Synfacts

Issue 07 · July 2021

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A105
SYNFORM ISSUE 2021/07 FREE ACCESS

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Synthesis of Natural Products and Potential Drugs
z0721
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0721
Synthesis of (+)-Manginoid A and (–)-Manginoid C FREE ACCESS

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0722
Synthesis of Sisunatovir

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0723
Synthesis of β-Secretase Inhibitor NB-360 FREE ACCESS

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0724
Synthesis of 9,11-Secosteroids (+)-Pinnigorgiol B and (–)-Pinnigorgiol E

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0725
Total Synthesis of (+)-Alstilobanine C, (+)-Undulifoline, and (−)-Alpneumine H

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0726
Formal Synthesis of BMT-362265

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0727
Synthesis of Tacalcitol

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0728
Synthesis of (–)-Koumimine

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0729
Total Synthesis of Perovskones and Hydrangenone

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0730
Synthesis of AG-270

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0731
Synthesis of P2X7 Receptor Antagonist Lu AF27139

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0732
Synthesis of Emitasvir

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0733
Synthesis of BPR1K871

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0734
Formal Synthesis of Telmisartan

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0735
Synthesis of Encequidar

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0736
Total Synthesis of (±)-Dehydroxypycnidione

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0737
Total Synthesis of (±)-Desacetylcolchicine and Formal Synthesis of (±)-Colchicine FREE ACCESS

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Synthesis of Heterocycles
z0739
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0739
One-Pot Stepwise Synthesis of γ-Lactams through Cycloadditions with Ketenes FREE ACCESS

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0740
Palladium-Catalyzed Synthesis of Benzoxepines from Vinyl-Substituted Cyclopropanes and Salicylaldehydes

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0741
Mild Regioselective Reduction of Pyridines to Dihydropyridines

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0742
Rhenium-Mediated Synthesis of Five- and Six-Membered Nitrogen-Containing Heterocycles

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0743
Sequential Palladium-Catalyzed Synthesis of Benzosultams

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0744
Regioselective Synthesis of Indoles form Azoarenes or Azoxyarenes with Ketones

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0745
Copper-Catalyzed Synthesis of Quinazolines and 1,2,4-Oxadiazoles

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0746
Iridium-Photocatalyzed Synthesis of Bioactive Tetracyclic Nitrogen-Containing Products

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0747
2-Pyridones from Enamides through Ni–Al Bimetallic Catalysis

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0748
Synthesis of Functionalized Benzimidazoles through C(sp³)–H Amination/C–N Bond Cleavage

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0749
Palladium-Catalyzed Synthesis of Enantiopure Eight-Membered Nitrogen Heterocycles

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0750
One-Pot Construction of 2,3-Dialkyl-Substituted Quinazolinones from Secondary Amides and Isocyanate

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0751
Iridium-Catalyzed Approach to Polycyclic Nitrogen-Containing Systems

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0752
Selectfluor-Promoted Synthesis of Functionalized Isothiazolones

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Synthesis of Materials and Unnatural Products
z0753
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0753
Powerful Rotamers for Asymmetric Synthesis

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0754
Inserting a Seventh Carbon into Perylene Bisimide

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0755
Site-Selective Electrophilic Substitution of 9-Substituted Triptycenes

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0756
Accessing Useful Quantities of CPP

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0757
Carbons by the Barrel

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0758
Efficient Six-Step Synthesis of peri-Heptacene

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0759
Synthesis of β-Isoindigo Derivatives

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0760
Elegant Ring Formation Aided by Iron

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0761
One Step to Spiro Nation

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0762
Selective Synthesis of Cyclo[9]pyrroles FREE ACCESS

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0763
Falling into Place: Facile Access to Modular 2,6-Dicyanoanilines

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0764
Silicon on the Run in a Gold-Catalyzed Cycloisomerization

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Metals in Synthesis
z0765
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0765
Nickel-Mediated C(sp³)–H Methylation via Photochemical Activation of Peroxides FREE ACCESS

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0766
Switchable Selectivity in the Asymmetric Rhodium-Catalyzed Hydrothiolation of Cyclopropenes

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0767
Ruthenium-Catalyzed Enantioselective Reductive Amination FREE ACCESS

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0768
NiH-Catalyzed Hydroamidation of Alkynes with Dioxazolones

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0769
Nickel-Catalyzed Site-Selective Heteroarylation of Cyclobutanols

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0770
Synthesis of Indoles from N-Benzoyloxyallylamines and Iodoarenes by Palladium/Norbornene Catalysis

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0771
Synthesis of Chiral Sulfones by Three-Component Radical Reaction

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0772
Photocatalyzed Decarboxylation of Carboxylic Acids

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0773
Iron-Catalyzed Oxidation of Olefins

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0774
Alkylation and Alkenylation of Neopentylamine

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0775
δ-Fluorination of N-Alkyl Sulfonamides

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0776
Fluoroalkylative Reductive Coupling of Alkyl Bromides

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0777
Dioxazolones as Nitrene Precursors under Iron Catalysis

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0778
Photoredox and Nickel-Catalyzed Aminoarylation

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0779
Preparation of Functionalized 1,3-Disbustituted BCBs

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0780
Visible-Light Assisted Sulfonylation of (Hetero)Aryl Halides

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0781
Dual-Ligand-Enabled Ruthenium-Catalyzed C–H Arylation of Buchwald Phosphine Ligands

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0782
Manganese-Catalyzed Hydroboration of Unsaturated C=X Bonds

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0783
Asymmetric, Light-Mediated Radical Sulfinyl-Smiles Rearrangement

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0784
ortho-C–H Imidation of Benzaldehydes using a Transient Directing Group

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0785
Nickel-Catalyzed Aldol Reactions

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0786
Preparation of Polycyclic Lactams

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0787
Asymmetric Synthesis of γ-Lactams by Palladium-Catalyzed Hydroesterificative Cyclization

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0788
Synthesis of Nitrogen-Containing Terminal Alkyl Chlorides via Copper-Catalyzed Chloromethylazidation

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0789
Synthesis of Fully Substituted Pyrroles from Imino Ethers and Enol Diazoacetates using Silver Catalysis

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0790
1,4-Acetoxychlorination of Dienes: The Bäckvall Reaction FREE ACCESS

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0791
Enantioselective Preparation of Propargylsilanes

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0792
Incorporation of gem-Difluoroalkene Motifs via Regioselective C(sp³)–H Functionalization

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Polymer-Supported Synthesis
z0793
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0793
A Polymeric Bipyridyl Nickel Composite for C–H Arylation of Heteroarenes

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0794
Suzuki–Miyaura Coupling with a Palladium-Complexed Azo Porous Organic Polymer

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0795
Hydroaminomethylation of Alkenes Promoted by Ruthenium on TiO₂

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0796
Sulfonation of Enamides, Acrylamides, and Enones Photocatalyzed by Single-Atom Nickel on TiO₂

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0797
C–C Coupling of Nitriles with Arylboronic Acids Catalyzed by Mesoporous Silica-Tethered Platinum

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0798
Photocatalytic Oxidative Amidation of Aldehydes with Magnetic Cadmium Sulfide Quantum Dots

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0799
Catalytic Esterification of Amides by Using a Zirconium-Based Metal–Organic Framework

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0800
Hydrogenation of Carbonyls, Nitriles, and Nitroarenes by Using Ni₂P Nanoalloy Catalyst in Water

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0801
Protection and Deprotection of Alcohols by Using a Zn Complex Supported on Magnetic Nanoparticles

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0802
Tandem Asymmetric Michael/Transfer Hydrogenation by Using a Dual Rh-Incorporated Micelle Reactor FREE ACCESS

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Organo- and Biocatalysis
z0803
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0803
Heterofunctionalization of Arenes by Electrophotocatalysis FREE ACCESS

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0804
Biosynthesis of Hirsutellones and Pyrrocidines through an exo-Selective Diels–Alder Cycloaddition

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0805
Pyrrolidine Aminocatalytic Asymmetric [12+2] Cycloaddition toward Cycl[3.2.2]azines

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0806
Activation of N-Heterocycles by Silylium Catalysis for C–C Bond Formation FREE ACCESS

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0807
Catalytic (3+2) Annulation of Aminocyclopropane Monoesters and Indoles

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0808
Organocatalytic, Visible-Light-Mediated Dicarboxylation with Carbon Dioxide via Anion Radicals

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0809
Catalytic Asymmetric Stereospecific Substitutions of Racemic α-Aryl Aldehydes

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0810
Catalytic Asymmetric α-Chlorination of Aldehydes

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0811
Two Work Better Than One: Cooperative NHC and Photoredox Catalysis for Benzylic C–H Bond Acylation

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Chemistry in Medicine and Biology
z0813
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0813
Spirocyclic Ketone Construction via Semipinacol-Type Rearrangement FREE ACCESS

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0814
Biphenyl Imidazopyridines as a New Scaffold for PD-L1 Inhibitors

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0815
Synthesis and Application of the 3-Phosphonofluoresceins

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0816
Selective Cannabinoid Type 2 Receptor Antagonists

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0817
Watching RNA Do Its Job

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0818
Site-Selective LYTACs for Targeted Protein Degradation

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0819
Scalable Synthesis of Opioids Enabled by a Palladium-Catalyzed Dearomative Arylation

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0820
Small-Molecule Inhibitor of an RNA-Modifying Enzyme for Acute Myeloid Leukemia Treatment

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0821
Late-Stage Alkylation of Purine Nucleoside at the C6 Position

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0822
Utorubicin: A Novel Anthracycline Cancer Prodrug

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0823
Next-Generation Macrolide Antibiotics FREE ACCESS

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0824
Stereostructure–Activity Studies of Spirooliganin

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Peptide Chemistry
z0825
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0825
Palladium-Catalyzed Olefination of Oxazole-Containing Peptides FREE ACCESS

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0826
Oxidative Peptide Bond Formation of 2-(Aminomethyl)malononitriles

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0827
Copper-Catalyzed Synthesis of Bulky Amides and Peptides

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0828
Hypervalent-Iodine-Mediated Peptide-Bond Formation to Synthesize Hindered Peptides

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0829
Nickel-Catalyzed Synthesis of β-Amino Acid Derivatives

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0830
Synthesis of Isoquinolone-Containing Amino Acids by Rhodium-Catalyzed C–H Annulation

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0831
Palladium-Catalyzed δ-C(sp³)–H Arylation of Amino Acids

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0832
Petasis Reaction for the Synthesis of Unnatural Amino Acids

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0833
Synthesis of N-Unprotected α-Amino Acid Methyl Esters FREE ACCESS

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0834
Photoredox-Catalyzed Synthesis of γ-Amino Acid Derivatives

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Flow Chemistry
z0835
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0835
N-Arylation of Amino Acid Esters using a Pd(OH)₂ Packed-Bed Reactor

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0836
Bromine–Sodium Exchange and Directed Metalations in Continuous Flow

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0837
Synthesis of Fluorinated Tertiary Alcohol Derivatives under Visible-Light Irradiation

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0838
Ru-promoted Photooxidative C–H Functionalization of Isoquinolines in a Microflow Reactor

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0839
Precise Control of cis−trans Isomerization of α-Anionic Stilbenes under Flow Conditions

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