DOI: 10.1055/s-00000131

Synfacts

Issue 08 · Volume 13 · August 2017 DOI: 10.1055/s-007-34437

Synform

A123
Zanda, Matteo: SYNFORM ISSUE 2017/08

Synthesis of Natural Products and Potential Drugs

z0779
All PDFs of this category
0779
Total Synthesis of (–)-Flueggenine C
0780
Synthesis of (+)-Lophirone H
0781
Synthesis of Epacadostat
0782
Synthesis of TEV-37440
0783
Synthesis of (+)-Wortmannin
0784
Regioselective Cyanomethylation of Imidazopyridines
0785
Synthesis of an HIV-1 Protease Inhibitor
0786
Synthesis of Flecainide
0787
Synthesis of 2,4,5-Trisubstituted Imidazoles
0788
Syntheses of Aurachin A and B
0789
Total Syntheses of Lycopodium Alkaloids
0790
Synthesis of (±)-Corymine
0791
Synthesis of (–)-Viridin and (–)-Viridiol

Synthesis of Heterocycles

z0793
All PDFs of this category
0793
Synthesis of C-Aryl Glycosides by Glycosyl C(sp3)–C(sp2) Stille Cross-Coupling
0794
Niobium-Catalyzed Intramolecular Hydrofunctionalization of Alkenes
0795
Lewis Acid Catalyzed Stereoselective Synthesis of Trisubstituted Tetrahydrofurans
0796
Dibenzoxazepinones and -thiazepinones by Dual Copper-Catalyzed Coupling Reactions
0797
Platinum-Catalyzed Synthesis of 2,3-Dihydro-pyrroles and Polyheterocyclic Compounds
0798
Organocatalytic Approach to Functionalized Furans
0799
Stereoselective Synthesis of Pyrrolidine-2,3-diones by a Claisen Rearrangement
0800
Iron-Catalyzed Spirocyclization–Arylation
0801
Synthesis of Pyridoimidazo-β-carbolines
0802
Visible-Light-Induced Iron-Catalyzed Synthesis of 3,3-Disubstituted Oxindoles
0803
Perhydroindolic Acid Catalyzed Synthesis of Chiral Tricyclic γ-Lactams
0804
Radical Cyclization Approach to Borylated Piperidines
0805
Synthesis of Oxazolidinones by a C–H Amination Reaction
0806
Pyrimidines and Pyridines by Ring Expansion of Cyclobutanones
0807
Alkylation of Amines under Mitsunobu Conditions

Synthesis of Materials and Unnatural Products

z0809
All PDFs of this category
0809
The Power of Light in Hexadehydro-Diels–Alder Chemistry
0810
Turning Entangled Molecules Inside Out
0811
Tellurium-Bridged Aromatics
0812
Bridged with Sulfur and Silicon: New Hetero[8]circulenes
0813
There’s More than One Way to Form Corona[5]arenes
0814
Donor–Acceptor Nanohoops
0815
A Radically New Rearrangement
0816
Supramolecularly-Catalyzed Knoevenagel Condensation
0817
Tetracene Dimers Exploring the World of SF (Singlet Fission)
0818
A Pyrene-Capped N-Heteroacene
0819
Direct Allylic/Benzylic C–H Alkylation
0820
Cross-Conjugated [36]Octaphyrins

Metal-Catalyzed Asymmetric Synthesis and Stereoselective Reactions

z0821
All PDFs of this category
0821
Silver-Catalyzed Intermolecular Bromotrifluoromethoxylation of Alkenes
0822
Stereoselective Cyclizations of Allylic Alcohols
0823
Regioselective Palladium-Catalyzed Alkynylation of Enallenes
0824
Palladium-Catalyzed Asymmetric Three-Component Coupling Reaction
0825
Iridium-Catalyzed Diastereoselective Allylation of Glycidols
0826
Ruthenium-Catalyzed Asymmetric Hydro-genation of Nitrogen-Containing Heterocycles
0827
Enantioselective Copper-Catalyzed Aminoarylation of Styrenes
0828
Nickel-Catalyzed Semihydrogenation of Alkynes by Sodium Borohydride
0829
Silver and Amine Co-catalyzed Desymmetrization of Cyclohexanones
0830
Hypervalent Iodine Reagents for the Selective Perfluoroalkyltriflation of Alkynes
0831
Rhodium-Catalyzed Enantioselective Oxidative Cyclization
0832
Iridium-Catalyzed Asymmetric Hydrogenation through Dynamic Kinetic Resolution
0833
Ruthenium-Catalyzed Asymmetric Hydrogenation of β-Acetamidovinyl Sulfides
0834
Copper-Catalyzed Enantioselective [3+1] Cycloaddition Reaction
0835
Rhodium-Catalyzed Enantioselective Synthesis of β′-Aryl Enones
0836
Regioselective Nickel-Catalyzed Hydrocarboxylation of Ynamides
0837
Enantioselective Iridium-Catalyzed Synthesis of Tetrahydroquinolines
0838
One-Pot Cascade Reaction to Form gem-Diarylbenzofuran-3(2H)-ones
0839
Rhodium-Catalyzed Enantioselective Conjugate Addition of Electron-Rich Alkenes
0840
Synthesis and Applications of Chiral Monophosphine Ligands
0841
Iridium-Catalyzed Enantioselective Borylation Reaction
0842
Asymmetric Copper- or Iron-Catalyzed Intramolecular Cyclopropanation
0843
Asymmetric Hydroarylation of Phospholene Oxides through Dynamic Kinetic Resolution
0844
Transition-Metal-Catalyzed Addition of 4-Pyridones to Allenes
0845
Iridium-Catalyzed Enantioselective Hydroarylation
0846
Rhodium-Catalyzed Ring Opening of Stereodefined Vinyl Aziridines
0847
Nickel–Bis(oxazoline)-Catalyzed Enantioselective [3+2] Cycloaddition
0848
Lipase/Iron-Catalyzed Dynamic Kinetic Resolution of Secondary Alcohols
0849
Utilizing Dynamic Kinetic Resolution in Asymmetric Dihydroxylation
0850
Asymmetric Decarboxylative [4+2] Cyclization

Metal-Mediated Synthesis

z0851
All PDFs of this category
0851
Palladium-Catalyzed Decarbonylative Cyanation
0852
Iridium-Catalyzed para-Selective Borylation of Aromatic Esters
0853
Palladium-Catalyzed Chemoselective Alkylation of Aryl Bromides
0854
Copper-Catalyzed Stereoselective Borylation
0855
Sulfone–Metal Exchange
0856
Anionic Fries-Type Rearrangements in Flow
0857
Domino Hydroboration/Trifluoromethylation
0858
Copper-Catalyzed Arylation of Benzylic C–H Bonds
0859
Activation of Earth-Abundant Metal Catalysts Using Sodium tert-Butoxide
0860
Catalytic Enantioselective Preparation of Tertiary Alcohols
0861
Palladium-Catalyzed Cross-Coupling of Silyl Electrophiles with Alkylzinc Halides
0862
Iridium-Catalyzed ortho-Borylation of Phenols
0863
Copper-Mediated 11C-Aromatic Cyanation
0864
Vinyl Azide Enolate [3+2] Cycloaddition

Organo- and Biocatalysis

z0865
All PDFs of this category
0865
NHC-Catalyzed Oxidative [4+2] Annulation of 2-Hydroxybenzaldehydes and Ketones
0866
Chiral Fullerene-Derived Thioureas as Recyclable Asymmetric Organocatalysts
0867
Catalytic Stereoselective Synthesis of Pronucleotides
0868
A Shuttling Strategy for the Enantioselective β-Protonation of Enals
0869
Enantioselective Photoorganocatalytic Formal α-Alkylation of Aldehydes
0870
Total Synthesis of (+)-Rishirilide B through Oxidative Kinetic Resolution
0871
Chemoenzymatic Route to Chiral Gamma Secretase Inhibitor Intermediates
0872
Chiral Phosphoric Acid Catalyzed Kinetic Resolution of 2-Pyridyl Esters
0873
Construction of a Quaternary Carbon by a Mannich Reaction
0874
Direct Hydroxylation of Benzene to Phenol by Cytochrome P450BM3
0875
N-Heterocyclic Carbene Catalyzed Oxidative Spirocyclization of Indoles

Polymer-Supported Synthesis

z0877
All PDFs of this category
0877
Parallel Kinetic Resolution of N-Heterocycles by N-Acylations in Flow
0878
Aerobic Oxidation of Aralkanes on Carbon Nanotube Supported Cobalt
0879
Suzuki Coupling on Eumelanin-Supported Palladium Nanoparticles
0880
Dehydrogenative Aromatization on a Ni–Mg–Al Layered Hydroxide-Supported Pd Catalyst
0881
Controlled Hydrogenation of Alkynes on Polymer-Coated Palladium Nanoparticles
0882
Graphene Oxide/NHC–Supported Pd Catalyst for Cross-Couplings in Water
0883
Silver Nanoparticle Catalyzed Carboxylation of Alkynes with Carbon Dioxide
0884
Friedel–Crafts Alkylation of Indoles with 3-Indolylmethanols
0885
Sonogashira Cross-Coupling on N,N-DMF-Stabilized Copper Nanoparticles
0886
Synthesis of Benzothiazoles by Using a Polythiazolium Catalyst
0887
Tsuji–Trost Allylation with Palladium Nanoparticles in Water
0888
Semihydrogenation of Alkynes on Ti- or Zr-Supported FeOx Nanoparticles
0889
Strecker Reaction with Sulfated Polyborate
0890
Hydrochlorination of Alkynes with Titania-Supported Gold Nanoparticles
0891
Synthesis of Carbonates with Phosphonium-Based Polyionic Liquids
0892
Acidic Zeolite Supported Ruthenium for Selenofunctionalization of Alkenes
0893
Gold-Catalyzed Synthesis of 2,5-Disubstituted Oxazoles