Synfacts

Issue 04 · April 2006

Issue
Synthesis of Natural Products and Potential Drugs
0299
Chen, K. X.; Njoroge, F. G.; Vibulbhan, B.; Prongay, A.; Pichardo, J.; Madison, V.; Buevich, A.; Chan, T.-M.: Synthesis of a Potent Hepatitis C Virus Serine Protease Inhibitor

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0300
Li, P.; Evans, C. D.; Joullié, M. M.: Synthesis of Ustiltoxin D

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0301
Iida, T.; Satoh, H.; Maeda, K.; Yamamoto, Y.; Asakawa, K.; Sawada, N.; Wada, T.; Kadowski, C.; Itoh, T.; Mase, T.; Weissman, S. A.; Tschaen, D.; Krska, S.; Volante, R. P.: Synthesis of a Neuropeptide Y Antagonist

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0302
Zeng, Y.; Aubé, J.: Synthesis of (±)-Stenine

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0303
Wardrop, D. J.; Bowen, E. G.: Synthesis of (+)-Lactacystin

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0304
Waters, S. P.; Tian, Y.; Li, Y.-M.; Danishefsky, S. J.: Synthesis of (-)-Scabronine G

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0305
Alibés, R.; Bayón, P.; de March, P.; Figueredo, M.; Font, J.; García-García, E.; González-Gálvez, D.: Synthesis of (-)-Norsecurinine

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0306
Sato, K.; Asao, N.; Yamamoto, Y.: Synthesis of (+)-Ochromycinone and(+)-Rubiginone B₂

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0307
Baran, P. S.; Richter, J. M.: Syntheses of Welwitindolinone A and Fischerindoles I

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0308
Hogan, P. C.; Corey, E. J.: Synthesis of a β-Lactam Proteasome Inhibitor

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0309
Wu, L.; Hartwig, J. F.: Synthesis of (±)-Verapamil

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0310
Bowie, A. J.; Hughes, C. C.; Trauner, D.: Synthesis of (±)-Rhazinilam

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0311
Yamashita, T.; Kawai, N.; Tokuyama, H.; Fukuyama, T.: Synthesis of (-)-Eudistomin C

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0312
Wrona, I. E.; Gabarda, A. E.; Evano, G.; Panek, J. S.: Synthesis of Reblastatin

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0313
Schnermann, M. J.; Boger, D. L.: Synthesis of Piericidins A1 and B1

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Synthesis of Heterocycles
0315
Chowdhury, C.; Mandal, S. B.; Achari, B.: Synthesis of Triazoles (I): Sequential Sonogashira Coupling and [2+3] Cycloaddition

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0316
Gracias, V.; Darczak, D.; Gasiecki, A. F.; Djuric, S. W.: Synthesis of Triazoles (II): van Leusen Imidazole Synthesis-Intramolecular [2+3] Cycloaddition

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0317
Yanai, H.; Taguchi, T.: Synthesis of Triazoles (III): Azidation of Dialkoxyacetylenes-Intramolecular [2+3] Cycloaddition

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0318
Rossi, E.; Abbiati, G.; Canevari, V.; Celentano, G.; Magri, E.: Synthesis of 2-Substituted Indoles by Cross-Coupling Reactions

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0319
Kuninobu, Y.; Tokunaga, Y.; Kawata, A.; Takai, K.: Synthesis of Phthalimidines via C-H Bond Activation

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0320
Linnepe, P.; Schmidt, A. M.; Eilbracht, P.: Synthesis of Indoles by a Combined Hydroformylation-Fischer Indolization Route

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0321
Handy, S. T.; Zhang, Y.: Predicting Regioselectivity in Cross-Coupling of Polyhaloheteroaromatics

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0322
Young, D. W.; Comins, D. L.: Synthesis of Dihydropyridones Involving Directed ortho-Metallation

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0323
Moonen, K.; Stevens, C. V.: Synthesis of Phosphono-β-Lactams

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0324
Tanaka, S.; Yasuda, M.; Baba, A.: Synthesis of Substituted Quinolines under Aerobic Conditions

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0325
Deng, X.; Mani, N. S.: Sonogashira-Mediated Synthesis of 4-Aryl-5-Pyrimidinylimidazoles

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0326
Wardrop, D. J.; Burge, M. S.: Stereocontrolled Synthesis of 4-6-Ring Lactams

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0327
Kuninobu, Y.; Nishimura, S.; Takai, K.: Synthesis of 4H-Pyrido[1,2-a]pyrimidin-4-ones

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0328
Mkhalid, I. A. I.; Coventry, D. N.; Albesa-Jove, D.; Batsanov, A. S.; Howard, J. A. K.; Perutz, R. N.; Marder, T. B.: Synthesis of Pyridyl and Pyridazyl Boropinacolates by Ir-Catalyzed C-H activation

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Synthesis of Materials and Unnatural Products
0329
Spencer, H. J.; Skabara, P. J.; Giles, M.; McCulloch, I.; Coles, S. J.; Hursthouse, M. B.: PEDOT vs. PEDTT: Subtle Variations, Large Consequences

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0330
Semetey, V.; Moustakas, D.; Whitesides, G. M.: Expeditive Synthesis of Rigid-Rod Oligopiperidines

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0331
Jin, L. Y.; Bae, J.; Ryu, J.-H.; Lee, M.: Cross-Linking Through the Core of a Mesogen

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0332
Nomoto, A.; Sonoda, M.; Yamaguchi, Y.; Ichikawa, T.; Hirose, K.; Tobe, Y.: An Abnormally Unstable Hexagonal Macrocycle

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0333
Guo, X.; Small, J. P.; Klare, J. E.; Wang, Y.; Purewal, M. S.; Tam, I. W.; Hong, B. H.; Caldwell, R.; Huang, L.; O’Brien, S.; Yan, J.; Breslow, R.; Wind, S. J.; Hone, J.; Kim, P.; Nuckolls, C.: Molecular Electronic Junctions with Nanotubes

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0334
Miao, S.; Bangcuyo, C. G.; Smith, M. D.; Bunz, U. H. F.: Derivatives of Octaethynylphenazine and Hexaethynylquinoxaline

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0335
Knapton, D.; Rowan, S. J.; Weder, C.: Metal-Ligand Binding Provides Route to High Molecular Weight Polymers

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0336
Itoh, T.; Nakata, Y.; Hirai, K.; Tomioka, H.: An Unusually Long-Lived Triplet Carbene

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0337
Koivisto, B. D.; Ichimura, A. S.; McDonald, R.; Lemaire, M. T.; Thompson, L. K.; Hicks, R. G.: Intramolecular π-Dimerization in a Diradical

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0338
Chen, R.-F.; Fan, Q.-L.; Zheng, C.; Huang, W.: Efficient Preparation of Polymerizable Heterofluorene Derivatives

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0339
Li, J.; Li, Y.; Liu, Y.; Wang, G.: Amino Acid Ester and Carbon Disulfide C₆₀ Functionalization

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0340
Leriche, P.; Blanchard, P.; Frère, P.; Levillain, E.; Mabon, G.; Roncali, J.: Ring-Closing Metathesis Approach to 3,4-Vinylenedioxythiophenes

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0341
Inokuma, Y.; Kwon, J. H.; Ahn, T. K.; Yoo, M.-C.; Kim, D.; Osuka, A.: Boron-Templated Synthesis of Subporphyrins

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Metal-Catalyzed Asymmetric Synthesis and Stereoselective Reactions
0343
Sanada, T.; Kato, T.; Mitani, M.; Mori, A.: Rhodium-Catalyzed Hydrosilylation of Internal Alkynes

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0344
Zhang, A.; RajanBabu, T. V.: Hydrovinylation of 1,3-Dienes

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0345
Yin, J.; Huffman, M. A.; Conrad, K. M.; Armstrong III, J. D.: Diastereoselective Catalytic MPV Reduction

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0346
Emmerson, D. P. G.; Hems, W. P.; Davis, B. G.: Carbohydrate-Derived Ligands for Asymmetric Alkynylation

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0347
Sieber, J. D.; Morken, J. P.: Sequential Pd-Catalyzed Asymmetric Allene Diboration/α-Aminoallylation

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0348
Bandini, M.; Melloni, A.; Piccinelli, F.; Sinisi, R.; Tommasi, S.; Umani-Ronchi, A.: Tetrahydro-β-Carbolines and Via Pd-Catalyzed Intramolecular Allylic Alkylation

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0349
Sasaki, M.; Higashi, M.; Masu, H.; Yamaguchi, K.; Takeda, K.: Asymmetric [2,3]-Wittig Rearrangement via Chirality Transfer

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0350
Liu, W.; You, F.; Mocella, C. J.; Harman, W. D.: Dihapto-Coordination of the Diene to Promote Sluggish Diels-Alder Reactions

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0351
Tsukamoto, H.; Ueno, T.; Kondo, Y.: trans-Alkylative Cyclization of Alkynals and Alkynones

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0352
Hamada, T.; Manabe, K.; Kobayashi, S.: Asymmetric Mannich-Type Reaction in Aqueous Media

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0353
Schultz, M. J.; Sigman, M. S.: Aerobic Dialkoxylation of Styrenes: A Profound Influence of an o-Phenol

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0354
Deschamp, J.; Chuzel, O.; Hannedouche, J.; Riant, O.: Copper-Catalyzed Asymmetric Domino Reductive Aldol Reactions

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0355
Xie, M.; Wang, J.; Gu, X.; Sun, Y.; Wang, S.: Three-Component Tandem Reaction to Synthesize Tetrasubstituted Olefins

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0356
Yamazaki, S.; Iwata, Y.: Cu(II)-Catalyzed Enantioselective Friedel-Crafts/Michael Addition of Indoles

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0357
Jia, Y.; Zhu, S.; Yang, Y.; Zhou, Z.: Friedel-Crafts Alkylations of Indoles with Nitroalkenes

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0358
Berkessel, A.; Ertürk, E.; Laporte, C.: Cr(III)-Porphyrin-Catalyzed Enantioselective Hetero-Diels-Alder Reactions

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0359
Kong, J.; Ngai, M.; Krische, M. J.: Enantioselective Direct Reductive Coupling of Conjugated Alkynes and α-Ketoesters

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0360
Dervisi, A.; Carcedo, C.; Ooi, L.-I.: Ambient Pressure Asymmetric Imine Hydrogenation

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0361
Davies, H. M. L.; Manning, J. R.: Rh-Catalyzed Enantioselective Synthesis of 4-Substituted Heterocycles

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0362
Reetz, M. T.; Li, X.: Asymmetric Transfer Hydrogenation of Alkyl/Aryl and Dialkyl Ketones

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0363
Nadeau, C.; Gosselin, F.; O’Shea, P. D.; Davies, I. W.; Volante, R. P.: Enantioselective Synthesis of (S)-γ-Fluoroleucine Ethyl Ester

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0364
Bell, S.; Wüstenberg, B.; Kaiser, S.; Menges, F.; Netscher, T.; Pfaltz, A.: Asymmetric Hydrogenation of Unfunctionalized Alkyl-Substituted Olefins

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0365
Itagaki, M.; Yamamoto, Y.: Asymmetric Cyclopropanation of Styrene with a Cu(I)-Cyclopropyl Bisoxazoline Ligand

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0366
Palomo, C.; Oiarbide, M.; Halder, R.; Laso, A.; López, R.: Enantioselective Aza-Henry Reactions Assisted by Zn(II) and N-Methylephedrine

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0367
Concellon, J. M.; Suarez, J. R.; Solar, V. del: Synthesis of Enantiopure Allyl Amines Using Reductive Alkylation

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0368
Chen, F. X.; Kina, A.; Hayashi, T.: High Performance Diene-Rhodium Catalyst for Conjugate Addition of Arylboroxines

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0369
Ros, A.; Magriz, A.; Dietrich, H.; Fernández, R.; Alvarez, E.; Lassaletta, J. M.: Synthesis of Vicinal Halohydrins via Dynamic Kinetic Resolution

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Metal-Mediated Synthesis
0371
Bedford, R. B.; Betham, M.; Bruce, D. W.; Danopoulos, A. A.; Frost, R. M.; M Hird: Iron-Ligand Catalysts for Aryl-Alkyl Cross-Coupling Reactions

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0372
López, F.; van Zijl, A. W.; Minnaard, A. L.; Feringa, B. L.: Cu-Catalyzed Enantioselective Allylic Substitution with Grignard Reagents

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0373
Walter, I. A. S.: One-Pot Negishi Coupling of Alkyl Bromides with Hetaryl Halides

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0374
Takahashi, H.; Hossain, K. M.; Nishihara, Y.; Shibata, T.; Takagi, K.: Rh-Catalyzed Coupling of Arylzinc Halides with (Iodomethyl)trimethylsilane

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0375
Kabalka, G. W.; Al-Masum, M.: Microwave-Enhanced Coupling of Alkenyltrifluoroborates with Allyl Acetates

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0376
Bica, K.; Gärtner, P.: Iron-Containing Ionic Liquid as Catalyst for Cross-Coupling of Grignard Reagents with Alkyl Halides

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0377
Denmark, S. E.; Butler, C. R.: Coupling of Aryl Bromides with Tetravinyltetrasiloxane

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0378
Fuchibe, K.; Akiyama, T.: Niobium-Mediated Double Activation of C-F/C-H Bonds: Fluorene Synthesis

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0379
Quntar, A. A. Aziz; Srebnik, M.: Direct Cyclopropanation of 1-Alkynylphosphonates

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0380
Yoshino, H.; Toda, N.; Kobata, M.; Ukai, K.; Oshima, K.; Utimoto, K.; Matsubara, S.: Sequential Cross-Coupling of gem-Dizincioalkanes

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0381
Tanino, K.; Arakawa, K.; Satoh, M.; Iwata, Y.; Miyashita, M.: (Z)-Vinylcopper Species from 1,1-Dibromoalkenes and its Reactions

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0382
Kudo, N.; Perseghini, M.; Fu, G. C.: A Versatile Method for Suzuki Cross-Coupling of Nitrogen Heterocycles

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0383
Kuwano, R.; Yokogi, M.: Cross-Coupling of Benzylic Acetates with Arylboronic Acids

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0384
Basheer, C.; Vetrichelvan, M.; Suresh, V.; Lee, H. K.: The Oxidation of Cyclohexene with an Ionic-liquid in a Microreactor

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Organo- and Biocatalysis
0385
Gröger, H.; May, O.; Hüsken, H.; Georgeon, S.; Drauz, K.; Landfester, K.: Enzyme Reactions in Miniemulsions

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0386
Malkov, A. V.; Liddon, A. J. P. Stewart; Ramírez-López, P.; Bendová, L.; Haigh, D.; KoČovsk, P.: Organocatalytic Asymmetric Hydrosilylation of Ketones and Ketimines

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0387
Bekele, T.; Shah, M. H.; Wolfer, J.; Abraham, C. J.; Weatherwax, A.; Lectka, T.: Enantioselective [4+2] Cycloadditions of Ketenes with o-Quinones

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0388
Rodriguez, B.; Bolm, C.: Microwave-Assisted Proline-Catalyzed Direct Asymmetric Mannich Reaction

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0389
Ooi, T.; Uematsu, Y.; Maruoka, K.: Organocatalytic Asymmetric Strecker Reaction

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0390
Menche, D.; Hassfeld, J.; Li, J.; Menche, G.; Ritter, A.; Rudolph, S.: Thiourea-Catalyzed Reductive Amination of Ketones

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0391
Wang, Z.; Ye, X.; Wei, S.; Wu, P.; Zhang, A.; Sun, J.: Ketimine Reduction Employing a Pipecolic Acid Derived Organocatalyst

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0392
Terada, M.; Ube, H.; Yaguchi, Y.: Axially Chiral Guanidine-Catalyzed Asymmetric Addition of Malonates to Nitroalkenes

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0393
Paizs, C.; Katona, A.; Rétey, J.: One-Pot Synthesis of l-Arylalanines from Arylaldehydes

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0394
Tamura, Y.; Itoh, J.; Morita, H.; Fuchibe, K.; Akiyama, T.: Enantioselective Aza-Diels-Alder Reaction Catalyzed by a Chiral Brønsted Acid

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0395
Tillman, A. L.; Ye, J.; Dixon, D. J.: Bifunctional Cinchonine-Catalyzed Asymmetric Mannich Reaction

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Polymer-Supported Synthesis
0397
Solodenko, W.; Bröker, P.; Messinger, J.; Schön, U.; Kirschning, A.: Synthesis of Unprotected Guanidines Using Polymer-Bound Pyrazole Derivatives

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0398
Kato, D.; Verhelst, S. H. L.; Sexton, K. B.; Bogyo, M.: Solid-Phase Synthesis of Diverse Azapeptides

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0399
Doherty, S.; Knight, J. G.; Betham, M.: Polymer-Bound Palladium Complexes of 2-Pyridyldiphenylphosphine

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0400
Pedatella, S.; Guaragna, A.; D’Alonzo, D.; Nisco, M. D.; Palumbo, G.: Efficient Acetonation of Sugar Deriavtives

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0401
Werner, H.; Herrerías, C. I.; Glos, M.; Gissibl, A.; Fraile, J. M.; Pérez, I.; Mayoral, J. A.; Reiser, O.: Merrifield Resin Supported Copper Catalyst for Asymmetric Cyclopropanation

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0402
Turner, K. L.; Baker, T. M.; Islam, S.; Procter, D. J.; Stefaniak, M.: Solid-Phase Approach to Tetrahydroquinolones

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0403
Back, T. G.; Zhai, H.: Polymer-Supported Acetylenic Sulfones

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0404
Wang, Y.; Sauer, D. R.; Djuric, S. W.: The Synthesis of 1,3,4-Oxadiazoles by Using PS-PPh₃

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0405
Kashiwagi, Y.; Ikezoe, H.; Ono, T.: Oxidation of Alcohols with Nitroxyl Radical Resins under Two-Phase Conditions

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0406
Ladziata, U.; Willging, J.; Zhdankin, V. V.: Polymeric N-(2-Iodyl-phenyl)-acylamide Reagent for Oxidation of Alcohols

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0407
Fuchter, M. J.; Hoffman, B. M.; Barrett, A. G. M.: Photooxygenation Using ROM Polymer Sphere-Supported seco-Porphyrazines

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0408
He, H. S.; Zhang, C.; Ng, C. K.-W.; Toy, P. H.: Polymer-Supported Triphenylarsines as Ligands and a Catalyst

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0409
Lysén, M.; Köhler, K.: Pd/C-Catalyzed Suzuki-Miyaura Cross-Coupling of Aryl Chlorides in Water

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0410
Thomas, G. L.; Böhner, C.; Ladlow, M.; Spring, D. R.: Synthesis and Utilization of Functionalized Polystyrene Resins

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