Synfacts, Table of Contents Synfacts 2023; 19(04): 0415DOI: 10.1055/s-0042-1752649 Innovative Drug Discovery and Development Macrocyclization and Scaffold Hopping Improves Selectivity and ADME Properties of HPK1 Inhibitors Authors Contributor(s): Antonia F. Stepan (Roche) Ferdinand H. Lutter (Janssen Pharmaceutica) Ulrich Lücking (FoRx Therapeutics) Recommend Article Abstract Buy Article(opens in new window)Key words Key wordsmacrocycles - kinase inhibition - selectivity - ADME - scaffold hopping Full Text