DOI: 10.1055/s-00000131

Synfacts

Issue 06 · Volume 11 · June 2015 DOI: 10.1055/s-005-29148

Synform

A76
Zanda, Matteo: SYNFORM ISSUE 2015/06

Synthesis of Natural Products and Potential Drugs

z569
All PDFs of this category
0569
Synthesis of Schilancitrilactones B and C
0570
Synthesis of Solabegron
0571
Synthesis of HCV Protease Inhibitor MK-6325
0572
Syntheses of Rubialatin A, Rubialatin B, and Related Congeners
0573
Synthesis of Reverse Transcriptase Inhibitor Tenofovir
0574
Total Synthesis of (+)- and (–)-Rocaglamide
0575
Synthesis of Doravirine
0576
Synthesis of (+)-Isatisine A
0577
Total Syntheses of Arnottin I and Arnottin II
0578
Total Synthesis of Leupyrrin A1
0579
Synthesis of SGLT2 Inhibitor Canagliflozin
0580
Synthesis of AMG 925
0581
Biomimetic Synthesis of (±)-Pallidol and (±)-Quadrangularin A

Synthesis of Heterocycles

z583
All PDFs of this category
0583
Pd-Catalyzed Ortho-Amination/ipso-Functionalization of Aryl Iodides
0584
Catalytic Enantioselective Piperidine Synthesis by [4+2] Cyclization
0585
Stereoselective Intramolecular [3+2] Annulations to Fused Heterocycles
0586
Synthesis of Fluorine-Containing 3-Hydroxypyridin-4-ones
0587
Quinoxalines from Pyrroloarylisocyanide by Photoredox Catalysis
0588
Synthesis of Heteroring-Annulated 1,4-Oxazepines
0589
Chirality Transfer in the Synthesis of Pyrrolidines
0590
Thia-Prins Cyclization Approach to Tetrahydrothiophenes and -furans
0591
Three-Component Synthesis of Fluorinated Pyrazoles
0592
2-Picolylamines and Imidazopyridines from Pyridotriazoles by Rh(II) Catalysis
0593
Palladium-Catalyzed Route to Ortholactones from Cyclic Enol Ethers
0594
Synthesis of Benzo[b]thiophenes by Sequential Cyclization Reactions
0595
Multicomponent Synthesis of Benzopyrans
0596
In Situ Generation of Difluoromethyl Diazomethane. Synthesis of Pyrazoles
0597
Iron-Catalyzed Synthesis of Isoxazoles from Homopropargylic Alcohols

Synthesis of Materials and Unnatural Products

z599
All PDFs of this category
0599
Sweet Fullerenes
0600
Just Add Water: Methanofullerene Synthesis in an Aqueous Two-Phase System
0601
Aryne’t You Doubly Impressed with this Cyclopropenone Insertion?
0602
Choose Your Own Silver Salt Adventure: The Heterocyclic Series
0603
One-Pot Prep: From Quinones to Dicyanoarenes in Two Easy Steps
0604
Polybenzoquinolines
0605
Chopping Cavitands
0606
Rigidifying Dyes for High Efficiency DSCs
0607
Loosening the Belt
0608
Dimethyl Sulfate Promoted Pd/Cu-Catalyzed Arylation
0609
Colorful on the Inside and Out
0610
One Shot to Nanographene Structures

Metal-Catalyzed Asymmetric Synthesis and Stereoselective Reactions

z611
All PDFs of this category
0611
Copper-Catalyzed Stereoselective 1,3-Dipolar [3+6] Cycloaddition
0612
Enantioseletive Rhodium-Catalyzed Hydrogenation of Enamides
0613
Asymmetric Cyclization of Ene-Allenes by Nickel Catalysis
0614
Dynamic Kinetic Allylic Alkylation with Zirconium Nucleophiles
0615
Enantioselective Remote Functionalization of Carbonyl Compounds
0616
Asymmetric Oxidative Carbocyclization-Borylation of Enallenes
0617
Enantioselective 1,4-Addition of Amides with α,β-Unsaturated Carbonyls
0618
Asymmetric Copper-Catalyzed Detrifluoroacetylative Aldol Reactions
0619
Silver-Catalyzed Asymmetric Cycloaddition Using Non-Biaryl Atropisomers
0620
Asymmetric Conjugate Addition of Grignard Reagents to Lactones
0621
Asymmetric Hydroalkoxylation of Non-Activated Alkenes at High Temperature
0622
Stereoselective Ruthenium/Copper-Catalyzed Synthesis of 2-Alkenyl Indoles
0623
Asymmetric Synthesis of α,α-Diaryl α-Amino Acid Derivatives
0624
Asymmetric Pd-Catalyzed C–H Arylation to Access P-Stereogenic Compounds
0625
Asymmetric [3+2] Cycloaddition of Azomethine Ylides with Acyclic 1,3-Dienes
0626
Iron-Catalyzed Asymmetric Hydrogenation of Ketones
0627
NHC–Rh Catalyzed Asymmetric 1,2-Addition of Boronic Acids to Aromatic Aldehydes
0628
Enantioselective Copper-Catalyzed Aldol Reaction Using α-Azido Amide
0629
Asymmetric Desymmetrization via Oxidative Heck Reaction
0630
Palladium-Catalyzed Synthesis of Branched Allylic Fluorides
0631
Palladium-Catalyzed Synthesis of P-Chiral Phosphinic Amides via C–H Activation
0632
Nickel–NHC Complex Catalyzed Asymmetric Cross-Hydroalkenylation
0633
Synthesis of Tetrahydroisoquinolines Catalyzed by Copper
0634
Asymmetric Hydroformylation of Vinylarenes Using Formaldehyde
0635
Isomerization–Asymmetric Tansfer Hydrogenation of Allylic Alcohols
0636
Palladium-Catalyzed C–H Activation for the Synthesis of Chiral Biaryl Phosphates
0637
Enantioselective 1,2-Perfluoroalkyl Migration Catalyzed by Zinc
0638
Asymmetric Nozaki–Hiyama–Kishi Allylation

Metal-Mediated Synthesis

z639
All PDFs of this category
0639
Hydrogermylations of CF3-Alkynes
0640
Copper-Catalyzed Enantioselective Borylstannation
0641
Direct Cross-Coupling of Diaryl Zinc Reagents
0642
Palladium-Catalyzed Carbonyl Allylation of Aldehydes and Isatins
0643
Cp2TiCl2-Catalyzed cis-Hydroalumination of Amines
0644
Nickel-Catalyzed Monofluoromethylation
0645
Copper-Mediated Trifluoromethylthiolation
0646
Synthesis of ortho-Boronated Phosphine Boranes
0647
Ruthenium(II)-Catalyzed C–H Arylation of Anilides
0648
Copper-Mediated C–H Sulfonylation of Benzoic Acid Derivatives
0649
Stereoselective Synthesis of γ-Substituted Homoallylic Alcohols
0650
Silaboration and Diboration of Alkynoates
0651
syn/anti-Selective Carboboration of Alkenes
0652
Reductive Coupling of Esters with Benzophenones Using Low-Valent Titanium
0653
Selective Hydrogenation of Potassium Trifluoroborates

Organo- and Biocatalysis

z655
All PDFs of this category
0655
Biocatalytic Site-Selective Halogenation of Large Bioactive Molecules
0656
Arylation of Allylic C–H Bonds by Cooperative Organo- and Photoredox Catalysis
0657
Chiral Phosphine Catalyzed [4+1] Annulations of Amines with Allenes
0658
Brønsted Acid Promoted Synthesis of Functionalized Furans
0659
Intramolecular Hydroacylation of Unactivated Alkenes by NHC Catalysis
0660
Brønsted Acid Catalyzed [4+2] Addition of Alkenes with ortho-Quinone Methides
0661
Oxidative C–H Alkenylation and Arylation of Tetrahydropyridines and Derivatives
0662
Functionalized Hydrocarbazoles by Catalytic Desymmetrization

Polymer-Supported Synthesis

z663
All PDFs of this category
0663
Hydrogen Autotransfer by Au/Pd Nanoparticles with Lewis Acids
0664
Cyclization of Tertiary Anilines with Maleimides Using P25/NiO
0665
SPS of Seragamide A via Relay-Ring-Closing Metathesis
0666
Tandem Hydroformylation–Imination–Hydrogenation with Supported Rh/NHC
0667
Hydrodeoxygenation of Vicinal OH Groups Using ReOx–Pd/CeO2
0668
Preparation of β-Amino Carbonyl Compounds by Different Pathways
0669
Solid-Supported 9-Amino-9-deoxy-epi-quinine as Chiral Organocatalyst
0670
Coupling of Aryl Halides with Disulfides Catalyzed by Cu-Doped ZSM-5
0671
One-Pot Synthesis of N-Aryl Dithiocarbamates
0672
Reduction of Quinolines with Formic Acid Using Au/TiO2-R
0673
The Heck Reaction Using Pd/Fe3O4@PIL-NH2
0674
Flow Aerobic Oxidation of Alcohols Using a Supported Nano Platinum Catalyst
0675
Synthesis of Benzopyranopyrimidines Using PS-Supported PTSA