Synfacts

Issue 06 · June 2020

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SYNFORM ISSUE 2020/06 FREE ACCESS

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Synthesis of Natural Products and Potential Drugs
z0617
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0617
Asymmetric Total Synthesis of (+)-Waihoensene FREE ACCESS

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0618
Total Synthesis of (±)-Ganocin A

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0619
Synthesis of Monobactam Antibiotic LYS228 FREE ACCESS

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0620
Synthesis of Lamivudine

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0621
Synthesis of PPARα Agonist GW641597X

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0622
Synthesis of Taniborbactam (VNRX-5133)

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0623
Total Synthesis of (+)-Cotylenin A

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0624
Synthesis of (+)-Cerapicol

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0625
Synthesis of (+)-Conocenolide E and (+)-10,11,12-Trihydroxytremulenone

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0626
Synthesis of SUVN-911

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0627
One-Pot Synthesis of a TGFβRI Inhibitor

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0628
Synthesis of a Janus Kinase Inhibitor

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0629
Total Synthesis of Pyrolaside B

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0630
Synthesis of Islatravir

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0631
Total Synthesis of (±)-Periplanone B FREE ACCESS

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Synthesis of Heterocycles
z0633
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0633
Synthesis of Alkene Carbonates through Carbon Dioxide Fixation Using Perfluorinated Triol Catalysts

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0634
Triazapentalene Synthesis by N–N Bond Formation

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0635
Sulfinylation of Indoles, Pyrroles, and Thiophenes

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0636
Ligand-Free Palladium(II)-Mediated Synthesis of 2,4-Disubstituted 1,3-Thiazoles

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0637
Determination of Basicities and Nucleophilicities of a Series of Organocatalysts FREE ACCESS

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0638
Direct C-2 Carboxylation of Electron-Deficient Indoles

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0639
Iridium-Catalyzed Synthesis of Indoles and Indolines

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0640
Synthesis of β-Lactams by a Kharasch–Sosnovsky Reaction

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0641
Nickel(0)-Catalyzed Enantioselective Synthesis of Butenolides and Lactams

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0642
Synthesis of Seven- and Nine-Membered Heteroatom-Containing Rings

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0643
Synthesis of 1,2,4-Oxadiazoles from Alkynes and Nitriles

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0644
Silver Acetate-Catalyzed Groebke-Blackburn-Bienayme Reaction to Synthesize Imidazo[1,2-a]Pyridines

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0645
Synthesis of [6,5]-Spirocycles through Redox-Neutral Cyclizations of Aurones

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0646
Stereoselective C–H Cyclopropanation of N-Phenoxysulfonamides

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0647
Access to Functionalized Chromanes by Asymmetric [4+2]-Cycloaddition

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Synthesis of Materials and Unnatural Products
z0649
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0649
Big Waggles Don’t Throw Off the Rotation FREE ACCESS

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0650
Octapodal Corannulene Porphyrin Captures Fullerene

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0651
A Shocking Approach to Axially Chiral Aldehydes

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0652
Whew, Vinyl-y! Gold-Catalyzed Synthesis of Vinyl Ethers from Diynes and Ketones

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0653
S_NAr-Based Synthesis of Chalcogen-Containing Helicenes

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0654
New Triarylamine Radical Shakes the Blues

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0655
A Greener Way to Asymmetrical Triarylamines

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0656
Lowering the LUMO: A Macrocyclic Organoborane

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0657
Living Polymers via Cumulation of β-Pinene

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0658
Diradicaloid Cage with 3D Global Aromaticity

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0659
Convert that COF

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0660
Polyynes to Polyfused Chalcogenophenes

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Metals in Synthesis
z0661
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0661
Nickel-Catalyzed Cross-Electrophile Coupling using Electrochemistry FREE ACCESS

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0662
Hydrogenation of Alkenes and Arenes Catalyzed by Bulky Alkaline Earth Metal Amides

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0663
Manganese-Catalyzed Methylation of C(sp³)–H Bonds α to Heteroatoms FREE ACCESS

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0664
Rhodium-Catalyzed Asymmetric Synthesis of Axially Chiral Polyaromatic Hydrocarbons

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0665
Dual-Metal Photocatalyzed Diastereoselective Isomerization of Allyl Chlorides to Chlorocyclopropanes

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0666
1,2-Diarylation of Alkenes Using Gold Catalysis

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0667
Preparation of Biaryls by Organic Oxidants

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0668
Decarboxylative para-Selective C–H Functionalization

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0669
Chromium-Catalyzed Cyclopropanation

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0670
Picolinate-Directed Arene meta-C−H Amination via FeCl₃ Catalysis

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0671
Oximes as Directing Groups for Iridium-Catalyzed β-Alkynylation of Primary C(sp³)–H Bonds

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0672
Enantioselective Aminomethylations

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0673
Enantioselective Conjunctive Cross-Couplings Leading to α-Boryl Allenes

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0674
Enantioselective Radical Reactions by Cu(I)/Chiral Phosphoric Acid Cooperative Catalysis

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0675
Cobalt-Catalyzed Radical Hydroxytrifluoromethylation of Alkenes

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0676
C–H Functionalization of Alkanes Using Cerium Catalysis

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0677
Nickel-Catalyzed Branched-Selective α-Crotylation of Ketones with 1,3-Butadiene

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0678
Synthesis of 5-Aryltetrazoles

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0679
Nickel-Catalyzed Decarbonylative Amination of Esters

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0680
Titanium-Catalyzed Anti-Markovnikov Alcohol Synthesis via Epoxide Ring Opening Using Green Light

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0681
Borocarbonylative Copper-Catalyzed Four-Component Coupling

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0682
Nickel-Catalyzed Acylation of Pyridinium Salts

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0683
Ni-Catalyzed Synthesis of 1,1-Diarylalkanes via Chain-Walking Hydroarylation of Alkenes with Boronic Acids

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0684
Palladium-Catalyzed Enantioselective Hydroarylation of Alkenes Using a Chiral Transient Directing Group

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0685
Enantioenriched Amine Derivatives by Pd- and Cu-Catalyzed Arylation and Acylation of Alkylzincs

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0686
Asymmetric Hydrogenation–Reductive Amination Cascade for the Synthesis of Julolidines

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0687
Electrophilic Amination of Diorganozinc Reagents Using N-Hydroxylamine Benzoates FREE ACCESS

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Polymer-Supported Synthesis
z0689
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0689
An Atomically Dispersed Platinum Catalyst for the Catalytic Diboration of Alkynes

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0690
Domino Knoevenagel/Hetero-Diels–Alder Reaction Catalyzed by Magnetically Separable Silica

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0691
SAB-15-Supported Rose Bengal as a Heterogeneous Photoredox Catalyst FREE ACCESS

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0692
C–H Halogenation of 2-Arylpyridines on Salen-Based Hypercrosslinked Polymer-Supported Palladium

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0693
Catalytic Hydrogenation and Photooxidation on a Flavin-Containing Mesoporous Network Polymer

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0694
Synthesis of Cyclohexylamines Catalyzed by Nickel Supported on Alumina

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0695
Preparation of 3-Alkoxyquinoxalin-2-ones by Electrooxidative C–H/O–H Cross-Coupling

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0696
Pd-Catalyzed Z-Selective Transfer Hydrogenation of Internal Alkynes with Butane-1,4-diol

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0697
Photocatalytic Oxidation of Alcohols to Aldehydes and Ketones Catalyzed by TiO₂-P25

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0698
Copper(II)/Ascorbic Acid-Coated TiO₂ Photocatalyst for Aerobic Oxidation of Benzylic Alcohols

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0699
Synthesis of Anilines and N-Heterocyclic Aromatic Compounds Catalyzed by Ni/C Nanocomposites

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0700
Hydrogenation of Nitroarenes by Formic Acid on N-Doped-Carbon-Supported Iron Nanoparticles

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Organo- and Biocatalysis
z0701
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0701
Photoexcitation of an Acridine Radical Generates a Strong Organic Single-Electron Reductant FREE ACCESS

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0702
Novel Borate-Ion Catalyzed Asymmetric Prins-Type Cyclization

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0703
Biocatalytic Oxidation of Silanes to Silanols

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0704
Chiral Phosphoric Acid Catalyst Serves a Dual Function in an Asymmetric Antilla Allylation of Aldehydes

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0705
HyperBTM-Catalyzed Asymmetric Tandem Sequential Synthesis of Tetrahydroindolizines

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0706
Strongly Acidic and Enzyme-Like Catalysts in Diels–Alder Reactions with Cross-Conjugated Dienophiles

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0707
A Catalytic Enantioselective Allenoate–Claisen Rearrangement

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0708
A Transition Metal-Free Catalytic Approach Towards Selective Transformations of ortho-Quinone Methides

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0709
Supramolecular Catalysis Permits Access to the Presilphiperfolanol Framework

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0710
Trapping an Achiral Anion Inside a Chiral Macrocycle for Enantioselective Catalysis

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0711
An Asymmetric Tail-to-Head Cyclization of Neryl Chloride Analogues

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Chemistry in Medicine and Biology
z0713
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0713
α-Ketoamide Inhibitors of SARS-CoV-2 Main Protease FREE ACCESS

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0714
Azithromycin – An Antibiotic to Fight COVID-19? FREE ACCESS

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0715
Crystal Structure of the Main Protease of Human Coronavirus NL63 FREE ACCESS

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0716
Hydroxychloroquine – An Antimalarial to Fight COVID-19? FREE ACCESS

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0717
C–H Trifluoromethylation Enabled by a Combination of Decatungstate and Copper Catalysis

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0718
Irreversible Covalent Inhibition of TrxR1 Prevents STAT3-Dependent Transcription Activation

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0719
MicroMap: Precise Proximity Labeling of Cell Surface Proteins

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0720
TREK Channel Family Activator for Relief of Pain and Neurogenic Inflammation

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0721
Unleashing the Full Power of the Streptavidin–Biotin Technology in Cellular Uptake

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0722
Phosphoglycolipids with Immunomodulatory Activity

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0723
Photocaged Dopamine Receptor Ligands

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0724
A Vincamine-Derived HCRTR2 Agonist Prevents Morphine-Seeking Behavior in Mouse Models

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0725
In Vivo Optochemical Control of Glutamate Receptors with Cloaked Glutamates

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0726
Accelerating Aiolos Ablation

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0727
Clickable UDP-Galactose Analogues

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Peptide Chemistry
z0729
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0729
Iridium-Catalyzed Synthesis of Quaternary α-Trifluoromethyl α-Amino Acids

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0730
Tantalum-Catalyzed Formation of Amide Bonds

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0731
Tantalum-or Titanium-Catalyzed Peptide Synthesis FREE ACCESS

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0732
Organocatalytic Synthesis of Axially Chiral Biaryl Amino Acids

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0733
Copper-Catalyzed Three-Component Coupling to Form α-Halo β-Amino Acid Derivatives

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0734
Copper-Catalyzed Stereoselective Synthesis of α-Amino Acid Precursors

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0735
Ytterbium-Catalyzed Synthesis of γ-Amino Acid Derivatives

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0736
Asymmetric Mannich-Type Reaction to Access Unnatural Amino Acids

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0737
Synthesis of Unnatural α-Amino Acids under Visible-Light Irradiation

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0738
Modification of Peptides through C(sp³)–H Alkylation

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0739
Catalyst-Free Synthesis of α-Amino Acid Derivatives

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0740
Metal-Free Synthesis of α-Amino Acid Derivatives from α-Bromo Amides

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0741
Chemical Ligation to Synthesize N-Hydroxy Peptides from O-Acyl Hydroxamic Acids FREE ACCESS

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Flow Chemistry
z0743
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0743
Peptide Synthesis in Continuous Flow

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0744
Aryl Alkyl Ether Formation via Copper-Catalyzed Photoredox Driven C–O Cross-Coupling

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0745
Flow Synthesis of Anilines through Photoredox/Ni(II)-Catalyzed C–N Cross-Coupling: Tetracaine

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0746
Aryl, Heteroaryl, and Benzylic Functionalization Using Potassium Organometallics Generated in Flow

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Erratum
0747
V1, Rotate: [1.1.1]Propellane Prepared to Takeoff FREE ACCESS

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