DOI: 10.1055/s-00000131

Synfacts

Issue 02 · Volume 13 · February 2017 DOI: 10.1055/s-007-33277

Synform

A18
Zanda, Matteo: SYNFORM ISSUE 2017/02

Synthesis of Natural Products and Potential Drugs

z0115
All PDFs of this category
0115
Divergent Syntheses of Aflavazole and 14-Hydroxyaflavinine
0116
Synthesis of MK-8666
0117
Total Synthesis of a Ladderane Phospholipid
0118
Total Synthesis of (–)-Nakadomarin A
0119
Synthesis of BMS-741672
0120
Synthesis of (–)-Cycloclavine
0121
Synthesis of Epothilone D
0122
Synthesis of Verubecestat
0123
Synthesis of a TRPV3 Antagonist
0124
Synthesis of (+)-Haplophytine
0125
Synthesis of (±)-Berkeleyone A
0126
Asymmetric Synthesis of an 11β-HSD-1 Inhibitor

Synthesis of Heterocycles

z0127
All PDFs of this category
0127
Palladium-Catalyzed Synthesis of Six- and Seven-Membered-Ring Heterocycles
0128
Enantioselective Organocatalytic Synthesis of Benzo-Fused Acetals
0129
Palladium-Catalyzed Carbonylation of Aliphatic Amines To Form β-Lactams
0130
Stereodivergent Diels–Alder Route to Bicyclic Lactones
0131
Lewis-Acid-Mediated Multistep Synthesis of (–)-Mersicarpine
0132
Direct Nickel-Catalyzed Synthesis of Oxaborins from Benzofurans
0133
Palladium-Catalyzed Synthesis of Cyclopropyl-Fused Azacycles
0134
Synthesis of Pyrrolopyridinones by the Ugi Reaction
0135
Synthesis of Acylated Benzimidazoles with Copper Catalysts
0136
Synthesis of 3-Cyano-1H-indolo-2′-deoxy-ribonucleosides
0137
Synthesis of Polyhydroxyindolizidines from Carbohydrates
0138
Nickel-Catalyzed Trifluoromethylation of Electron-Rich Heteroarenes
0139
Synthesis of 3,4-Dihydroquinazolinones from 2-Aminobenzaldehydes
0140
Synthesis of 6-Phosphorylated Phenanthridines
0141
Synthesis of Pyrroloquinolinones from Donor–Acceptor Cyclopropanes

Synthesis of Materials and Unnatural Products

z0143
All PDFs of this category
0143
Electrochromism of Porous Network Thin Films
0144
Nonplanar Polycyclic Aromatic Hydrocarbons
0145
Toward Automated Oligo[n]rotaxanes
0146
Photoredox Activation of SF6 for Fluorination
0147
A Facile Approach to DTT
0148
A Negotiation between Different Nucleophiles in SNAr Reactions
0149
From 1,4-Dibromo-bis-alkynes to Heptacyclic Heteroacenes in One Step
0150
Thiophene-Bridged Carbazole-Based Diporphyrin
0151
Aryl(triethyl)silanes for Biaryl and Teraryl Synthesis by Copper(II) Catalysis
0152
Unsymmetric Dibenzopentalenes
0153
Bis-Lactam as Acceptor
0154
Azaanthracenes via Inverse Electron-Demand Diels–Alder Reaction

Metal-Catalyzed Asymmetric Synthesis and Stereoselective Reactions

z0155
All PDFs of this category
0155
Enantioselective α-Arylation of α-Fluoroketones
0156
Enantioselective Copper-Catalyzed Cyanotrifluoromethylation
0157
Enantioselective Rhodium-Catalyzed α-Allylation of Aldehydes
0158
1,3-Dipolar Cycloaddition of Alkenyl Arenes with Azomethine Ylides
0159
Enantioselective Coupling of Diazoalkanes with Terminal Alkynes
0160
Catalytic Asymmetric α-Vinylation of β-Keto Amides/Esters
0161
Enantioselective Desymmetrization of Cyclohexadienones
0162
Iridium-Catalyzed Asymmetric Hydrogenation of Alkenoic Acids
0163
Palladium-Catalyzed Asymmetric Benzylic C–H Arylation of Amines
0164
Cobalt-Catalyzed Asymmetric Hydrosilylation of Alkynes
0165
Molybdenum-Catalyzed Deoxygenation of Epoxides
0166
Asymmetric Hydrogenation of Lactones through Dynamic Kinetic Resolution
0167
Iridium-Catalyzed Asymmetric Allylic Alkylation of β-Keto Esters
0168
Ligand Effect on Diastereoselectivity in Suzuki–Miyaura Coupling
0169
Copper-Catalyzed Propargylation of Cyclic Aldimines
0170
Enantioenriched Borylalkanes by Copper-Catalyzed Hydroallylation
0171
Regio- and Enantioselective Palladium-Catalyzed Hydroesterification
0172
Asymmetric Cross-Coupling with Organoaluminum Reagents
0173
Iridium-Catalyzed Stereoselective Hydrogenation of α-Alkyl β-Keto Esters
0174
Catalytic Asymmetric Cycloisomerization and Parallel Kinetic Resolution
0175
CF3-Substituted Pyrrolidines through Cycloaddition of Azomethine Ylides
0176
Palladium-Catalyzed Decarboxylative Asymmetric [4+2] Cycloaddition
0177
Rhodium-Catalyzed Asymmetric Hydroacylation of Trisubstituted Alkenes
0178
Samarium-Catalyzed Asymmetric Synthesis of Aminocyclopropanes
0179
Rhodium-Catalyzed Enantioselective Cascade Cyclopropanation
0180
Palladium-Catalyzed Asymmetric Alkynylation of Axially Chiral Biaryls
0181
Enantioselective Synthesis of α-Mercapto-β-Amino Esters
0182
Enantioselective Narasaka–Heck Cyclization

Metal-Mediated Synthesis

z0183
All PDFs of this category
0183
Direct Primary Amination and Hydroxylation of (Hetero)arylmetals
0184
Synthesis of Tertiary Aminocyclopropanes
0185
Cross-Coupling of O-Based Electrophiles
0186
Synthesis of 3-Aminoaryne Precursors
0187
Synthesis of β-Alkoxy- and β-Aryloxyacrylates
0188
Directed Arylation and Alkenylation of C(sp3)–H Bonds
0189
Synthesis of Aryl Amines by Metal-Free C–N Coupling
0190
N-Arylation of 2-Imidazolines
0191
Radical-Type Cross-Coupling Reactions
0192
Suzuki–Miyaura Cross-Coupling of Triazolopyrimidines
0193
Multicomponent Synthesis of β-Hydroxy- and β-Aminocarbonyl Compounds
0194
Borylative Cyclization for the Formation of Benzofurans and Benzothiophenes
0195
Nickel-Catalyzed CO2 Rearrangement
0196
Selective Addition of Alkyl Grignard Reagents to Pyridine-N-oxides
0197
Silaboration of Oxetanes and Unactivated Epoxides

Organo- and Biocatalysis

z0199
All PDFs of this category
0199
Asymmetric Enzymatic Carbon–Silicon Bond Formation
0200
Phosphoric Acid Catalyzed Asymmetric Synthesis of SPINOL Derivatives
0201
Catalytic Enantioselective Vinylogous Pinacol Rearrangement
0202
Construction of Adjacent Quaternary Stereocenters
0203
Annulation of Donor–Acceptor Cyclobutanes with N-Heterocyclic Carbenes
0204
Photocatalytic Hydrodefluorination Promoted by π-Hole–π Interactions
0205
Hydrogen-Bonding Catalysis with Sulfonium Salts
0206
Catalytic Asymmetric Synthesis of C2-Symmetric Secondary Amines
0207
Transaminase-Catalyzed Enantioselective Synthesis of Piperidines
0208
ortho-Selective Chlorination of Anilines

Polymer-Supported Synthesis

z0209
All PDFs of this category
0209
Alcohol Oxidation with Ionic Liquid Supported IBX Generated in situ
0210
Reduction of 4-Nitrophenol with Porphyrin Polymer Supported Gold
0211
Azide–Alkyne Cycloaddition with a Melanin-Supported Copper(I) Catalyst
0212
MOF-Catalyzed N-Arylation of Heterocycles with Aryl Iodides
0213
Knoevenagel Condensation Catalyzed by Nickel Ferrite Nanoparticles
0214
Asymmetric Ethylation of Aryl Aldehydes with a PEG-Supported Chiral Ligand
0215
A Cr(salen)-Based Metal–Organic Framework as a Chiral Lewis Acid Catalyst
0216
Direct Oxidative C(sp3)–H/N–H Coupling on a Copper/Metal–Organic Framework
0217
Preparation of β-Enaminones with Copper(II) Oxide Nanoparticles
0218
C–C Bond Formation by Using a Supported Palladium–Schiff Base Complex
0219
Synthesis of Propargylamines on Thiolate-Protected Gold Nanoclusters
0220
Oxidation and Reduction of Olefins on Copper/Metal–Organic Framework Catalysts
0221
Chemoselective Hydrogenation of Nitroarenes on Cobalt/Silicon Carbonitride
0222
Cerum Oxide Catalyzed Oxidative Coupling of Alcohols with Amines to Form Imines
0223
Oxidative Amidation with Heteropolyanion-Based Ionic Liquids
0224
Synthesis of Pyrazolo[3,4-b]pyridines on Cobalt Ferrite/Sulfonated Graphene Oxide