DOI: 10.1055/s-00000131

Synfacts

Issue 08 · Volume 14 · August 2018 DOI: 10.1055/s-008-40980

Synform

A117
Zanda, Matteo: SYNFORM ISSUE 2018/08

Synthesis of Natural Products and Potential Drugs

z0775
All PDFs of this category
0775
Synthesis of PF-06751979
0776
Synthesis of Shld
0777
Total Synthesis of (+)-Hosieine A
0778
Synthesis of Silanediol FXIa Inhibitors
0779
Synthesis of (+)-Belizentrin Methyl Ester
0780
Synthesis of HIV-1 Protease Inhibitors
0781
Total Synthesis of (–)-Quinine
0782
Synthesis of EPZ015666
0783
Synthesis of Fluorinated BACE Inhibitors
0784
Formal Synthesis of (+)-Kibdelone C
0785
Total Synthesis of (–)-17-nor-Excelsinidine
0786
Synthesis of Pitavastatin
0787
Synthesis of Cyrneine Diterpenoids
0788
Total Syntheses of (–)-Crinipellin A and (–)-Crinipellin B

Synthesis of Heterocycles

z0789
All PDFs of this category
0789
Selective N-Alkylation of 2-Pyridones
0790
A Halocyclization Approach to Enantioenriched Lactones
0791
NHC-Catalyzed Asymmetric Synthesis of Cyclopentene-Fused Tetrahydroquinolines
0792
Ferrocene-Catalyzed Electrosynthesis of Oxindoles and Dihydroquinolin-2-ones
0793
Synthesis of Chromenopyridopyrazines and -diazepines
0794
One-Catalyst, One-Pot, Two C–H Bond Activations
0795
Double C–H Activation Approach to Chromenes
0796
Stereoconserved Synthesis of Triazole-Fused Ketopiperazines
0797
Enantioselective Syntheses of Indolines, Indoles, and Dihydro-2-quinolones
0798
Zinc-Catalyzed Four-Component Synthesis of Highly Substituted Pyridines
0799
Regiocontrolled Synthesis of Pentasubstituted Pyrroles
0800
Rhodium-Catalyzed Indole/Pyrrole Cascade Synthesis
0801
Tetrahydropyrans by an Enantioselective Cross-Dehydrogenative Coupling
0802
Synthesis of Quinoline-4-carboxamides from Ketoxime Acetates and Isatins
0803
Synthesis of Fused Benzothiophenes, Indoles, and Other Heterocycles

Synthesis of Materials and Unnatural Products

z0805
All PDFs of this category
0805
Buckbowls Hold Radical Fare
0806
Hypervalent Iodine Reagents Offer New Choice for Indole–Heteroaryl Coupling
0807
Annulation Expands π−System of Naphthalene Dicarboximide
0808
Arsoles with Strong Solid-State Emission
0809
#Azaacenes #Axialchirality #CPL
0810
Reductive Aromatization of Naphthalene Diimide to 2,7-Diazapyrene
0811
Cooperativity is Always Key: Controlled Copolymerization Achieved with Lewis Pairs
0812
Investigating the Antiaromaticity of Planar 12π and 16π Rings
0813
Fluctuating Macromolecules from Controlled Defects
0814
New Compounds Departing Trifluoromethoxylation Station
0815
Flexible Pillar[6]arene for Enhanced Host–Guest Properties
0816
A New Dimension to Nanographenes

Metal-Catalyzed Asymmetric Synthesis and Stereoselective Reactions

z0817
All PDFs of this category
0817
Enantioselective Decarboxylative Cycloaddition by Palladium Catalysis
0818
Asymmetric 1,3-Dipolar Cycloaddition of Cyclobutenones with Azomethine Ylides
0819
Cobalt-Catalyzed Enantioselective Hydrogenation of Enamides
0820
Intramolecular Enantioselective Palladium-Catalyzed Cycloaddition
0821
Asymmetric Nickel-Catalyzed Intramolecular Hydroalkenylation
0822
Pd/Ti Cooperative Catalysis: Diastereo-selective Synthesis of Spiro-Heterocycles
0823
Rhodium-Catalyzed anti-Hydrosilylation of Internal Ynamides
0824
Enantioselective Synthesis of N-Arylamines via Copper-Catalyzed Hydroamination
0825
Copper-Catalyzed Synthesis of Chiral 1,2-Diamines
0826
Ni-DBFOX Complex as a Bifunctional Photoredox and Lewis Acid Catalyst
0827
Enantioselective Iridium-Catalyzed Allylation Using Enolate Surrogates
0828
Enantioselective N-Allylic Alkylation of Hydrazones with Allylic Acetates
0829
Copper-Catalyzed Asymmetric [3+2] Cycloaddition Reaction
0830
1,4-Protosilylation of α,β-Unsaturated Ketimines
0831
Palladium-Catalyzed Enantioselective Synthesis of α-Quaternary Succinimides
0832
Rhodium-Catalyzed Asymmetric Hydrogenation to Form Chiral γ-Lactams
0833
Enantioselective Alkenylation of Acyclic Enol Ethers
0834
Selective Remote Ring Opening by Palladium Catalysis
0835
Enantioselective Arylative Intramolecular 1,4-Allylations
0836
Silver-Catalyzed Cycloaddition of Glycine Aldimino Esters to Imines
0837
Enantioselective Arylation of γ,δ-Unsaturated β-Ketophosphonates
0838
Biaryl Atropisomers by Pd/Norbornene-Catalyzed Three-Component Reaction
0839
Rhodium-Catalyzed Enantioselective Synthesis of β-Stereogenic Amines
0840
Enantioselective Palladium-Catalyzed Aza-Wacker Cyclization
0841
Cooperative Lewis Base/Palladium-Catalyzed Allylic Alkylation of Esters
0842
Palladium/Brønsted Acid Co-catalyzed Diazo Insertion to C–O or C–N Bonds
0843
Enantioselective Aldol Reaction of an α-Vinylacetamide
0844
Ytterbium-Catalyzed Enantioselective Reduction of Ketones
0845
Palladium-Catalyzed Enantioselective Synthesis of Tetrahydroquinazolines
0846
Copper-Catalyzed Enantioselective Formal [3+3] Annulation

Metal-Mediated Synthesis

z0847
All PDFs of this category
0847
Nickel-Catalyzed 1,2-Dialkylation of Alkenes
0848
Light-Induced 1,2-Carboboration of Unactivated Alkenes
0849
Nickel-Catalyzed Decarbonylative Methylation of Phenyl and Methyl Esters
0850
Iron-Catalyzed Difluoroalkylation of Grignard Reagents
0851
Stereospecific SN2-Type Substitution Using Arylboronic Acids
0852
Electron-Catalyzed C(sp2)–C(sp2) Cross-Coupling
0853
Mild Amination of Organoboronic Acids Using N-Hydroxylamines
0854
Zirconium-Catalyzed Carboalumination–Transmetalation
0855
Synthesis of Trifluoroborate-Iminiums and their Transformation into α-Aminotrifluoroborates
0856
A Novel Palladium(II)-Initiated Borono-Catellani Reaction Under Air
0857
Grignard-Mediated Synthesis of Trisubstituted Triazenes
0858
Nickel-Catalyzed Cross-Couplings of Benzylic Pyridinium Salts
0859
Regioselective Hydrostannation of Alkynes Using a Molybdenum Catalyst
0860
Efficient Hydrotrifluoromethylation of Unactivated Alkenes

Organo- and Biocatalysis

z0861
All PDFs of this category
0861
Hydrogen-Bonding Phase-Transfer Catalyst Enabled Asymmetric Fluorination
0862
9-Fluorenone as Photocatalyst for the Oxidation of Alcohols with Air
0863
Enantioconvergent Allylation of (Arylpropargyl)acetates by an SN1 Reaction
0864
Chiral Amidophosphate-Induced Halooxy- and Haloazacyclizations
0865
Indanol as Scaffold for Chiral Organoiodine Catalysts
0866
α-Oxidation of Cyclic Ketones with 1,4-Benzoquinone through Enol Catalysis
0867
Organocatalytic Synthesis of Axially Chiral Sulfone-Containing Styrenes
0868
Chiral Acid Catalyzed Asymmetric Cloke–Wilson Rearrangement
0869
Whole-Cell Biotransformation of Benzene to Phenol
0870
(–)-Ambrox Production by Biocatalysis Using Squalene Hopene Cyclase

Polymer-Supported Synthesis

z0871
All PDFs of this category
0871
Photodehydrogenation of N-Heterocycles with Hexagonal Boron Carbon Nitride
0872
Epoxidation of Alkenes on an Organosilica-Supported Molybdenum Complex
0873
Controlled Oxidation of Alcohols on a Polymeric Copper Composite
0874
Pyrido[2,3-d]pyrimidines by Domino Cyclization on a Solid Acid Catalyst
0875
Annulation of Ynamides with Nitriles on a Gold(I) Catalyst
0876
Controlled Hydrogenation of Alkynes on Au@N-Doped Carbon/TiO2
0877
[2+2+2] Cycloaddition of Alkynes by Using Pd–Au Alloy Nanoparticles
0878
Cyclization of Alkynoic Acid Derivatitives Catalyzed by Magnetic PdO Nanoparticles
0879
Chemoselective Hydrogenation of α-Keto Amides on Ceria Nanospheres
0880
Decarboxylative A3-Coupling on a Chitosan-Supported Copper Catalyst
0881
Oxidative Esterification of Thiols with Alcohols on a Cobalt Nanocatalyst
0882
The Suzuki–Miyaura Reaction Catalyzed by Supported Pd50Co50 Nanoalloys
0883
Synthesis of Imidazo[1,2-a]pyrimidines by A3-Coupling on CuO Nanoparticles