DOI: 10.1055/s-00000131

Synfacts

Issue 06 · Volume 14 · June 2018 DOI: 10.1055/s-008-40151

Synform

A83
Zanda, Matteo: SYNFORM ISSUE 2018/06

Synthesis of Natural Products and Potential Drugs

z0553
All PDFs of this category
0553
Syntheses of Daphniphyllum Alkaloids
0554
Synthesis of Verubecestat
0555
Synthesis of Verubecestat
0556
Total Synthesis of (–)-Lagunamide A
0557
Total Synthesis of (+)-Arenolide
0558
Synthesis of (±)-Sinensilactam A
0559
Synthesis of α-Amanitin
0560
Synthesis of (S)-Omeprazole
0561
Synthesis of GDC-0575
0562
Synthesis of PF-06424439
0563
Synthesis of Entecavir
0564
Synthesis of (+)-Siladenoserinol A
0565
Synthesis of LY426965

Synthesis of Heterocycles

z0567
All PDFs of this category
0567
Heterocycles by NHC-Catalyzed Aerobic Oxidative Annulation
0568
Ligand-Free Catalytic Synthesis of Heterocyclic Sulfones
0569
Vanadium-Promoted Stereoselective Radical Cyclizations to Tetrahydrofurans
0570
Photocatalyzed Synthesis of Sulfonated Isoindolinones
0571
Enantioselective [5+2] Annulations with a Cooperative Catalytic System
0572
Transition-Metal-Free Synthesis of 1,3,5-Triazines
0573
Enantioselective Friedel–Crafts Alkylation of Indoles
0574
Cobalt–Carbene-Catalyzed Synthesis of Indolines
0575
Ruthenium-Catalyzed Remote C–H Activation of Purines
0576
N2-Selective CuO-Catalyzed Coupling of 1H-Indazoles with Diaryliodonium Salts
0577
One-Step Syntheses of 1,4-Diazo Hetero-cycles by Formal [n+2] Cyclizations (n = 4–6)
0578
Dibenzo[f,h]quinolines by Palladium-Catalyzed Decarboxylative Annulation
0579
Michael Addition/[1,2]-Stevens Rearrangement Approach to Piperidines
0580
Synthesis of Oxindolylidene Acetates and Spirooxindolopyrrolidones

Synthesis of Materials and Unnatural Products

z0581
All PDFs of this category
0581
Metal-Free Routes for Biaryls
0582
Aromatic Diels–Alder Annulations Achieved with the Help of the Sun
0583
A Nanographene Propeller with [7]Helicene Blades
0584
Golden Key Unlocks Internal Alkyne Reactivity in Push-Pull Systems
0585
Fluorophore with Two-Photon-Excited and Emissive Behaviors in the NIR Region
0586
Ambiphilicity of Dibromodihydropentacene
0587
Two-Fold Hydroarylation Makes Indolizine
0588
A Super Method to Utilize Ethylene as a C2 Building Block
0589
π-Extended Helicene with Quantum Yield >80%
0590
Controlled Polymerization with the MIDA’s Touch
0591
Red-Emissive Carbon-Bridged Triangulenium Dyes with Long Lifetime
0592
Trichlorosilane Paves the Way from Phosphoric Acid to Phosphorous Molecules

Metal-Catalyzed Asymmetric Synthesis and Stereoselective Reactions

z0593
All PDFs of this category
0593
Iridium-Catalyzed Alkylation of Allenylic Electrophiles
0594
Synthesis of Enantioenriched 2,3-Disubstituted Indolines
0595
Nickel-Catalyzed Asymmetric C–H Functionalization of Pyridones
0596
Rhodium-Catalyzed Enantioselective Alkenylation of Cyclic Ketimines
0597
Rh-Catalyzed Asymmetric Addition of Aryl-boronic Acids to α,β-Unsaturated Ketimines
0598
Palladium-Catalyzed Diastereoselective Synthesis of Imidazolidines
0599
Enantioselective Cyclopropanation of α-Azo Rhodium Carbenoids and Styrenes
0600
Palladium–Catalyzed Unsymmetrical Bis-Silylation of Alkynes
0601
Ru-Catalyzed Dynamic Kinetic Resolution of α-Substituted β-Keto Sulfonamides
0602
Hybrid Phosphorus Ligands for Anti-Markovnikov Hydroformylation
0603
Design of a Bifunctional Chiral Phenanthroline Ligand
0604
Copper-Catalyzed Decarboxylative β-Amino Alcohol Synthesis
0605
Aza-Friedel–Crafts Addition of Phenols to N‑Sulfonyl Aldimines
0606
Rhodium-Catalyzed Desymmetrization of Oxa- and Azabenzonorbornadienes
0607
Copper-Catalyzed Enantioselective Friedel–Crafts Alkylation
0608
Enantio- and Diastereoselective Hydrogenation of α‑Substituted β‑Keto Esters
0609
Enantioselective Allylic Alkylation of 4-Substituted Isoxazolidin-5-ones
0610
Copper-Catalyzed Regio- and Enantio-selective Aminoboration of Alkenes
0611
Iron-Catalyzed Hydrosilylation of Unactivated Terminal Alkenes
0612
Palladium-Catalyzed Synthesis of Chiral-at-Cage Carboranes
0613
Platinum-Catalyzed Asymmetric Hydrosilylation of Alkenylboronates
0614
Asymmetric Catalytic Hydrocarbo-functionalization of Nonactivated Alkenes
0615
Palladium-Catalyzed Trifluoromethyl Indoline Synthesis with Sulfur Ylides
0616
Asymmetric Desymmetrization of Cyclopentenediones
0617
Enantioselective Rhodium–Catalyzed [2+2] Cycloaddition of Allenamides
0618
Rh(II)/Sc(III) Co-catalyzed Multi-component Synthesis of γ-Sulfur-Substituted Ketones
0619
Chiral Pyridoferrocenes by Imidoylative C–H Bond Activation Reaction
0620
Asymmetric Synthesis of Alkyl Aryl(cyano)-[hydroxy(pyridin-2-yl)amino]acetates
0621
Palladium-Catalyzed Asymmetric 1,6-Conjugate Addition of Arylboronic Acids
0622
Stereoselective Friedel–Crafts/Michael Cascade Reaction by Gold Catalysis

Metal-Mediated Synthesis

z0623
All PDFs of this category
0623
Trifluoromethylation of Sulfinamides with Fluoroform
0624
Palladium-Catalyzed Cross-Coupling of Alkylindium Reagents
0625
Synthesis of [11C]Nitriles from Arylboronic Acids and Arylstannanes
0626
Nickel-Catalyzed Cross-Coupling for the Difluoromethylation of Aromatics
0627
Transition-Metal-Free Cross-Coupling of Bis(Sulfones) and Organolithium Reagents
0628
Cyanotrifluoromethylthiolation of Alkynes via Cyano Migration
0629
Synthesis of N-Heterocycles with Continuous Flow Photochemistry
0630
Directed ortho-Metalation and ortho-Fries Rearrangement of Chrysenes
0631
Cyclopropylation of Phenols and Azaheterocycles
0632
Halogen Dance of Bromothiophenes
0633
Nickel-Catalyzed Dearomative Carboamination
0634
Asymmetric Cascade Reaction for the Synthesis of Tetrahydropyrans
0635
Nickel-Catalyzed Cross-Coupling of Enol Ethers
0636
Synthesis of Nitrosobenzene Derivatives from TMS-Substituted Benzenes
0637
Formation of α-Quaternary Aldehydes by Formylation of Allylzinc Reagents

Organo- and Biocatalysis

z0639
All PDFs of this category
0639
Cation Radical Diels–Alder Reactions via Asymmetric Counteranion-Directed Catalysis
0640
Access to Enantioenriched Organosilanes from Enals and β-Silyl Enones
0641
Acridinium-Mediated Photocatalytic Aliphatic C–H Functionalization
0642
Mild Friedel–Crafts Alkylation Inside a Hexameric Resorcinarene Capsule
0643
Hypervalent Iodine Derivatives as Halogen Bonding Based Organocatalysts
0644
Ammonia Lyase Catalyzed Synthesis of Electron-Rich l-Phenylalanines
0645
Chiral Aryl Iodide Catalyzed Fluoroamination of Cinnamyl Derivatives
0646
Selenide-Catalyzed Asymmetric Construction of C–SCF3 Bonds
0647
Superbase-Catalyzed Anti-Markovnikov Addition Reactions

Polymer-Supported Synthesis

z0649
All PDFs of this category
0649
Pt-Catalyzed Chemoselective Hydrogenation of Dienes and Nitroarenes
0650
Photocatalytic C–N Bond Activation and Cross-Coupling of Anilines
0651
Graphitic Carbon Nitride–Magnetite Nanocatalyst for the Synthesis of 4H-Pyrans
0652
Ag–Cu/Metal Oxide Framework for Carboxy-lative Cyclization of Propargylic Compounds
0653
Mukaiyama Aldol Reaction with Iron-Modified Mesoporous Silica
0654
Cobalt-Catalyzed Aerobic Oxidation of Benzylic Alcohols
0655
Dehydrative Cross-Etherification of Alcohols on a Tungsten–Titanium Mixed Oxide
0656
Photocatalytic Aerobic Oxidative Coupling of Amines on a Metal–Organic Framework
0657
Palladium-Catalyzed Formal Cross-Coupling of Diaryl Ethers and Amines
0658
Microwave-Assisted Continuous-Flow Mizoroki–Heck Reaction
0659
Benzylic Homocoupling of Alkylbenzenes on a Pt–Pd Bimetal Catalyst
0660
Synthesis of Benzimidazoles by a Palladium-Catalyzed Hydrogen Transfer
0661
Chemoselective Hydrogenation of Nitroarenes on Cobalt Phosphide/Carbon Nanocubes
0662
Chemoselective Hydrogenation of Nitro-arenes on Supported Nickel Nanoparticles