Synfacts

Issue 04 · April 2024

Recommend Journal

Issue
Synform
A053
SYNFORM ISSUE 2024/04 FREE ACCESS

Full Text

PDF (3031 kb)
Synthesis of Natural Products
z0335
All PDFs of this category

Full Text

PDF (336 kb)
0335
Total Synthesis of (±)-Daphenylline FREE ACCESS

Full Text

HTML

PDF (142 kb)
0336
Enantioselective Total Synthesis of (–)-Daphenylline

Full Text

HTML

PDF (90 kb)
0337
Synthesis of (+)-Archangiumide

Full Text

HTML

PDF (83 kb)
0338
Total Synthesis of (+)-Bipolarolide A

Full Text

HTML

PDF (79 kb)
0339
Total Synthesis of (+)-Heilonine

Full Text

HTML

PDF (86 kb)
0340
Total Synthesis of (+)-Pedrolide

Full Text

HTML

PDF (85 kb)
0341
Total Synthesis of (+)-Zaragozic Acid C FREE ACCESS

Full Text

HTML

PDF (123 kb)
Synthesis of Heterocycles
z0343
All PDFs of this category

Full Text

PDF (372 kb)
0343
Efficient Syntheses of Complex Benzoxaboracycles

Full Text

HTML

PDF (73 kb)
0344
Late-Stage Selective Functionalization for Bioactive Indole Derivatives

Full Text

HTML

PDF (87 kb)
0345
1,3-Dipolar Cycloaddition Approach to Functionalized Tetrahydropyridines

Full Text

HTML

PDF (77 kb)
0346
Palladium-Mediated Synthesis of Functionalized Unsaturated Dicarbonyl Compounds

Full Text

HTML

PDF (84 kb)
0347
Chemodivergent Cyclization of Propargylamines to Enable Indole and Quinoline Heterocycles

Full Text

HTML

PDF (90 kb)
0348
Synthesis of Amides Using Triazine Esters as Stable Acylation Reagents

Full Text

HTML

PDF (71 kb)
0349
Selective Synthesis of exo- and endo-3-Azabicyclo[3.1.0]hexane-6-carboxylates

Full Text

HTML

PDF (86 kb)
0350
Synthesis of Fused Imidazoles via Iron-Catalyzed C(sp³)–H Amination–Cyclization

Full Text

HTML

PDF (70 kb)
0351
Skeletal Editing of Indazoles via Silver-Catalyzed Carbene Insertion FREE ACCESS

Full Text

HTML

PDF (145 kb)
0352
Copper-Catalyzed Synthesis of 4,5,6-Trisubstituted Pyrimidines

Full Text

HTML

PDF (100 kb)
0353
Diastereoselective Scandium-Catalyzed Route to Difluorinated Pyrrolidines

Full Text

HTML

PDF (79 kb)
Synthesis of Materials and Unnatural Products
z0355
All PDFs of this category

Full Text

PDF (348 kb)
0355
N-Heterocyclic Olefins with Applications to ROP FREE ACCESS

Full Text

HTML

PDF (140 kb)
0356
Sequential Annulation of Arene Diamines

Full Text

HTML

PDF (88 kb)
0357
A Facile Access to Phosphet-2-ones

Full Text

HTML

PDF (73 kb)
0358
Photochemical Conversion of Nitroarenes to Bicyclic Pyrrolines

Full Text

HTML

PDF (86 kb)
0359
Rippled Nanographene Rich in Nonhexagons

Full Text

HTML

PDF (77 kb)
0360
N-doped Holey Nanographene

Full Text

HTML

PDF (72 kb)
0361
Azaboraacenium with Photo- and Air-Stability

Full Text

HTML

PDF (71 kb)
0362
Antiaromatic Chalcogenopyrano Chalcogenopyrans

Full Text

HTML

PDF (76 kb)
0363
A Rotaxane of [6]Cycloparaphenylene

Full Text

HTML

PDF (72 kb)
0364
A One-Pot Cascade Synthesis of Phenanthrenes

Full Text

HTML

PDF (80 kb)
0365
One-Pot Synthesis of 1,4-Azaborines from Diarylamide

Full Text

HTML

PDF (76 kb)
Metals in Synthesis
z0367
All PDFs of this category

Full Text

PDF (1279 kb)
0367
Palladium-Catalyzed Carbonylative Cycloaddition of Acylsilanes and Imines to Access β-Lactams FREE ACCESS

Full Text

HTML

PDF (135 kb)
0368
Synthesis of 2-Aminopyridines from 1,2,3,4-Tetrazoles via Iron/Blue Light-Promoted Benzylic C–H Activation

Full Text

HTML

PDF (84 kb)
0369
Terminal C–H Borylation Enabled by Visible Light Iron Photocatalysis FREE ACCESS

Full Text

HTML

PDF (122 kb)
0370
Synthesis of Branched Sulfides via Cobalt-Catalyzed Markovnikov Thiyl Radical Addition to Alkenes

Full Text

HTML

PDF (80 kb)
0371
Asymmetric Hydrocyanation of Aromatic Alkenes by Merging Photoredox and Copper Catalysis

Full Text

HTML

PDF (542 kb)
0372
Synthesis of Diverse 1,5-Boroacylated Products via Cooperative Cu/Pd-Catalysis

Full Text

HTML

PDF (73 kb)
0373
Nickel-Catalyzed Intramolecular Carboamination: Efficient Synthesis of N-Heterocycles

Full Text

HTML

PDF (75 kb)
0374
Rhodium-Catalyzed Asymmetric Aziridination of Unactivated Terminal Olefins

Full Text

HTML

PDF (71 kb)
0375
Direct Carboxylation of Secondary Alkyl Bromides under Dual Photoredox and Nickel Catalysis

Full Text

HTML

PDF (82 kb)
0376
Synthesis of Arylamines via a C–N Coupling, Ring Expansion and Dehydrogenative Aromatization Cascade

Full Text

HTML

PDF (81 kb)
0377
A Copper-Catalyzed [2,3]-Stevens Rearrangement to Access Functionalized Tetrahydro Oxepines

Full Text

HTML

PDF (82 kb)
0378
Enantioselective Synthesis of Isoindolinones via Cobalt-Catalyzed C–H Carbonylation

Full Text

HTML

PDF (87 kb)
0379
Pd/Visible Light-Promoted 2,5-Difunctionalization/Spirocyclization of Alkene-Tethered Furans

Full Text

HTML

PDF (82 kb)
0380
Three-Component Defluorinative Alkylboration of Alkenes Under Dual Photoredox and Copper Catalysis

Full Text

HTML

PDF (91 kb)
0381
Doubly Enantioconvergent Construction of Vicinal Stereocenters by Iridium-Catalyzed Allylic Alkylation

Full Text

HTML

PDF (89 kb)
0382
Strained-Alkene-Mediated Divergent Synthesis of Fluorenones and Fused Dibenzocycloheptenones

Full Text

HTML

PDF (90 kb)
0383
Synthesis of Seven-Membered Lactones via Palladium-Catalyzed Ring-Opening [5+2] Annulation

Full Text

HTML

PDF (77 kb)
0384
Synthesis of Ynones and γ-Butenolides with In Situ-Formed CO from a Palladium Difluorocarbene Complex

Full Text

HTML

PDF (137 kb)
0385
Palladium-Catalyzed Asymmetric α-Arylation of Azlactones and 5H-Oxazol-4-ones

Full Text

HTML

PDF (99 kb)
0386
Copper-Catalyzed Synthesis of Enantioenriched β-Boryl-α-Aryl Carboxylic Acids

Full Text

HTML

PDF (93 kb)
0387
Ring Expansion of Indenes Using α-Iodonium Diazo Compounds as Functionalized Carbyne Precursors

Full Text

HTML

PDF (87 kb)
0388
Carboxylic Phosphoric Anhydrides: New Partners for Pd-Catalyzed Decarbonylative Sonogashira

Full Text

HTML

PDF (70 kb)
0389
Asymmetric Synthesis of γ-Alkoxy-α,β-Imides via Gold Catalysis

Full Text

HTML

PDF (86 kb)
0390
Aerobic Asymmetric Oxidative Allylation of β-Keto Esters Enabled by Amine–Pd Catalysis

Full Text

HTML

PDF (85 kb)
0391
The Takai–Oshima–Lombardo Methylenation of Carbonyl Compounds FREE ACCESS

Full Text

HTML

PDF (129 kb)
0392
Stereodivergent Homocoupling of Benzoxazolyl Acetates by Dual Nickel and Copper Electrocatalysis

Full Text

HTML

PDF (79 kb)
Polymer-Supported Synthesis
z0393
All PDFs of this category

Full Text

PDF (853 kb)
0393
Asymmetric Hydrogenation of Acrylates by COF with Chiral Frustrated Lewis Pairs FREE ACCESS

Full Text

HTML

PDF (124 kb)
0394
Photocatalytic Synthesis of (2-Tosylvinyl) Sulfides and Selenides by Graphitic Carbon Nitride

Full Text

HTML

PDF (78 kb)
0395
“Activated Borane” – Porous Borane-Organic Clusters as Lewis Acid Catalysts

Full Text

HTML

PDF (138 kb)
0396
Semihydrogenation of Alkynes with a Pd-Carbide Composite Encapsulated in an MFI Zeolite

Full Text

HTML

PDF (269 kb)
0397
The Suzuki–Miyaura Coupling Catalyzed by Palladium on a Phenanthroline-Based COP

Full Text

HTML

PDF (95 kb)
0398
Photocatalytic Oxidation of Benzylic C(sp³)–H Bonds, Thioanisoles, and Benzylamines

Full Text

HTML

PDF (86 kb)
0399
Photocatalytic Hydrogenolysis of Lignin β-O-4 Models by a Ni-Containing Polyoxometalate/CdS QDs System

Full Text

HTML

PDF (95 kb)
0400
Hydrogenation of Furfurals by Pd-Based Bimetallic Alloys in Aqueous Micelles

Full Text

HTML

PDF (69 kb)
0401
Knoevenagel Reaction and Synthesis of 2,3-Dihydroquinazolin-4(1H)-ones Using Urea-Rich POP

Full Text

HTML

PDF (96 kb)
0402
Light-Driven Hydrogenation of Nitroarenes by Iron Catalysts Supported on TiO₂

Full Text

HTML

PDF (70 kb)
0403
Reductive N-Formylation of Amines with CO₂ Using an NHC-Based Porous Organic Polymer

Full Text

HTML

PDF (394 kb)
0404
Decarbonylation of Thioesters Catalyzed by CeO₂- or Hydroxyapatite-Supported Ni, Pd, or Rh Nanoparticles

Full Text

HTML

PDF (84 kb)
Organo- and Biocatalysis
z0405
All PDFs of this category

Full Text

PDF (1127 kb)
0405
Organo- and Biocatalysis in One-Pot Chemoenzymatic Oxidation and Michael Reaction Cascade

Full Text

HTML

PDF (169 kb)
0406
Stereo- and Regioselective Hydroxylation of Cyclobutyl- and Bicyclo[1.1.1]pentylamines via Biocatalysis

Full Text

HTML

PDF (104 kb)
0407
Catalytic Enantioselective Wagner–Meerwein Rearrangement of Alkenyl Cycloalkanes FREE ACCESS

Full Text

HTML

PDF (123 kb)
0408
Trialkylphosphines-Catalyzed C–F Activation of Highly Fluorinated Arenes and Heteroarenes

Full Text

HTML

PDF (70 kb)
0409
Dearomative [2π+2σ] Photocycloaddition of Phenols and Bicyclobutanes

Full Text

HTML

PDF (98 kb)
0410
NaCl-Mediated Catalytic Enantioselective α-Chlorination of Ketones

Full Text

HTML

PDF (92 kb)
0411
Atroposelective Synthesis of Axially Chiral 1,3-Dienes via C(sp²)–H Functionalization

Full Text

HTML

PDF (735 kb)
0412
Photocatalyst-Free Catalytic Single-Electron Reduction by 1H-1,2,3-Triazol-5-ylidenes

Full Text

HTML

PDF (81 kb)
0413
Radical (Hydro)Sulfonylation of Alkenes Promoted by Formation of an Electron Donor–Acceptor Complex

Full Text

HTML

PDF (110 kb)
Innovative Drug Discovery and Development
z0415
All PDFs of this category

Full Text

PDF (1015 kb)
0415
Arenophile Cycloaddition-Mediated Dearomative Pyridine Oxidation FREE ACCESS

Full Text

HTML

PDF (122 kb)
0416
Photoactivated Gene Therapy: Targeted Retinal Pathologies with Caged Ethinylestradiol

Full Text

HTML

PDF (73 kb)
0417
A Twist-to-Open Mechanism for the VGIC Subtype KCNQ2 is Revealed Using a Novel Small Molecule Activator

Full Text

HTML

PDF (213 kb)
0418
Simple Synthesis of Indazoles

Full Text

HTML

PDF (103 kb)
0419
Novel [2+2+1] Reaction with Triplet Nitrene

Full Text

HTML

PDF (506 kb)
0420
Straightforward Access to Azepanes from Nitroarenes

Full Text

HTML

PDF (70 kb)
0421
Discovery of Indazole-Based Selective IRAK4 Inhibitors

Full Text

HTML

PDF (77 kb)
0422
Selectfluor Electrochemistry Enables Site-Selective Synthesis of Versatile Aryl DABCOnium Salts

Full Text

HTML

PDF (93 kb)
0423
Decagram-Scale Synthesis of an Anti-Cancer Drug Candidate

Full Text

HTML

PDF (82 kb)
0424
Convenient Access to N-Difluoromethyl Amides, Urea, Carbamate and Thiocarbamate Derivatives

Full Text

HTML

PDF (79 kb)
0425
The First Total Synthesis of Camphor and the Industrial Standard FREE ACCESS

Full Text

HTML

PDF (121 kb)
0426
Late-Stage TBADT-Catalyzed Oxidation Guides Structural Modification to Improve Half-Life

Full Text

HTML

PDF (68 kb)
Peptide Chemistry
z0427
All PDFs of this category

Full Text

PDF (452 kb)
0427
Quinoline-8-carboxamides Synthesis via Aldehyde C–H Bond Activation Using Palladium Catalyst

Full Text

HTML

PDF (72 kb)
0428
Organocatalytic Stereoselective Synthesis of β-Hydroxy-α-Amino Acids

Full Text

HTML

PDF (93 kb)
0429
Recyclable Bicyclic Benziodazolone-Mediated Peptide Coupling Reaction FREE ACCESS

Full Text

HTML

PDF (114 kb)
0430
B(C₆F₅)₃-Catalyzed Diastereoselective Synthesis of Carbocyclic β-Amino Acid (CBAA) Derivatives

Full Text

HTML

PDF (98 kb)
0431
Mn-Catalyzed Visible-Light-Mediated Synthesis of Amide via Aminocarbonylation

Full Text

HTML

PDF (68 kb)
0432
Lewis Base-Catalyzed β-Amino Acids Synthesis from Trifluoro and Trichloro Acetamide and MBH Carbonates

Full Text

HTML

PDF (86 kb)
0433
Synthesis of Peptides via Nicotinate-Directed Transamidations by Zinc Catalysis

Full Text

HTML

PDF (76 kb)
0434
Synthesis of Chiral α-Vinylic Amino Acids via Enantioselective Aza-Nozaki–Hiyama–Kishi Reaction

Full Text

HTML

PDF (93 kb)
0435
α-Functionalization of Glycine to Access Functionalized Amino Acids and Peptides

Full Text

HTML

PDF (81 kb)
0436
Synthesis of Cross-Linked Pseudopeptides Using Pd-Catalyzed Carbonylative Coupling

Full Text

HTML

PDF (85 kb)
0437
Synthesis of Difluoroalanine (dfa) and Their Applications in Peptide Synthesis

Full Text

HTML

PDF (71 kb)
0438
Ru/Cu-Catalyzed Modification of Diphenyl Ketoimine Amino Acids and Peptides

Full Text

HTML

PDF (82 kb)
0439
Two Step Synthesis of β^2,2-Amino Acids from Alkylidenemalononitriles and Cbz-Gly

Full Text

HTML

PDF (83 kb)
0440
Palladium-Catalyzed C(sp²)–H Activation for Site-Selective Functionalization of Peptides

Full Text

HTML

PDF (99 kb)
0441
CDMT-Mediated Peptide Synthesis FREE ACCESS

Full Text

HTML

PDF (128 kb)
Flow Chemistry
z0443
All PDFs of this category

Full Text

PDF (621 kb)
0443
Asymmetric Rh-Catalyzed Reductive Enyne Cyclization Using a Continuous-Flow Setup

Full Text

HTML

PDF (71 kb)
0444
Development and Exploitation of a New Flow Reactor for Electrophotocatalysis (EPC)

Full Text

HTML

PDF (515 kb)
0445
Flow Chemistry Enables Safe, Kilogram-Scale Synthesis of 2-Hydroxypyridine-N-Oxide (HOPO)

Full Text

HTML

PDF (128 kb)
Most Read
Archive
Articles by Category
Free Sample Issue

Journal

More About This Journal
Synfacts Videos
Editorial Board
Editorial Office
Brochure

Authors

Instructions for Authors

Subscription

Subscription Information & Contacts
Institutional Licensing

Nobel Prize 2016

Instructions for Authors

Journals
Book Series
Login
Help
Portal
Return to Classic Website

German English

Thieme E-Books & E-Journals is a service of Georg Thieme Verlag and Thieme Medical Publishers, Inc.
© Georg Thieme Verlag KG

Imprint | Privacy policy statement

Your Current IP Address: 13.58.244.184