DOI: 10.1055/s-00000131

Synfacts

Issue 09 · Volume 12 · September 2016 DOI: 10.1055/s-006-32295

Synform

A126
Zanda, Matteo: SYNFORM ISSUE 2016/09

Synthesis of Natural Products and Potential Drugs

z883
All PDFs of this category
0883
Synthesis of Millingtonine
0884
Synthesis of a MK-8876 Fragment
0885
Total Synthesis of (−)-Communesin F
0886
Organocatalytic Synthesis of Enantiopure 2H- and 3H-Pyrroles
0887
Synthesis of Letermovir by an Asymmetric Aza-Michael Reaction
0888
Synthesis of (+)-SCH 351448
0889
Synthesis of (±)-Integrifolin
0890
Synthesis of Lotronex through anti-Azacarboxylation of a 2-Alkynylaniline
0891
Synthesis of a PDE4 Inhibitor by C–H Activation
0892
Synthesis of Calophyline A
0893
Total Synthesis of (±)-Aplydactone
0894
Synthesis of the CHK1 Inhibitor MK-8776
0895
Synthesis of Thailanstatin A
0896
Formal Synthesis of HIV Integrase Inhibitor BI 224436

Synthesis of Heterocycles

z897
All PDFs of this category
0897
Synthesis of Palbociclib: An SNAr Reaction on a Kilogram Scale
0898
Pyrimido[4,5-d]pyridazines by the Reaction of Pyrimidines with Tetrazines
0899
Four-Component Synthesis of 1-Pyrimidin-2-yl-3,4-dihydropyridin-2(1H)-ones
0900
Synthesis of Trifluoromethylated Isoxazoles by [2+3] Cycloaddition
0901
Synthesis of Azabicycloalkanes by Gold(I)-Catalyzed Amination of Ynones
0902
Microwave-Assisted Synthesis of 1-Arylnaphtho[2,1-b]furans
0903
Regiocontrolled Synthesis of Benzo-Fused (Hetero)aromatics from Dihydrofuran Acetals
0904
Copper(I)-Promoted Synthesis of Halogenated Tetrahydrothiophenes
0905
Synthesis of Pyrrolidines and Piperidines with Tin Amine Reagents
0906
Synthesis of Oxindoles from α,β-Unsaturated Amides and Aldehydes
0907
Rhodium-Catalyzed Synthesis of Fused Heterocycles
0908
Synthesis of Functionalized 1,4-Oxazines by Activation of Diazoenals
0909
Functionalized Isoquinolines by Rh(III)-Catalyzed C–H Conjugate Addition
0910
Synthesis of 2-Quinolinones by Lactamization of 2-Alkenylanilines with CO2

Synthesis of Materials and Unnatural Products

z911
All PDFs of this category
0911
Molecular Knot Inducing Allosteric Control of Catalysis
0912
Let the Acid Do the Job
0913
Oligomeric Ferrocene Rings
0914
First Experimental Evidence for the Formation of the Cyclic Carbon Dioxide Trimer
0915
Neutral Diboron Analogues of Archetypal Aromatic Species by Cycloaddition
0916
Five- and Seven-Membered Rings Containing Isomeric Pentacene
0917
Combinations of 1,2- and 1,4-Additions to an Acene Dione
0918
Between Diamond and Graphene
0919
A Creative Route to Perfluororubrene
0920
Embedding Nitrogen Atoms in Polymers to generate n-Type FETs
0921
One-Pot Synthesis of Complex Polymers via Copper Catalysis
0922
Palladium-Catalyzed Annulation of Internal Alkynes to Ullazines

Metal-Catalyzed Asymmetric Synthesis and Stereoselective Reactions

z923
All PDFs of this category
0923
Copper-Catalyzed Asymmetric Nucleophilic Addition to Ketones
0924
Asymmetric Hydroarylation of Vinylarenes with CuH and Pd Catalysts
0925
Copper-Catalyzed Asymmetric [4+1] Annulation of Sulfur Ylides
0926
Kinetic Resolution by Asymmetric Amide Addition
0927
Neodymium-Catalyzed [3+2] Cycloaddition of Aziridines and Aldehydes
0928
Iridium-Catalyzed Asymmetric Hydroalkynylation of Enamides
0929
Rhodium-Catalyzed Enantioselective Macrolactonization
0930
Rhodium-Catalyzed E-Selective Hydro-formylation of Alkynes
0931
Noncovalent Ion Pair Interaction in Rhodium-Catalyzed Asymmetric Hydrogenation
0932
Enantioselective Synthesis of α-Allyl-α-Aryl-cyclopentanones
0933
Nickel-Catalyzed Asymmetric C-Acylation of Lactams
0934
Enantio- and Diastereoselective Addition of 1,1-Diborylalkanes to α-Keto Esters
0935
Rhodium-Catalyzed Asymmetric Hydrogenation of Acroleins
0936
Asymmetric Desymmetrization of meso-Epoxy Diketones
0937
Asymmetric Rearrangement of N-Acylaziridines to Oxazolines
0938
Iridium-Catalyzed Asymmetric Hydrogenation of Simple Ketones
0939
Enantioselective C–H Activation for the Formation of Chiral Isochromans
0940
Synthesis of Chiral Tryptamines under Cu(I) Catalysis
0941
Rhodium-Catalyzed Asymmetric Radical Amination Activated by Visible Light
0942
Asymmetric Benzylic Alkylation of Active Methylene Compounds
0943
Nickel-Catalyzed Asymmetric Synthesis of Imidazolines
0944
Asymmetric Hydroformylation by Rh-BIBOP Complex
0945
Supported Copper(II) Catalysts for the Asymmetric Henry Reaction
0946
Rhodium-Catalyzed Synthesis of trans-Dimethylenecyclobutane-1,2-diamines
0947
Iridium-Catalyzed Asymmetric Allylation of Fluorinated Methylene Derivatives
0948
Copper-Catalyzed Aerobic Asymmetric Cross-Dehydrogenative Coupling
0949
Copper-Catalyzed Cycloaddition for the Synthesis of Chiral Bicycloprolines
0950
Cyclization of Dearomatized Alkylidene Dihydropyridines
0951
Copper-Catalyzed Cascade Aldol-Cyclization Reaction
0952
Catalytic Asymmetric [2+2+2] Cycloaddition

Metal-Mediated Synthesis

z953
All PDFs of this category
0953
Palladium-Catalyzed Alkynylation
0954
Synthesis of 1,3-Dienes
0955
Direct Cross-Couplings of Propargylic Diols
0956
Ruthenium-Catalyzed Hydroboration of Pyridines
0957
anti-Carbometalation of Alkynes via Alkenylnickel Intermediates
0958
O-Acylation of Alcohols and Phenols by Using Cp2TiCl
0959
Copper-Catalyzed Isomerization of α-Hydroxy Ynamides
0960
Oxidative β,β-Fluoroarylation
0961
Nickel-Catalyzed Borylation
0962
Enantioselective Construction of Quaternary Carbon Stereocenters
0963
Stereoselective Cycloaddition of Nitrone Ylides with Aldehydes using n-BuLi
0964
Oxidative Cyclization of Diarylalkynes to Indoloindole Derivatives
0965
Regioselective Functionalization of 2-Phenyltetrahydropyran
0966
Oxyarylation of Furans
0967
Direct Amidation of Unprotected Amino Acids

Organo- and Biocatalysis

z969
All PDFs of this category
0969
Single-Step Enzymatic Synthesis of β-Methyltryptophans
0970
Brønsted Acid Catalyzed Synthesis of Chiral Tetrahydroacridines
0971
Brønsted Acid Catalyzed Transfer Hydrogenation of Imines and Alkenes
0972
Chiral NHC-Catalyzed Benzoin Reaction Permits a Dynamic Kinetic Resolution
0973
Enantioselective Intermolecular [2+2] Photocycloaddition
0974
Conformational Control of Thiourea Catalysts for Improved Performance
0975
Enantioenriched γ-Butenolides via Chiral Electrophilic Selenium Catalysis
0976
Alkynylogous Mukaiyama Aldol Reaction

Polymer-Supported Synthesis

z977
All PDFs of this category
0977
Photocatalytic Sonogashira Coupling on Polymeric Pyrazine–CuO Nanoparticles
0978
Oxidation of α-Hydroxy Ketones by Dendrimer-Stabilized Gold Nanoclusters
0979
Supported Gold Nanoparticles Catalyzed the α-Oxygenation of Amines to Amides
0980
Hydrogenation of Nitro Compounds by Using a Porous Carbon–Cobalt Catalyst
0981
Oxidative α-Cyanation of Tertiary Amines by a Gold Complex on Magnetic Nanoparticles
0982
Sonogashira Coupling by Using a Mesoporous Carbon Nitride–Pd Catalyst
0983
C–C Bond Formation by Using Magnetite-Supported Pd(II)–β-Cyclodextrin
0984
Dehydrogenative Cyclization of ortho-Alkenylphenols by Using Pd/C
0985
Copper-Catalyzed Oxidation of Benzaldehydes to Benzonitriles
0986
Transamidation Catalyzed by Fe3O4 Nanoparticles
0987
Controlled Hydrogenation of Nitrobenzenes to Anilines on RhIn/SiO2
0988
Aminocarbonylation of 1-Alkynes by Using Palladium/Carbon
0989
Pd-Catalyzed N-Methylation of Amines with Paraformaldehyde and Calcium Hydride
0990
Asymmetric Aldol Reaction Catalyzed by a Polystyrene-Supported Triazolylproline
0991
Synthesis of 4(3H)-Quinazolinones by Using a CuCO3–K2CO3 Nanocomposite
0992
Synthesis of Phthalazine Derivatives with a Supported Organocatalyst
0993
Silver Iodide Catalyzed Synthesis of Carbo-nates from Propargylic Alcohols and CO2

Erratum

995
Kalaitzakis, D.; Triantafyllakis, M.; Sofiadis, M.; Noutsias, D.; Vassilikogiannakis, G.: Pyrrolizidines and Indolizidines by Photooxidation of Furylalkylamines
996
Tian, Q.; Bai, J.; Chen, B.; Zhang, G.: Asymmetric Chromium-Catalyzed Dearomative 1,2-Addition
997
Zhu, D.; Ma, J.; Luo, K.; Fu, H.; Zhang, L.; Zhu, S.: Enantioselective Rhodium-Catalyzed C−H Insertion of Carbenes