhodium-Catalyzed Asymmetric Si–H Insertion
0386
Azacyclic Nucleosides by Asymmetric Copper-Catalyzed [3+2] Cycloaddition
0387
Decarboxylative Coupling by Photoredox and Chiral Nickel Catalysis
0388
Enantioselective Rhodium-Catalyzed [2+2+2] Cycloaddition of 1,6-Enynes
0389
Asymmetric Cobalt-Catalyzed α-Amination of 1,3-Dicarbonyl Compounds
0390
Copper-Catalyzed Asymmetric Synthesis of Amino Acid Esters
0391
Copper-Catalyzed Divergent Addition Reactions of Nitrones
0392
Diastereoselective 1,3-Dipolar Cycloaddition Forming Spirocyclic Oxindoles
0393
Cycloisomerization of Dienynes by a Planar-chiral Gold(I) Complex
0394
Copper-Catalyzed Asymmetric Conjugate Addition
0395
Lithium(I)-Catalyzed Enantioselective Cyanosilylation of Ketones

Metal-Mediated Synthesis

z397
All PDFs of this category
0397
Palladium Cross-Couplings with a Silicon-Based Transfer Agent
0398
Copper-Catalyzed Borylcupration
0399
Silaborative Cyclization of 1,7-Enynes
0400
Oxyboration for the Preparation of 4-Borylated Isoxazoles
0401
Trifluoromethylthiolation of Heteroaryl Bromides
0402
Ring-Opening Reactions of Furans with Boronic Acids
0403
Copper-Catalyzed Cross-Coupling of Organoaluminum Reagents
0404
Tandem Nucleophilic Addition and Transesterification Reaction of Nitrones
0405
Enantioselective Assembly of Tertiary Stereocenters
0406
Enantioselective Allylic Substitution with a Diborylmethane Reagent
0407
Manganese-Catalyzed Synthesis of Isobenzofuranones
0408
Olefin-Directed Hydroboration of Allenes
0409
Asymmetric Vinylogous Michael Cascade
0410
Copper-Catalyzed Boron-Selective Cross-Coupling
0411
Chemoselective Homologation of Disulfides to Dithioacetals

Organo- and Biocatalysis

z413
All PDFs of this category
0413
Phosphoric Acid Catalyzed [4+2] Cycloadditions and Imino–Ene Reactions
0414
Chiral Phosphoric Acid Catalyzed Self-Redox Reaction of Indolines
0415
Enantioselective Aldol Reactions with Fluoroacetate Surrogates
0416
Biocatalytic Olefination of Aldehydes
0417
Enol Catalysis with α-Branched Ketones and a Michael Acceptor Surrogate
0418
Redox Esterification of α- and β-Substituted α,β-Unsaturated Aldehydes
0419
Diels–Alder Trapping of Photochemically Generated Hydroxy-o-Quinodimethanes

Polymer-Supported Synthesis

z421
All PDFs of this category
0421
Hydrogenolysis of Diaryl Ether C–O Bonds Using a Nickel/Carbon Catalyst
0422
A Recyclable Homochiral Polymer for Kinetic Resolution of (±)-Mefloquine
0423
Conversion of Alkenes into Nitriles by Using Cobalt-Doped ZSM-5 Zeolite
0424
Heterodimerization of Vinylarenes with 1,1-Diphenylethene by Snβ Zeolite
0425
Synthesis of α-Aminophosphonates with l-Cysteine Functionalized MNPs
0426
Multicomponent Synthesis of Pyrans with Boron Nitride Supported Fe3O4
0427
One-Pot Synthesis of Aminoindolizine Derivatives on Cu@Fe2O3 Nanoparticles
0428
Synthesis of Benzylbarbiturocoumarins Using a Silica-Supported Base
0429
Esterification of Oleic Acid by Using a Polymeric Acid Catalyst
0430
Conversion of Aldehydes into Nitriles Catalyzed by Silver Nanoparticles
0431
Mesoporous Aluminosilicate-Catalyzed Pummerer Reaction of Sulfoxides
0432
Silica-Supported Triptycene-Type Phosphine for Suzuki–Miyaura Coupling
0433
Compatible Linker for the Synthesis of Peptide o-Aminoanilides
0434
Asymmetric Addition of Et3Al to Aldehydes with Polymeric BINOL Ligands
0435
Magnetically Separable Carbapalladacycle for C–C Couplings

Erratum

436
Chung, L. Y. L.; Scott, J. P.: Synthesis of Omarigliptin