DOI: 10.1055/s-00000084

Synthesis

Issue 22 · Volume 48 · November 2016 DOI: 10.1055/s-006-32752

review

3821
Rossi, Renzo; Lessi, Marco; Manzini, Chiara; Marianetti, Giulia; Bellina, Fabio: Direct (Hetero)arylation Reactions of (Hetero)arenes as Tools for the Step- and Atom-Economical Synthesis of Biologically Active Unnatural Compounds Including Pharmaceutical Targets
https://www.thieme-connect.de/media/synthesis/201622/i_e0361_ga_10-1055_s-0036-1588303.gif

short review

3863
Rintjema, Jeroen; Kleij, Arjan W.: Substrate-Assisted Carbon Dioxide Activation as a Versatile Approach for Heterocyclic Synthesis
https://www.thieme-connect.de/media/synthesis/201622/i_z0459_ga_10-1055_s-0035-1562520.gif
3879
Besson, Thierry; Fruit, Corinne: Recent Developments in Microwave-Assisted Metal-Catalyzed C–H Functionalization of Heteroarenes for Medicinal Chemistry and Material Applications
https://www.thieme-connect.de/media/synthesis/201622/i_z0461_ga_10-1055_s-0035-1562608.gif
3890
Vargas-Caporali, Jorge; Juaristi, Eusebio: The Diamino Analogues of Privileged Corey–Bakshi–Shibata and Jørgensen–Hayashi Catalysts: A Comparison of Their Performance
https://www.thieme-connect.de/media/synthesis/201622/i_z0464_ga_10-1055_s-0035-1562793.jpg

paper

3907
Lesma, Giordano; Luraghi, Andrea; Rainoldi, Giulia; Mattiuzzo, Elena; Bortolozzi, Roberta; Viola, Giampietro; Silvani, Alessandra: Multicomponent Approach to Bioactive Peptide–Ecdysteroid Conjugates: Creating Diversity at C6 by Means of the Ugi Reaction
https://www.thieme-connect.de/media/synthesis/201622/i_z0190_ga_10-1055_s-0035-1562497.gif
Supporting Information
3917
Coman, Anca G.; Paraschivescu, Codruta C.; Hadade, Niculina D.; Juncu, Andrei; Vlaicu, Ovidiu; Popescu, Costin-Ioan; Matache, Mihaela: New Acyloxymethyl Ketones: Useful Probes for Cysteine Protease Profiling
https://www.thieme-connect.de/media/synthesis/201622/i_t0294_ga_10-1055_s-0035-1562781.gif
Supporting Information
3924
Zhang, Lutao; Tang, Dong; Gao, Jing; Wang, Jing; Wu, Ping; Meng, Xu; Chen, Baohua: Direct Access to 1,3,5-Trisubstituted 1H-1,2,4-Triazoles from N-Phenylbenzamidines via Copper-Catalyzed Diamination of Aryl Nitriles
https://www.thieme-connect.de/media/synthesis/201622/i_f0248_ga_10-1055_s-0035-1562490.gif
Supporting Information
3931
Akimura, Nozomi; Fujii, Ayaka; Kamada, Fuma; Nogiwa, Ryoki; Yamamoto, Syota; Sato, Teppei; Ishikawa, Syuji; Okazaki, Tatsuya; Kaneda, Kyosuke: Synthesis of Tetracyclic Molecules Containing Medium-Sized Heterocycles: Scope Expansion of Cascade Nicholas and Pauson–Khand Methodology
https://www.thieme-connect.de/media/synthesis/201622/i_f0377_ga_10-1055_s-0035-1562780.gif
Supporting Information
3941
Yu, Yanhan; Yue, Yixia; Wang, Deqiang; Li, Xue; Chen, Chunxia; Peng, Jinsong: Modular Synthesis of Quinazolinone-Fused Phenanthridinones by a Palladium-Catalyzed Cascade C–H/N–H Arylation Process
https://www.thieme-connect.de/media/synthesis/201622/i_h0154_ga_10-1055_s-0035-1561481.gif
Supporting Information
3951
Yin, Hongli; Meng, Zhe; Liu, Bo: Construction of the Core Structure of Trichotomone
https://www.thieme-connect.de/media/synthesis/201622/i_h0225_ga_10-1055_s-0035-1562491.gif
Supporting Information
3957
Kamiyama, Takuya; Sigrist, Lukas; Cvengroš, Ján: Synthesis of Tröger’s Base Analogues via a Phase-Transfer-Catalyzed Double Aza-Michael Reaction under Base-Free Conditions
https://www.thieme-connect.de/media/synthesis/201622/i_t0263_ga_10-1055_s-0035-1562461.gif
Supporting Information
3965
Lashmanova, Eugeniya A.; Rybakov, Victor B.; Shiryaev, Andrey K.: Synthesis of Adamantylated Pyrimidines Using the Biginelli Reaction
https://www.thieme-connect.de/media/synthesis/201622/i_z0221_ga_10-1055_s-0035-1562459.gif
Supporting Information
3971
Omura, Ryuji; Fujiya, Akitoshi; Yamaguchi, Eiji; Tada, Norihiro; Miura, Tsuyoshi; Itoh, Akichika: One-Pot Aerobic Photooxidative Darzens Reaction from Styrene and Benzyl Alcohol via Phenacyl Iodide and Benzaldehyde by Using­ Iodine
https://www.thieme-connect.de/media/synthesis/201622/i_f0297_ga_10-1055_s-0035-1562455.gif
Supporting Information
3976
Ye, Xinglin; Yuan, Jianjun; Zhou, Yirong; Deng, Zhihong; Mao, Xuechun; Peng, Yiyuan: Palladium-Catalyzed Cross-Coupling of 4-Tosyloxyquinazolines with Organoindium Reagents: An Efficient Route to 4-Substituted Quinazolines
https://www.thieme-connect.de/media/synthesis/201622/i_h0230_ga_10-1055_s-0035-1562504.gif
Supporting Information
3985
Wang, Qi; Wang, Meirong; Li, Hui-Jing; Zhu, Shuai; Liu, Ying; Wu, Yan-Chao: Synthesis of Quinolines via Iron-Catalyzed Redox Condensation of Alcohols with 2-Nitrobenzyl Methyl Ether/2-Nitrobenzyl Alcohols
https://www.thieme-connect.de/media/synthesis/201622/i_h0276_ga_10-1055_s-0035-1562496.gif
Supporting Information
3996
Kadam, Kishorkumar S.; Gandhi, Thirumanavelan; Gupte, Amol; Gangopadhyay, A. K.; Sharma, Rajiv: Alkyl Nitrites: Novel Reagents for One-Pot Synthesis of 3,5-Disubstituted Isoxazoles from Aldoximes and Alkynes
https://www.thieme-connect.de/media/synthesis/201622/i_z0198_ga_10-1055_s-0035-1561464.gif
Supporting Information
4009
Mondal, Susmita; Samanta, Sadhanendu; Singsardar, Mukta; Mishra, Subhajit; Mitra, Shubhanjan; Hajra, Alakananda: Zwitterionic-Type Molten Salt Catalyzed Iodination in Water: Synthesis of Iodoimidazoheterocycles
https://www.thieme-connect.de/media/synthesis/201622/i_z0258_ga_10-1055_s-0035-1562492.gif
Supporting Information

book review

4016
Lutz, Ackermann: Science of Synthesis: Catalytic Transformations via C–H Activation, Workbench Edition, 2 Vol.