Synfacts

Issue 04 · April 2020

Recommend Journal

Issue
Synform
A51
Zanda, Matteo: SYNFORM ISSUE 2020/04

Full Text

PDF (1628 kb)
Synthesis of Natural Products and Potential Drugs
z0371
All PDFs of this category

Full Text

PDF (463 kb)
0371
Synthesis of an Indoleamine-2,3-dioxygenase-1 (IDO1) Inhibitor FREE ACCESS

Full Text

HTML

PDF (130 kb)
0372
Total Synthesis of (–)-Cymoside

Full Text

HTML

PDF (89 kb)
0373
Total Synthesis of (+)-Corymine and (–)-Deformylcorymine FREE ACCESS

Full Text

HTML

PDF (130 kb)
0374
Synthesis of (–)-FD-594

Full Text

HTML

PDF (91 kb)
0375
Total Syntheses of ent-Kaurane Diterpenoids

Full Text

HTML

PDF (98 kb)
0376
Synthesis of Aztreonam

Full Text

HTML

PDF (89 kb)
0377
Total Synthesis of Tetrodotoxin

Full Text

HTML

PDF (80 kb)
0378
Synthesis of Simurosertib (TAK-931)

Full Text

HTML

PDF (82 kb)
0379
Synthesis of (–)-Pepluanol B

Full Text

HTML

PDF (104 kb)
0380
Synthesis of BMS-986260

Full Text

HTML

PDF (104 kb)
0381
Synthesis of (±)-Saudin FREE ACCESS

Full Text

HTML

PDF (135 kb)
Synthesis of Heterocycles
z0383
All PDFs of this category

Full Text

PDF (365 kb)
0383
2-Arylpiperidines by Palladium-Catalyzed Addition of Arylboronic Acids to Acylated 2-Hydroxypiperidines FREE ACCESS

Full Text

HTML

PDF (117 kb)
0384
Synthesis of Phosphorylpyrroloindoles by Photocatalytic Phosphinoylation/Cyclization Reactions

Full Text

HTML

PDF (87 kb)
0385
Synthesis of Thiochromenes by Palladium-Catalyzed Ring Opening of Cyclopropyl Thioethers

Full Text

HTML

PDF (80 kb)
0386
Regioselective Synthesis of Polyfluorinated o-Hydroxyacetophenones

Full Text

HTML

PDF (91 kb)
0387
Chemodivergent and Enantiospecific Synthesis of Benzazepines and Allyl Fluorides

Full Text

HTML

PDF (77 kb)
0388
Organocatalyzed Synthesis of Fully Substituted Furans from Ynamides and Quinoxaline N-Oxides

Full Text

HTML

PDF (99 kb)
0389
Diastereoselective De Novo Synthesis of Functionalized Piperidines

Full Text

HTML

PDF (80 kb)
0390
Construction of Highly Substituted Furans and Thiophenes with Sulfur Ylides

Full Text

HTML

PDF (82 kb)
0391
C(sp³)–H Functionalization of Aliphatic Acids through β-Lactonization

Full Text

HTML

PDF (100 kb)
0392
Asymmetric Copper-Catalyzed Synthesis of Dihydrobenzofuran-3-ols

Full Text

HTML

PDF (89 kb)
0393
Palladium(II)-Catalyzed Synthesis of Tribenzo[b,d,f]azepines

Full Text

HTML

PDF (95 kb)
0394
Three-Component Synthesis of 3-(Trifluoromethyl)pyrazoles

Full Text

HTML

PDF (72 kb)
0395
Base-Promoted Annulations in the Synthesis of Ring-Fused N-Substituted-4-Quinolinones

Full Text

HTML

PDF (88 kb)
Synthesis of Materials and Unnatural Products
z0397
All PDFs of this category

Full Text

PDF (408 kb)
0397
Approaching a Pyridine by Aza-APEX

Full Text

HTML

PDF (92 kb)
0398
All Aboard the EBXpress to Dithioalkenes

Full Text

HTML

PDF (81 kb)
0399
Put Phosphorus in Your Rhodamine

Full Text

HTML

PDF (74 kb)
0400
From Simple to Complex: One-Pot Synthesis of Dimeric Pyrrolo-Fused Isoquinolines

Full Text

HTML

PDF (76 kb)
0401
Spin Me Right Round: Spirocyclic Organic Electronic Materials

Full Text

HTML

PDF (84 kb)
0402
Fountain of Pyrenes

Full Text

HTML

PDF (82 kb)
0403
Lighting Up Helicenes

Full Text

HTML

PDF (90 kb)
0404
Small Helicenes, Big Deal

Full Text

HTML

PDF (74 kb)
0405
Party of Rotaxanes

Full Text

HTML

PDF (75 kb)
0406
Ion Pair Receptors: Bambusuril–Crown Ether Conjugates

Full Text

HTML

PDF (75 kb)
0407
‘A One and A Two’: Orchestrating Polymer Backbone Breakdown

Full Text

HTML

PDF (159 kb)
0408
Expansion of Coumarins by One-Pot Synthesis

Full Text

HTML

PDF (92 kb)
Metals in Synthesis
z0409
All PDFs of this category

Full Text

PDF (761 kb)
0409
Bismuth Redox-Catalyzed Fluorination of Arylboron Reagents FREE ACCESS

Full Text

HTML

PDF (127 kb)
0410
A Diastereo- and Enantioselective Copper-Catalyzed Allylation of Imines Using Allylic gem-Diboron Reagents

Full Text

HTML

PDF (77 kb)
0411
Palladium-Catalyzed γ-C(sp³)–H Bond Activation of Tertiary Alkyl Amines FREE ACCESS

Full Text

HTML

PDF (135 kb)
0412
Coupling Reactions of Aldehydes and Hydrocarbons

Full Text

HTML

PDF (73 kb)
0413
Synthesis of Conjugated 1,3-Diynes

Full Text

HTML

PDF (73 kb)
0414
Aryl Thioether Metathesis under Nickel Catalysis

Full Text

HTML

PDF (73 kb)
0415
Enantioselective Preparation of Propargyl Amides

Full Text

HTML

PDF (71 kb)
0416
Axially Chiral 2,3-Disubstituted Indoles via Palladium-Catalyzed Enantioselective Cacchi Reaction

Full Text

HTML

PDF (93 kb)
0417
Copper-Catalyzed Coupling of Remote C(sp³)–H Bonds with Terminal Alkynes

Full Text

HTML

PDF (91 kb)
0418
meta-Selective Inverse Sonogashira Coupling

Full Text

HTML

PDF (91 kb)
0419
Nickel-Catalyzed Carboxylation of Arylsulfonium Salts Using CO₂

Full Text

HTML

PDF (73 kb)
0420
Palladium-Catalyzed Asymmetric Cycloadditions

Full Text

HTML

PDF (88 kb)
0421
C–H Functionalization of Alkenes

Full Text

HTML

PDF (84 kb)
0422
Enantioselective Rhodium-Catalyzed Hydroformylation of α-Substituted Acryl Acid Derivatives

Full Text

HTML

PDF (89 kb)
0423
Photocatalytic Umpolung Strain-Release Amino-Functionalization of [1.1.1]-Propellanes

Full Text

HTML

PDF (76 kb)
0424
Transthioetherification of Aryl Halides with Thioethers or Thioesters under Palladium Catalysis

Full Text

HTML

PDF (78 kb)
0425
Stereodivergent Allylic Alkylation/Fluorination of Acyclic Ketones

Full Text

HTML

PDF (82 kb)
0426
Dual Catalysis: Photoredox/Chromium-Catalyzed Dialkylation of 1,3-Dienes

Full Text

HTML

PDF (80 kb)
0427
Chromium/Iridium-Photoredox Dual-Catalyzed Formal Addition of α-Amino Carbanions to Carbonyls

Full Text

HTML

PDF (112 kb)
0428
Hydroamination of Alkenes

Full Text

HTML

PDF (72 kb)
0429
Radical Cascade Synthesis of Azoles

Full Text

HTML

PDF (79 kb)
0430
Nickel-Catalyzed Reductive Acylation of Aliphatic Amines

Full Text

HTML

PDF (78 kb)
0431
Intermolecular Palladium-Catalyzed Atropo-Enantioselective C–H Arylation of Heteroarenes

Full Text

HTML

PDF (73 kb)
0432
Synthesis of 1,3-Dienes by a Photoinduced C(sp²)−H/C(sp²)−H Cross-Coupling of Alkenes

Full Text

HTML

PDF (89 kb)
0433
Fused Tricyclic Hydronaphthofurans through Rhodium-Catalyzed Desymmetrization

Full Text

HTML

PDF (81 kb)
0434
Scandium-Catalyzed Enantioselective C–H Transfer Across an Alkene

Full Text

HTML

PDF (77 kb)
0435
Low Catalyst Loading: Rhodium(II)-Catalyzed Asymmetric Cyclopropanation

Full Text

HTML

PDF (71 kb)
0436
Photoredox-Catalyzed Benzylic C–H Activation and Coupling with Aldehydes

Full Text

HTML

PDF (86 kb)
0437
The Corey–House Reaction: An Early Transition-Metal-Mediated Cross-Coupling FREE ACCESS

Full Text

HTML

PDF (125 kb)
Polymer-Supported Synthesis
z0439
All PDFs of this category

Full Text

PDF (342 kb)
0439
Photocatalytic C–H Alkylation of Quinoxalin-2-ones on a Covalent Organic Framework FREE ACCESS

Full Text

HTML

PDF (137 kb)
0440
Palladium/Alumina-Catalyzed Decarbonylative Aldol Condensation of Aldehydes

Full Text

HTML

PDF (75 kb)
0441
Photocatalytic Oxidative Coupling of Benzylamines on a Hydrazone-Based Covalent Organic Framework

Full Text

HTML

PDF (80 kb)
0442
A Zirconium–Tannin Hybrid Catalyst for Meerwein–Ponndorf–Verley Reduction

Full Text

HTML

PDF (75 kb)
0443
Reductive Amination of 5-(Hydroxymethyl)furfural on Immobilized Palladium Nanoparticles

Full Text

HTML

PDF (85 kb)
0444
C–C, C–O, C–S, and C–N Bond Formation from Diazo Compounds on Mesoporous Silica-Supported Triflic Acid

Full Text

HTML

PDF (79 kb)
0445
Silver Nanoparticle Catalyzed Selective Reduction of Nitro Compounds and Nitriles

Full Text

HTML

PDF (81 kb)
0446
Aza-Semipinacol Rearrangement Catalyzed by Graphene Oxide

Full Text

HTML

PDF (80 kb)
0447
Flow Esterification on a Second-Generation m-Phenolsulfonic Acid–Formaldehyde Resin Catalyst

Full Text

HTML

PDF (92 kb)
0448
Reduction of Aryl Ketones and Aldehydes to Hydrocarbons Catalyzed by Palladium/Carbon

Full Text

HTML

PDF (91 kb)
0449
CuMoO₄ Nanoparticles-Catalyzed Cross-Coupling of Aryl Halides with Thiols

Full Text

HTML

PDF (72 kb)
0450
One-Pot Sequential Cross-Aldol Condensation/Aza-Michael Addition on Graphene Oxide

Full Text

HTML

PDF (75 kb)
0451
Dehydrogenation of NH–NH Bonds Catalyzed by Ni–Fe Supported on N-Doped Carbon from Chitosan

Full Text

HTML

PDF (69 kb)
Organo- and Biocatalysis
z0453
All PDFs of this category

Full Text

PDF (314 kb)
0453
Pot-Economic Organocatalytic Asymmetric Synthesis of the Corey Lactone FREE ACCESS

Full Text

HTML

PDF (136 kb)
0454
Superbase-Catalyzed Enantioselective Aldol Addition of Aryl Ketones to α-Fluorinated Ketones

Full Text

HTML

PDF (98 kb)
0455
A Modified Tripeptide Catalyst Changes Conventional Diastereoselectivity in Michael Additions

Full Text

HTML

PDF (87 kb)
0456
Organic Single-Electron Reductants Permit Photocatalytic Borylation of C–O, C–N, and C–X Bonds

Full Text

HTML

PDF (84 kb)
0457
N-Functionalized Azaheterocycles through P^III/P^V=O-Catalyzed Cascade Synthesis

Full Text

HTML

PDF (85 kb)
0458
NHC-Catalyzed Generation of p-Quinodimethanes through ε-Umpolung: Nucleophilic Addition to Ketones

Full Text

HTML

PDF (98 kb)
0459
Two Distinct Hydrogen Atom Transfer Steps Permit Selective Epimerization of Pyranose Frameworks

Full Text

HTML

PDF (78 kb)
0460
NHC-Catalyzed Umpolung Approach Toward Heteroaryl Ynones

Full Text

HTML

PDF (84 kb)
0461
Reductive Electrophotocatalysis

Full Text

HTML

PDF (86 kb)
Chemistry in Medicine and Biology
z0463
All PDFs of this category

Full Text

PDF (539 kb)
0463
RIBOTACs – Targeted Degradation of RNA FREE ACCESS

Full Text

HTML

PDF (227 kb)
0464
Stronger Together!

Full Text

HTML

PDF (84 kb)
0465
Protein Modification by Cope Rearrangement

Full Text

HTML

PDF (84 kb)
0466
Potent and Selective Acid Sphingomyelinase Inhibitors with Antidepressant Activity

Full Text

HTML

PDF (70 kb)
0467
Replacing HN₃ with Nitromethane for Schmidt-Type Formation of Amides and Nitriles

Full Text

HTML

PDF (83 kb)
0468
Lasonolide A is a Prodrug Activated by LDAH, a Serine Hydrolase

Full Text

HTML

PDF (79 kb)
0469
PEP-K: A New Reagent for the O-Phosphorylation of Alcohols

Full Text

HTML

PDF (78 kb)
0470
Modular, Targeted IDO Inhibitor for Cancer Immunotherapy

Full Text

HTML

PDF (83 kb)
0471
A Potential anti-Pertussis Vaccine Based on Lipopolysaccharide Endotoxins of B. pertussis

Full Text

HTML

PDF (101 kb)
0472
A Carbapenemase Probe that Switches on the Light

Full Text

HTML

PDF (82 kb)
0473
Cyclic Naphthoquinone Imine Based Antagonists of the RIG-I Innate Immune Receptor

Full Text

HTML

PDF (77 kb)
0474
Optical Control of CENP-E Function

Full Text

HTML

PDF (81 kb)
0475
A Classic Way of Forming Amide Bonds FREE ACCESS

Full Text

HTML

PDF (132 kb)
Peptide Chemistry
z0477
All PDFs of this category

Full Text

PDF (376 kb)
0477
Boronic Acid Catalyzed Dehydrative Peptide Synthesis FREE ACCESS

Full Text

HTML

PDF (122 kb)
0478
Phase-Transfer-Catalyzed Enantioselective α-Trifluoromethylthiolation

Full Text

HTML

PDF (97 kb)
0479
Stereoselective Synthesis of β-Amino Acid Precursors by Organocatalysis

Full Text

HTML

PDF (88 kb)
0480
Copper-Catalyzed [3+1] Cycloaddition to Form Substrates for α-Amino Acid Synthesis

Full Text

HTML

PDF (87 kb)
0481
Synthesis of Selenocystine-based Peptides through Cyclization Reactions

Full Text

HTML

PDF (74 kb)
0482
Copper-Catalyzed Synthesis of Cyanated Peptides

Full Text

HTML

PDF (73 kb)
0483
Stereoselective Synthesis of Unnatural α-Amino Acids

Full Text

HTML

PDF (121 kb)
0484
Palladium-Catalyzed N-Arylation of Amino Acids and Ketoxime Peptide Ligation

Full Text

HTML

PDF (79 kb)
0485
Synthesis of α-Quaternary Chiral Amino Acids by Palladium-Catalyzed Arylation

Full Text

HTML

PDF (97 kb)
0486
Synthesis of Fmoc-Aminoacyl‑N‑alkylcysteine Dipeptides by Using the Ugi Reaction

Full Text

HTML

PDF (74 kb)
0487
Solid-State Synthesis of a β-Turn Mimetic FREE ACCESS

Full Text

HTML

PDF (141 kb)
Flow Chemistry
z0489
All PDFs of this category

Full Text

PDF (130 kb)
0489
Synthesis of Biaryl Compounds in Flow via a Lithiation, Borylation, Suzuki–Miyaura Cross-Coupling Pathway

Full Text

HTML

PDF (88 kb)
0490
Ferrocenyl Azide Synthesis via Halogen–Lithium Exchange in Continuous Flow

Full Text

HTML

PDF (85 kb)
0491
Acylation with Grignard Reagents in Continuous Flow

Full Text

HTML

PDF (66 kb)
Most Read
Archive
Articles by Category
Free Sample Issue

Journal

More About This Journal
Synfacts Videos
Editorial Board
Editorial Office
Brochure

Authors

Instructions for Authors

Subscription

Subscription Information & Contacts
Institutional Licensing

Nobel Prize 2016

Instructions for Authors

Journals
Book Series
Login
Help
Portal
Return to Classic Website

German English

Thieme E-Books & E-Journals is a service of Georg Thieme Verlag and Thieme Medical Publishers, Inc.
© Georg Thieme Verlag KG

Imprint | Privacy policy statement

Your Current IP Address: 3.147.73.41