DOI: 10.1055/s-00000131

Synfacts

Issue 07 · Volume 12 · July 2016 DOI: 10.1055/s-006-31955

Synform

A94
Zanda, Matteo: SYNFORM ISSUE 2016/07

Synthesis of Natural Products and Potential Drugs

z657
All PDFs of this category
0657
Synthesis of IPI-926
0658
Synthesis of (–)-Daphenylline
0659
Synthesis of (−)-Rubriflordilactone B
0660
Syntheses of Periconiasins A–E
0661
Synthesis of (–)-Terengganensine A
0662
Synthesis of AMG 337
0663
Synthesis of a BACE1 Inhibitor
0664
Total Synthesis of Integrastatin B
0665
Total Synthesis of (–)-Strychnopivotine
0666
Synthesis of (–)-Cannabimovone

Synthesis of Heterocycles

z667
All PDFs of this category
0667
Synthesis of 6-Amino-2,3-dihydro-4-pyridones from Homoallylamines
0668
O-Benzoylhydroxylamine-Promoted Electrophilic Amination of Alkenes
0669
Azaarenes by Palladium-Catalyzed α-Arylation of Ketimines with Aryl Sulfides
0670
Three-Component Aryne-Mediated Synthesis of Dibenzooxazonines
0671
Regioselective Preparation of Tetrazoles without the Use of Azides
0672
Pd-Catalyzed Selective 2-Amination of 2,4-Dichloro-5-(trimethylsilyl)pyrimidine
0673
Three-Component Synthesis of Benzo[e]pyrazolo[1,5-c][1,3]thiazines
0674
Pyrrolidines by Coupling of Olefins with β-Aminoethyl Trifluoroborates
0675
Regiodivergent Synthesis of Dihydroquinolines and Chromenes
0676
Synthesis of 6-Perfluoroalkylated Bicyclic 1,2,3-Triazolo-1,4-oxazines
0677
Tricyclic Indoles by Sequential Friedel–Crafts/Allylic Amination Reactions
0678
Synthesis of 2H-Indazole-Fused Tetrahydroisoquinolinoquinoxalines
0679
Ir-Mediated Cascade Approach to Chiral Indole-Annulated Medium-Sized Rings
0680
Polyfunctional Alkenyl Organometallic Reagents for Heterocycle Synthesis

Synthesis of Materials and Unnatural Products

z681
All PDFs of this category
0681
Some Non-Planar Polycyclic Aromatic Hydrocarbons
0682
Synthesis of Tetraphenylenes by Palladium-Catalyzed C–H Functionalization
0683
Doubling Down on Diamines for Direct Arylation Polymerization
0684
Fantastic Four-Membered Rings
0685
Mobile Hydroxide Ion Shuttles
0686
Going Retro with Ester-Sulfonyl Poly(imides)
0687
CNTs and Au–Pd Alloys – Amine Combination
0688
Ring It Up
0689
Stitching Heterocycles into Buckyballs
0690
Boron-Fused Double Helicenes
0691
A New Route to Polymers with NBN Backbone
0692
First Synthesis of an Oxygen-Bridged Planarized Triphenylborane

Metal-Catalyzed Asymmetric Synthesis and Stereoselective Reactions

z693
All PDFs of this category
0693
Gd-Catalyzed Photocycloaddition of Aryl Cyclopropyl Ketones to Alkenes
0694
Asymmetric Reductive Coupling of Alkenes with Carboxylic Anhydrides
0695
Stereodivergent Synthesis of Chiral Amino Alcohols by Copper(I) Catalyst
0696
Copper(I)-Catalyzed Asymmetric Dearomatization of Indole Acetamides
0697
Ir(I)/NHC-Catalyzed Asymmetric Intramolecular Allylic Amination of Indoles and Pyrroles
0698
Asymmetric C–H Functionalization of Electron-Deficient Methyl Groups
0699
Synthesis of Chiral Cyclopropylamines by Rhodium(I) Catalysis
0700
Rhodium-Catalyzed Enantioselective Synthesis of Allylic Amines
0701
Ru-Catalyzed Synthesis of Oxazolidin-2-ones by Hydrogen Transfer
0702
Asymmetric Rhodium-Catalyzed 1,2- and 1,4-Addition Reactions
0703
Ru-Catalyzed Asymmetric Propargylation through Transfer Hydrogenation
0704
Copper-Catalyzed Asymmetric Synthesis of 3-Alkynyl-3-hydroxyoxindoles
0705
Enantioselective [2+2] Cycloaddition of Alkynones to Silyl Enol Ethers
0706
Magnesium-Catalyzed Enantioselective Synthesis of Oxazoles
0707
Catalytic Enantioselective Synthesis of Halocyclopropanes
0708
Access to Chiral Alkyl-Aryl-Substituted Secondary Amines
0709
Pd-Catalyzed Carboamination Reaction for the Synthesis of Cyclic Sulfamides
0710
Asymmetric Addition of P-Chiral H-Phosphinates to Aldehydes
0711
Enantiodivergent Gold(I)-Catalyzed Hydroazidation and Hydroamination of Allenes
0712
Ir-Catalyzed Asymmetric Hydrogenation of β,β-Disubstituted Nitroalkenes
0713
Asymmetric [3+2] Cycloaddition through Desilylation Activation
0714
Regio- and Enantioselective Hydrovinylation of Vinylarenes
0715
Synthesis of Chiral Allenes by Rhodium(I) Catalysis
0716
Rhodium-Catalyzed Cycloaddition of Phenyldiynes with Nitriles
0717
Catalytic Asymmetric Allylic Substitution Reactions
0718
Silver(I)-Catalyzed Atroposelective Desymmetrization of N-Arylmaleimide
0719
Rh-Catalyzed Vinylogous Asymmetric Ring-Opening of Oxabicycles
0720
Cu-Catalyzed Desymmetrization of meso-α,α′-Diazido Alcohols
0721
Ir-Catalyzed Sequential Asymmetric Allylic Alkylation/Cope Rearrangement
0722
Asymmetric Hydrogenation of Unprotected β-Enamino Phosphonates

Metal-Mediated Synthesis

z723
All PDFs of this category
0723
Nickel-Catalyzed Decarboxylative Alkyl–Alkyl Cross-Coupling
0724
Cobalt-Catalyzed Multicomponent Coupling Reactions with Alkynes
0725
Cascade Reaction for the Synthesis of Cyclooctatetraenes
0726
Nickel-Catalyzed Borylation of Polyfluoroarenes
0727
Aryl Ether Alkylation
0728
One-Pot Sulfoxide Synthesis
0729
Stereoselective Silylzincation of Alkynes
0730
Iron-Catalyzed Stereoselective Cross-Coupling
0731
Nickel-Catalyzed Suzuki–Miyaura Biaryl Synthesis
0732
Chemoselective Ketone Synthesis
0733
Allyl Zinc-Brook Rearrangement
0734
Chemoselective Carboxylic Acid Aldol Reaction
0735
Nickel-Catalyzed Cross-Coupling Reactions from Amides
0736
Asymmetric Dearomatization Reaction of β-Naphthols
0737
Ring Opening of Cyclopropanated 7-Azabenzonorbornadienes

Organo- and Biocatalysis

z739
All PDFs of this category
0739
Enantioselective Formation of Quaternary Carbons by Radical Conjugated Addition
0740
Catalytic Diastereoselective Difluorination of Alkenes
0741
Biocatalytic syn-Selective Aldol Reaction of Fluoropyruvate
0742
Desymmetrization of Cyclohexanones by Enantioselective α-Arylation
0743
Trifunctional Squaramide Catalyzed Enantioselective Henry Reaction
0744
Development of a Binaphthyl-Based Chiral DMAP Catalyst
0745
Photobiocatalytic Reduction of α,β-Unsaturated Enones and Amides
0746
Organocatalytic Transformation of Epoxides into Thiiranes
0747
Asymmetric Catalysis with CO2: The Direct α-Allylation of Ketones
0748
Lewis Acid Catalyzed Formal [3+2] Cycloaddition of Cyclopropyl Acetals
0749
Enantioselective Organocatalytic [4+2] Cycloaddition on Water

Polymer-Supported Synthesis

z751
All PDFs of this category
0751
Hydrosilylations Catalyzed by Iron-Doped Metal–Organic Layers
0752
Aerobic Oxidation of Amines to Nitriles Catalyzed by Supported Co3O4
0753
Selective Cleavage of Carbon–Carbon Bonds with Palladium/Carbon
0754
Coupling of Aryl Iodides with Triarylbismuthines on Supported Pd Complex
0755
Oxidative Dehydrogenative Cross-Coupling of Aryl Amines on Rh/C
0756
Friedel–Crafts Alkylation of Indoles by Using Supported Imidazolidinones
0757
Iridium/Molybdenum Carbide Catalyzed Chemoselective Hydrogenation of Enals
0758
Platinum–Molybdenum Oxide/Titania-Catalyzed Reduction of Sulfoxides
0759
A Polymer-Supported Phosphazene Catalyst for Phospha-Michael Additions
0760
Direct Olefination of Alcohols with Sulfones on Pt/C Nanoparticles
0761
Pd/Metal-Organic Framework Catalyzed Selective C–H Halogenation
0762
Synthesis of 4-Arylcoumarins by Using Palladium Oxide/Magnetite
0763
Controlled Hydrogenation of Alkynes by Ammonium Formate on Gold/Titania
0764
Three-Component Coupling of Amines, Aryl Iodides, and CS2 with CuO/Fe3O4
0765
Synthesis of Tetrazoles with Copper(II) on l-Arginine-Functionalized Fe3O4–SiO2
0766
Sonogashira Reaction on a Polymer-Supported Palladium Nanocatalyst