DOI: 10.1055/s-00000131

Synfacts

Issue 06 · Volume 12 · June 2016 DOI: 10.1055/s-006-31745

Synform

A79
Zanda, Matteo: SYNFORM ISSUE 2016/06

Synthesis of Natural Products and Potential Drugs

z547
All PDFs of this category
0547
Synthesis of an 11-β-HSD-1 Inhibitor via Asymmetric Methallylation
0548
Synthesis of Tofogliflozin
0549
Total Synthesis of Indole Alkaloids
0550
Synthesis of Rivaroxaban
0551
Synthesis of (+)-Piperarborenine B
0552
Synthesis of (–)-Mandelalide A
0553
Synthesis of CPI-0610
0554
Synthesis of MK-8831
0555
Asymmetric Synthesis of (+)-Phorbol
0556
Synthesis of Citalopram
0557
Synthesis of Escitalopram
0558
Asymmetric Synthesis of (–)-Nakadomarin A
0559
Synthesis of Cryptocaryol A
0560
Synthesis of Huprine Derivatives
0561
Synthesis of Daclatasvir by C–H Activation
0562
Synthesis of Lundurines A–C

Synthesis of Heterocycles

z563
All PDFs of this category
0563
Benzofurans from β-Pyrones and Phenols
0564
4-Bromo-1,2-dihydroisoquinolines from ortho-Triazolylbenzyl Bromides
0565
Lewis Base-Catalyzed Dynamic Kinetic Resolution of Azole Esters
0566
Synthesis of Indazoles by Oxidative N–N Bond Formation
0567
Benzoxazocindiones from Phthalic Acids and Cyclic Sulfamidates
0568
Palladium-Catalyzed Three-Component Synthesis of 2-Aroylbenzofurans
0569
Tetrahydronaphthyridines by a Radical Pictet–Spengler Reaction
0570
Pyrrolizidines and Indolizidines by Photooxidation of Furylalkylamines
0571
Enantioselective Synthesis of Piperidines from Pyridines
0572
Three-Component Synthesis of Pyrazolo [3,4-d]thiazolo[3,2-a]pyrimidines
0573
Triazole–Gold Catalyzed Approach to Substituted 2,3-Dihydrooxepines
0574
Copper-Catalyzed C–N Coupling/Madelung Synthesis of Indoles
0575
Direct Ketone Synthesis by Hetaryl Grignard Addition to Carboxylic Acids

Synthesis of Materials and Unnatural Products

z577
All PDFs of this category
0577
PET-RAFT + ROP = Copolymers!
0578
Coplanar Triply Linked 2H-Corrole Dimers
0579
All-Carbon Carbodicarbene
0580
Locked and Loaded!
0581
Inspiration via Hydroboration
0582
Oligo(thienylene-vinylene) by Deprotonative Cross-Coupling
0583
Azole-Fused B,N-Naphthalenes via Hydroboration
0584
C-Terminal Modification of Fully Unprotected Peptide Hydrazides
0585
Sterically Congested PAHs Based on a 1,7-Naphthodiyne Platform
0586
It’s an Alcohol, It’s a Lactide, It’s a Superelectrophile!
0587
Synthesis of High Electron Affinity Materials Using Aryl C–H Iodination
0588
Synthesis of A Newly Class of Si-Bridged π-Conjugated Compounds

Metal-Catalyzed Asymmetric Synthesis and Stereoselective Reactions

z589
All PDFs of this category
0589
Ruthenium(II)-Catalyzed Asymmetric Transfer Hydrogenation Reaction
0590
Iridium-Catalyzed Reverse Prenylation of Indole and Tryptophan Derivatives
0591
Palladium-Catalyzed Asymmetric Carboetherification of Dihydrofurans
0592
Pd-Catalyzed Enantioselective Alkene Aryloxyarylation through Oxopalladation
0593
Nickel-Catalyzed Asymmetric Propargyl Claisen Rearrangement
0594
Spiroketals and -aminals by Gold(I)/ Nickel(II) Asymmetric Relay Catalysis
0595
Scandium-Catalyzed Regio- and Enantioselective Bromoaminocyclization
0596
Iridium-Catalyzed Asymmetric C–H Alkylation of N-Sulfonylbenzamides
0597
Catalytic Asymmetric [3+2] Annulation through C–H Activation
0598
Palladium-Catalyzed Enantioselective Allylic Alkylation of CF3-Substituted Compounds
0599
Regio- and Stereoselective Pd-Catalyzed 1,3-Difunctionalization of Alkenyl Nonaflates
0600
Copper-Catalyzed trans-Hydroboration of Terminal Aryl Alkynes
0601
Pd-Catalyzed Asymmetric Aminomethylamination of Conjugated Dienes
0602
Enantioselective CuH-Catalyzed Hydroallylation of Vinylarenes
0603
Molybdenum Complex Catalyzed Z-Selective Cross-Metathesis
0604
Rhodium-Catalyzed Asymmetric Conjugate Addition of Arylboronic Acids to Enones
0605
Copper-Catalyzed Aminoboration of Alkylidenecyclopropanes
0606
Asymmetric Ir-Catalyzed Spirocyclization and Migration Forming Tetrahydro-β-Carbolines
0607
Enantioselective Copper(II)-Catalyzed Conjugate Addition
0608
Palladium-Catalyzed Multicomponent Carbonyl Allylation Reaction
0609
Iridium-Catalyzed Reductive Amination of Arylacetones
0610
Asymmetric Chromium-Catalyzed Dearomative 1,2-Addition
0611
Palladium-Catalyzed Three-Component Reaction for the Allylation of Aldehydes
0612
Cu-Catalyzed Asymmetric Synthesis of 3,4-Dihydro-2H-1,4-benzoxazines
0613
Asymmetric Copper-Catalyzed 1,4-Addition to β-Substituted Enones
0614
Asymmetric Indole Cyclization toward (–)-Aspidophylline A
0615
Rhodium-Catalyzed Stereoselective Synthesis of Isoindolines

Metal-Mediated Synthesis

z617
All PDFs of this category
0617
Suzuki Coupling of Heteroaryl Fluorosulfates
0618
Synthesis of Trimethylstannanes
0619
Enantioselective Arylation of Pyridine
0620
One-Pot, Modular Approach to Functionalized Ketones
0621
Spirocyclization via Hydroarylation of N–Ac Indoles
0622
Catalytic Asymmetric Addition of Organolithium Reagents
0623
Copper-Catalyzed 1,2-Additon of Dialkylzinc Reagents
0624
Diastereoselective Allylzincation of Nonracemic Imines
0625
Annulation/Arylthiolation Cascade with Arylboronic Acids
0626
Carbochlorination of Arylacetylene
0627
Copper-Catalyzed Aminoalkylations
0628
Suzuki–Miyaura Cross-Coupling Reactions of Aminopyrazoles
0629
Difluoroalkylation of Arylborons
0630
One-Pot Synthesis of Arylketones from Aromatic Acids
0631
Synthesis of Azoles Sulfides via Copper-Catalyzed Cross-Coupling

Organo- and Biocatalysis

z633
All PDFs of this category
0633
Direct Mannich-Type Reaction Using a Chiral Organosuperbase Catalyst
0634
Organocatalytic Kinetic Resolution of Sulfoximines with Enals
0635
Enzymatic Nitrene Transfer/Sigmatropic Rearrangement to Access Allylic Amines
0636
Asymmetric Ugi Reaction Catalyzed by a Chiral Phosphoric Acid
0637
Data Set Design for the Asymmetric Fluorination of Allylic Alcohols
0638
Biomimetic Photoorganocatalytic Chlorination of Arenes
0639
Enantioselective Synthesis of Silacyclopentanes
0640
NHC-Catalyzed Enantioselective Enamide−Aldehyde Cross-Coupling

Polymer-Supported Synthesis

z641
All PDFs of this category
0641
Doped Carbon Shell Catalysts for Oxidation of Alkanes
0642
Heterogeneous Photocatalyst for C–H Alkylation of Aliphatic Nitriles
0643
Sequential C–C Bond Formation via Allylic and Benzylic Boronic Acids
0644
Phosphonylation of Aryl Halides with a Palladium Complex on Fe(III) Oxide in Water
0645
Chemoselective Reduction of Nitroarenes on Platinum Nanoparticles
0646
Reusable Polyacid Catalyst for Oxidation of Sulfides and Allylic Alcohols
0647
Iron(III) Oxide Nanoparticle-Catalyzed Hydrogenation of Nitro Compounds
0648
Bisoxazoline–Palladium Composite-Catalyzed Suzuki–Miyaura Coupling
0649
A Gold-NP-Supported Organocatalyst for Asymmetric Aldol Reactions
0650
Copper(0)/Magnetite-Catalyzed Cyclization of Terminal Alkynes with Isocyanides
0651
Stabilized Ruthenium Nanoparticles for Oxidation and Hydrogenation Reactions
0652
Cobalt/Titania-Catalyzed Aerobic Oxidation of Alcohols and Alkanes
0653
Multistep Continuous-Flow Synthesis of Nitrogen-Containing Compounds
0654
Au–Cu Alloy Nanoparticles for Photocatalytic Reduction of Nitrobenzenes
0655
Synthesis of Chromene Derivatives Using PS-Supported PTSA
0656
Hydrogenation of Halonitrobenzene by Using a Platinum–Zinc Bimetallic Catalyst