Synfacts

Issue 04 · April 2019

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A48
Zanda, Matteo: SYNFORM ISSUE 2019/04

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Synthesis of Natural Products and Potential Drugs
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Synthesis of an HIV-1 Integrase Allosteric Site Inhibitor FREE ACCESS

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Synthesis of Paspaline A and Emindole PB

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Synthesis of Eburnane-Type Alkaloids FREE ACCESS

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Synthesis of (+)-Dysoline

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Synthesis of Atuveciclib

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Synthesis of a Glucokinase Activator

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Synthesis of Gefitinib

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Asymmetric Total Synthesis of (+)-Laurallene

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Asymmetric Synthesis of Netarsudil

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0342
Synthesis of 2′-Fluoro-6′-methylene-carbocyclic Adenosine (FMCA)

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0343
Syntheses of Δ¹²-Prostaglandin J Natural Products

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Synthesis of LX2761

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Synthesis of (+)-Pleurocins A and B

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Synthesis of (±)-Estrone FREE ACCESS

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Synthesis of Heterocycles
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0347
Three-Component Synthesis of Quinazolinones

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0348
New Biocatalytic Synthesis of Caprolactone by Oxidative Lactonization

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0349
Organocatalytic Synthesis of Enantioenriched Five- and Six-Membered Cyclic Ureas

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0350
Synthesis of Indolo[1,2-α]indole Derivatives by Gold(I)-Catalyzed Cycloisomerization

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0351
Gold Carbene Route to Several Classes of Azaheterocycles

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0352
Photodecarboxylative Azidation of Cyclic Amino Acids with Rhodamine 6G

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0353
Palladium(II)-Catalyzed Activation for Nucleophilic Substitution Reactions

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0354
Cobalt-Catalyzed Synthesis of Quinolines and Acridines from Anthranils

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0355
Spiroindolines by Visible-Light-Mediated Intramolecular Cycloadditions

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0356
Synthesis of Pyrrolophenanthridine Alkaloids by the Schmidt Reaction

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0357
Synthesis of 2-Aminopyrroles and Quinoline-Based Polyazaheterocycles

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0358
Titanocene-Catalyzed Synthesis of Functionalized Ring-Fused Piperidines

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0359
Electrochemical Synthesis of Fluorinated 2-Oxazolines

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0360
Synthesis of Carbazoles and Indolines by Gold-Catalyzed Diels–Alder Reactions

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0361
Synthesis of (5E)-5-(Iodomethylene)-1,3-selenazolidin-2-ones

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Synthesis of Materials and Unnatural Products
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0363
A New Twist on Sydnones FREE ACCESS

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0364
A Mechanically Stabilized Helical Chiral Macrocycle

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0365
Thiophenes through Thiolates

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0366
Copper-Catalyzed Oxidation of Siloxanes to Polar Siloxanes

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0367
Open and Shut Synthesis of an Oligoparaphenylene Dual Nanohoop

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0368
Stars Align for Liquid Crystals via a New Supramolecular Click Mechanism

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0369
Mind the Gap: Finite Nanotubes with Periodic Wall Defects

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0370
A Rare Example of a Retro Baeyer–Villiger Reaction

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0371
Spontaneous CO₂ Conversion into Polymeric Materials

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0372
Loose Canon: Tunable Quiniodal Macrocycles with Canonical and Zwitterionic Ground States

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0373
Copper-Mediated Homocoupling for Naphthotetraindole Synthesis

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0374
Everybody Loves Pie: Nitrogen-Doped Pyrenes

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Metals in Synthesis
z0375
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0375
Cyclohexane Desymmetrization via Rhodium-Catalyzed C–H Activation FREE ACCESS

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0376
Iron(III)-Catalyzed Carbonyl-Olefin Metathesis of Aliphatic Ketones

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0377
Enantioselective Arylative Trifluoromethylation of Alkenes FREE ACCESS

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0378
Bimetallic Hydroaminomethylation of α-Olefins

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0379
Nickel-Catalyzed Alkylation of Heterocycles

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0380
Cross-Dehydrogenative Heteroarylation of Cyclic Amines

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0381
Asymmetric C(sp³)–H Arylation Through a Hybrid Palladium Catalyst

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0382
Asymmetric C(sp³)–H Amidation of Thioamides Catal-yzed by a Cobalt^III/Chiral Carboxylic Acid Hybrid System

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0383
Diastereoselective Formation of All-cis-(Multi)Fluorinated Piperidines

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0384
Iron(II)-Catalyzed Alkyl Heck Coupling

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0385
Enantioselective Iron-Catalyzed Couplings of Aldehydes and Alkenes

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0386
Cobalt(III)-Catalyzed [4+2] Annulation

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0387
Cobalt-Catalyzed [2+2] Cycloaddition

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0388
Chromium-Catalyzed Asymmetric Allylation

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0389
Synthesis of Fully Substituted Cyclopentenones

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0390
Rhodium-Catalyzed Enantioselective Cyclopropanations

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0391
Sequential meta-C–H/ipso-C–O Functionalization of Phenols via Directing-Group Strategy

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0392
Copper-Catalyzed Remote Trifluoromethylation

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0393
A New Late-Stage Defluorosilylation

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0394
Catellani Reaction: Synthesis of o,o′-Disubstituted Vinylarenes FREE ACCESS

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0395
Copper-Catalyzed Enantioselective Reduction of α,β-Unsaturated Esters FREE ACCESS

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0396
Iridium-Catalyzed Three-Component Coupling Reaction

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0397
Palladium-Catalyzed Dearomative Intermolecular [4+1] Spiroannulation by C(sp³)–H Activation

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0398
Iridium-Catalyzed Asymmetric Allylic O-Alkylation of Ketones

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0399
Iron-Catalyzed Carbon (sp²)–Carbon (sp²) Oxidative Homo-Coupling

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0400
Molybdenum-Catalyzed Direct Amination of Boronic Acids

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0401
Stereoselective Synthesis of anti-Isomers of γ-Boryl-Substituted Homoallylic Alcohols

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0402
Enantioselective Aryl Transfer using Chiral Lithium Amido Aryl Zincates

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0403
Dual Photoredox/Copper Catalysis for C–H Functionalizations

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0404
Gold-Catalyzed Temperature-Controlled Divergent Hydroamination/Cycloaddition Cascade Reactions

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Polymer-Supported Synthesis
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0405
Hydroamination of Terminal Alkynes on Gold Nanoclusters

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0406
Selective Catalytic Hydrogenation of α,β-Unsaturated Aldehydes FREE ACCESS

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0407
Oxidation of Alcohols on Thermoresponsive-Polymer-Supported TEMPO

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0408
A³ Coupling Reactions on Green-Synthesized Gold Nanoparticles

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0409
Palladium-Catalyzed Carbocyclization–Borylation of Enallenols

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0410
Tandem Catalytic C–H Arylation/Suzuki–Miyaura Coupling

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0411
Photocatalytic Coupling Reactions on a Mixed-Ligand Metal–Organic Framework

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0412
Knoevenagel–Michael and Click Reactions on a Cu(II)/Natural Phosphate Catalyst

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0413
Pd(II)-Complex-Catalyzed Mizoroki–Heck Reaction in γ-Valerolactone

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0414
Synthesis of Pyranopyrazoles Using TiO₂-Coated Fe₃O₄-Immobilized Tungstic Acid

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0415
Palladium-Photocatalyzed Self-Condensation of Primary Amines

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0416
Synthesis of 4H-Pyrimido[2,1-b]benzothiazoles with a Heterogeneous Cu(II) Catalyst

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0417
Denitrative Cyclizations of β-Nitrostyrenes on Supported Pd Nanoparticles

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0418
Synthesis of Benzimidazoles Promoted by Rh@PS

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Organo- and Biocatalysis
z0419
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0419
Application of Chemoinformatics in Asymmetric Catalysis FREE ACCESS

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0420
Asymmetric Enzymatic Aminohydroxylation of Styrenyl Olefins

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0421
Directed Evolution Permits Heme-Protein-Catalyzed sp³-C–H Alkylation

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0422
Asymmetric Synthesis of Trifluoromethylated Spirooxindole Lactones

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0423
Asymmetric Synthesis of All-Carbon Spirocycles by a Stetter/Aldol Cascade

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0424
Chiral Bifunctional Phase-Transfer Catalysts for Asymmetric Aminations

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0425
Electrophilic Sulfenylation of Indoles by P^III/P^V=O Catalysis

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0426
NHC-Catalyzed Aza-Stetter Reaction of Aldimines To Give 3-Methylenechromanones

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0427
Aminoxyl-Catalyzed Electrochemical Diazidation of Alkenes

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0428
The Knoevenagel Condensation FREE ACCESS

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Chemistry in Medicine and Biology
z0429
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0429
A Chemoselective Conjugation of Peptides with Electron-Rich (Hetero)Arenes FREE ACCESS

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0430
Specific Functionalization of Cysteine and Lysine Using Dinitroimidazoles

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0431
Late-Stage Functionalization of Complex Primary Sulfonamides via NHC Catalysis

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0432
Application of Hemithioindigo Photoswitches in Photopharmacology

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0433
Synthesis of Aglaroxin C Analogues for Hepatitis C Viral Infection Inhibition

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0434
Synthesis of a cGAMP Analogue

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0435
A Small Clickable and Photoconvertible Fluorophore

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0436
Synthesis of AWZ1066S, an anti-Wolbachia Drug Candidate

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0437
Pyrazolopyrimidines: Molecular Correctors for MALT1-Related Immune Defects

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0438
Selective Targeting of p38 MAPK Isoforms Using PROTACs

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0439
Synthesis of Human Interleukin-8 by Native Chemical Ligation FREE ACCESS

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0440
Synthesis of a Fluorescent Probe for Cell Surface Phosphatidylserine

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0441
Synthesis of ‘Stretched’ Isosteres of Saturated Nitrogen Heterocycles

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0442
Targeting Zinc Homeostasis in Cancer

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0443
A Glutathione-Labile Oligonucleotide Protecting Group

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Peptide Chemistry
z0445
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0445
O-Glycosylation of Unprotected Peptides FREE ACCESS

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0446
One-Pot Peptide Modifications Using the MeDbz Linker

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0447
Synthesis of Free α-Amino Acids from 1,2-Diols

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0448
Two-Step Strategy for Thioamide Bond Formation by Using an Ynamide

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0449
Photoredox-Catalyzed α-Fluoro-α-Amino Acid Synthesis

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0450
Photoredox Catalysis with Amino Acid- and Peptide-Derived Katritzky Salts

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0451
Petasis Reaction for Late-Stage Functionalization of Peptides

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0452
Photocatalytic Decarboxylative C(sp³)–H Alkylation of Glycine or Peptides

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0453
Manganese-Catalyzed Synthesis of Acylic, Hybrid, and Stapled Peptides

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0454
Palladium-Catalyzed Asymmetric Aminomethylation

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0455
Total Chemical Synthesis of a Glycoprotein by Native Chemical Ligation FREE ACCESS

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Flow Chemistry
z0457
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0457
Automated Titration of Organometallic Reagents in Continuous Flow

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0458
Oxidation of Csp³–H Bonds in Flow Using Methyl(trifluoromethyl)dioxirane

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0459
Continuous-Flow Chemoenzymatic Dynamic Kinetic Resolution of Amines

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0460
Continuous-Flow Diazotization

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Erratum
0461
Gong, T.-J; Hea, S.-J; Lu, X; Pi, J.-J; Fu, Y; Wang, X.-X: Defluorinative Alkylation using Redox-Active Esters

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0461
Seidl, F J; Min, C; Lopez, J A; Burns, N Z: Regio- and Enantioselective Haloazidation of Allylic Alcohols

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