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Synfacts 2022; 18(05): 0484
DOI: 10.1055/s-0041-1738013
Synthesis of Heterocycles

Enhanced Potency and Properties by Exploiting Substituted Oxetane as a Cyclobutane Bioisostere

(Pfizer) Contributor(s):
Paul Richardson
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Key words

IDO1 inhibitors - oxetane - Mitsunobu reaction - bioisosteres - oncology


Publication History

Article published online:
20 April 2022

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