DOI: 10.1055/s-00000131

Synfacts

Ausgabe 05 · Volume 12 · Mai 2016 DOI: 10.1055/s-006-31580

Synform

A65
Zanda, Matteo: SYNFORM ISSUE 2016/05

Synthesis of Natural Products and Potential Drugs

z437
All PDFs of this category
0437
Syntheses of (+)-Grandilodine and (+)-Lapidilectine B
0438
Total Synthesis of Axinellamines A and B
0439
Synthesis of TP-2758
0440
Synthesis of K777
0441
Synthesis of (±)-Hippolachnin A
0442
Synthesis of a P2X7 Inhibitor
0443
Synthesis of (R)-(–)-Thiazesim
0444
Synthesis of (±)-Naupliolide
0445
Synthesis of (–)-Alstoscholarisine A
0446
Total Syntheses of Conidiogenone, Conidiogenone B, and Conidiogenol
0447
Synthesis of Birinapant
0448
Synthesis of Aliskiren
0449
Synthesis of PF-04995274
0450
Synthesis of a TRPV1 Antagonist
0451
Synthesis of (–)-Haliclonin A

Synthesis of Heterocycles

z453
All PDFs of this category
0453
Multicomponent Diastereoselective Synthesis of Tetrahydropyridines in Aqueous Micelles
0454
Reductive Fischer Indole Synthesis from N-Aryl Conjugated Hydrazones
0455
Stereocontrolled Late-Stage Remote Arylation of Bioactive Saturated N-Heterocycles
0456
Imidazopyridines by SNAr Addition of Metalated Isonitriles to 2-Chloro Heterocycles
0457
Synthesis of Fluorinated Indoles by Oxidative Dearomatization of Anilines
0458
DDQ-Promoted C–H Activation Approach to Pyrrolidine Alkaloids
0459
SN2′/SNV Reactions in the Synthesis of 2-Fluoro-2-pyrrolines
0460
Synthesis of Medium-Ring S,N-Heterocycles Using a Dithiadiazocane
0461
Synthesis of Strained Heterocycles by Flow Photochemistry
0462
Rhodium-Catalyzed Synthesis of Indoles from Imidamides and Diazo Keto Esters
0463
Palladium-Catalyzed Synthesis of Difluoromethylthiolated Heterocycles
0464
Photoredox Synthesis of 3,3-Difluoroindol-2-ones
0465
Ligand-Free Palladium-Catalyzed Synthesis of Carbazoles

Synthesis of Materials and Unnatural Products

z467
All PDFs of this category
0467
Bifunctional Perfluoroalkyl Building Blocks
0468
Tossing the Extra Carbon
0469
Alkaline Stable Anion Exchange Membrane
0470
Ladder-Type Thienoacenes Based On Benzo-[1,2-b:4,5-b′]dithiophene
0471
Back on the Chain Gang! (Poly)imidiazolium-Based Ionic Liquids
0472
Optical Barrel Rolls with X-Wing Paracyclophanes
0473
Anthraphane: A D3h-Symmetric Anthracene-Based Propeller
0474
Pucker Up to Diaminopentacenes
0475
N-Heteroacenes: Ball-Milling out!
0476
Furantastic! Polyfurans via Catalyst-Transfer Polymerization
0477
Preparation of Tetrahedral Cages from Simple Tritopic Precursors
0478
Twisted Truxene Dimer and Trimer

Metal-Catalyzed Asymmetric Synthesis and Stereoselective Reactions

z479
All PDFs of this category
0479
Zinc-Catalyzed Asymmetric Mannich Reaction Forming β-Amino Ketones
0480
Asymmetric Intramolecular Metallo-Ene Reaction
0481
Rhodium-Catalyzed Enantioselective Cycloisomerization to Cyclohexenes
0482
Iridium-Catalyzed Transfer Hydrogenation of 1,10-Phenanthrolines
0483
Palladium-Catalyzed Enantioselective Synthesis of α-Amino Phosphonates
0484
Iridium-Catalyzed Asymmetric Hydroxymethylation
0485
Zinc-Catalyzed Alkynylation with Terminal Ynamides
0486
Asymmetric Copper-Catalyzed Allylation of Azoles
0487
Z-Selective C–H Arylation of Unsubstituted Acrylamide Derivatives
0488
Rhodium-Catalyzed Enantioselective Synthesis of Chiral Tribenzothiepins
0489
Iridium-Catalyzed Chemo- and Stereoselective Dearomatization Reaction
0490
Gold(I)/Chiral Tertiary Amine Catalyzed Synthesis of Oxindoles
0491
Catalyst-Controlled Cycloadditions of Vinyl Aziridines and Alkynes
0492
Zinc-Catalyzed Diastereoselective Hydrosilylation of N-(tert-Butylsulfinyl)imines
0493
Asymmetric α-Addition of γ-Butyrolactam to Ketimines
0494
Rhodium-Catalyzed Diastereoselective Hydroalkylation of Dienes
0495
Transfer Hydrogenation of Ketones by Iridium(III) with Metal Centrochirality
0496
Rhodium-Catalyzed Asymmetric Synthesis of Silicon-Bridged Arylpyridinones
0497
Rhodium-Catalyzed Asymmetric Synthesis of Spirocyclic Sultams
0498
Rhodium-Catalyzed Asymmetric Hydrogenation of α-Dehydroamino Ketones
0499
Enantioselective Synthesis of Dihydroquinolines by Rhodium(I) Catalysis
0500
A Chiral Disulfoxide Ligand for the 1,2-Addition of Arylboroxines to Imines
0501
Nickel-Catalyzed Allylborylation via Transposition of Alkenyl Boronates
0502
Asymmetric Epoxidation Catalyzed by a Manganese Aminopyridine Complex
0503
Diastereoselective Copper-Catalyzed 1,2-Addition to N-tert-Butanesulfinyl Aldimines
0504
Asymmetric Addition of Arylboroxines to Aryl Ketones by Rh(I) Catalysis
0505
Asymmetric Hydrogenation of Cyano-Substituted Acrylate Esters
0506
Copper-Catalyzed Asymmetric Synthesis of Pyrrolo[2,1-a]isoquinolines
0507
Asymmetric Ruthenium-Catalyzed Allylic Alkylation of Silyl Enolates

Metal-Mediated Synthesis

z509
All PDFs of this category
0509
Palladium-Catalyzed Cross-Couplings with HandaPhos
0510
Synthesis of Substituted Allenes through Iron-Catalyzed Cross-Coupling
0511
Asymmetric Fukuyama Cross-Coupling of Racemic Benzylic Zinc Reagents
0512
Hydroboration and Dihydrocoupling Catalyzed by an Aluminum Dihydride
0513
Copper-Promoted Nitrogen Transfer of Cyanide to Aldehyde
0514
Trifluoromethylation of Arynes
0515
Difluoromethylation of Aryl Halides
0516
One-Pot Synthesis of 3,5-Diarylpyridines
0517
Nickel-Catalyzed Aryl–Alkyl Cross-Coupling
0518
Nickel-Catalyzed Negishi Cross-Couplings
0519
Stereodefined Tetrasubstituted Olefins
0520
Synthesis of β,β-Disubstituted Vinylboronates via Palladium 1,4-Migration
0521
Metallacycle-Mediated Coupling of Cyclopropenes with Alkynes
0522
Alkynylation of Alkylboronic Esters
0523
Nickel-Catalyzed Four-Component Couplings with Alkylfluorides

Organo- and Biocatalysis

z525
All PDFs of this category
0525
A Silylated C–H Acid Catalyst for Asymmetric Diels–Alder Reactions of Cinnamates
0526
Diol-Catalyzed Enantioselective Diboration of Alkenes
0527
Hypervalent Iodine-Catalyzed Dimerization of Styrenes
0528
Organocatalytic Asymmetric Mannich Reaction through Hydrogen Bonding
0529
Efficient Total Biosynthesis of Opiates by Using Engineered Escherichia Coli
0530
One-Pot Cascade of Synergistic Catalysis toward Tetrahydroisochromenes
0531
Hypervalent Iodine Catalyzed Oxidative Phenol Couplings
0532
Oxyallyl Cation Catalysis

Polymer-Supported Synthesis

z533
All PDFs of this category
0533
Graphene Oxide Promoted C–H Arylation of Benzene with Aryl Halides
0534
Photocatalyzed Selective Bromination of Aromatic Compounds
0535
Supported Copper Hydroxide Catalyst for Dehydrogenative N–S Cross-Coupling
0536
Double Carbonylation of Aryl Iodides Promoted by CTF-Supported Palladium
0537
Hydrogenation of Terminal Alkynes with a Palladium–Copper(II) Oxide Nanocomposite
0538
Palladium/Magnetite: Direct Arylation Reactions of Heterocycles
0539
Polymer-Supported Palladium Nanoparticles Catalyze the Suzuki–Miyaura Coupling
0540
Oxidative Amidation of Aldehydes Using Phosphotungstate Ionic Liquids
0541
Propargylamines by Using a Supported Copper(II)–Schiff Base Complex
0542
Ag- and Ru-Composites of Poly(PAr3) with Azo Groups for CO2 Conversion
0543
Direct Arylation of Indoles by Using Mesoporous Solid-Supported Palladium
0544
Direct C2-Vinylation of Thiophenes by Palladium on Zeolite Y Nanosheet
0545
Controlled Hydrogenation of Alkynes with HAP-Supported Pd@Ag
0546
N-Dealkylation/Carbonylation of Tertiary Amines by Using Palladium/Carbon