DOI: 10.1055/s-00000131

Synfacts

Issue 01 · Volume 12 · January 2016 DOI: 10.1055/s-005-30635

Synform

A1
Zanda, Matteo: SYNFORM ISSUE 2016/01

Synthesis of Natural Products and Potential Drugs

z1
All PDFs of this category
0001
Synthesis of ent-Ketorfanol
0002
Synthesis of (+)-Crotophorbolone
0003
Synthesis of Portentol
0004
Synthesis of Bosutinib
0005
Total Synthesis of (–)-Isoschizogamine
0006
Total Syntheses of (±)-Crotobarin and (±)-Crotogoudin
0007
Synthesis of KAE609 by Catalytic Asymmetric Alkynylation
0008
Synthesis of (+)-MPC1001B
0009
Synthesis of Epoxyeujindole A
0010
Total Synthesis of (–)-Jiadifenolide
0011
Synthesis of Filorexant
0012
Synthesis of NS5B Polymerase Inhibitor GSK852A

Synthesis of Heterocycles

z13
All PDFs of this category
0013
Synthesis of Benzo[1,3]oxathiins from Benzobisthietes
0014
Enantioselective Propargylation of Cyclic N-Sulfonylketimines
0015
Palladium-Catalyzed Synthesis of Ring-Fused Benzosultams and Benzosultones
0016
Oxidative Cross-Dehydrogenative Coupling of N-Heterocycles with Aldehydes
0017
Rhodium-Catalyzed C-7 Functionalization of Indoles
0018
Three-Component Synthesis of Dihydropyridopyrimidines
0019
Synthesis of Substituted Isoquinolines from Aryl 1,2,3-Triazoles
0020
Cobalt(III)-Catalyzed Synthesis of Isoquino-lines from O-Acyl Oximes and Alkynes
0021
Ruthenium-Catalyzed Synthesis of Hydroxybutenolides
0022
Convenient Access to Sulfinyl Derivatives of Heterocycles
0023
Palladium-Catalyzed Enantioselective Synthesis of Benzoxazinoindoles
0024
Silver-Catalyzed Heteroannulation Route to Benzofuro- and Benzothienopyridines
0025
Substituted 1,2,3-Triazoles by Copper-Catalyzed Cycloaddition/N-Alkylation
0026
Enantioselective Synthesis of 1,2-Dihydro-pyridines by Formal [4+2] Cycloaddition
0027
Synthesis of Oxazoles from Methyl Ketones and Amino Acids

Synthesis of Materials and Unnatural Products

z29
All PDFs of this category
0029
Double Spiros
0030
Te/B Heterocycles
0031
Selective Functionalization of DTT
0032
Intramolecular Friedel–Crafts Acylation Reaction Promoted by HFIP
0033
Solution-Stable Cages Connected By B–N Bonds
0034
Sulfur Makes a Difference
0035
Putting Nitrogen Atoms in Coronene
0036
Photocyclodehydrogenation Produces Polycyclic Aromatic Hydrocarbons
0037
Iterative Exponential Growth of Stereo- and Sequence-Controlled Polymers
0038
An n-Type Semiconducting Near-Infrared Dye
0039
Fixed It! 9-Phenylanthracene Goes Plane
0040
Multicomponent Synthesis of Polythioamides

Metal-Catalyzed Asymmetric Synthesis and Stereoselective Reactions

z41
All PDFs of this category
0041
Asymmetric Rhodium-Catalyzed C–C Activation of Cyclobutanones
0042
Enantioselective Rhodium-Catalyzed Addition of Boronic Acids to Ketimines
0043
Stereodivergent Iridium- and Amine-Catalyzed α-Allylation of Aldehydes
0044
Rhodium(I)-Catalyzed Asymmetric Synthesis of Piperidines
0045
Asymmetric Cycloisomerizations Promoted by Cyclopentadienyl Iridium(III)
0046
Minimization of Aryloxy Elimination in Asymmetric Hydrogenation
0047
Palladium-Catalyzed Enantioselective 1,2-Difunctionalization of 1,3-Dienes
0048
Diastereoselective Synthesis of Aldol Products by Dual Catalysis
0049
Rhodium-Catalyzed Asymmetric Hydro-acylation of ortho-Allylbenzaldehydes
0050
Asymmetric Allylboration by Combining Copper and Palladium Catalysis
0051
Rhodium-Catalyzed Asymmetric Hydrogenation of α-Dehydroamino Ketones
0052
Ruthenium-Catalyzed Asymmetric Synthesis of γ-Secondary Amino Alcohols
0053
Asymmetric Hydrogenation of Alkenes by an Iridium-P/S Complex as Catalyst
0054
Enantioselective Inverse Electron Demand Aza-Diels–Alder Reaction
0055
Remarkable Substituent Effects in Gold-Catalyzed Cycloadditions
0056
Palladium-Catalyzed Dearomative Indole Bisfunctionalization
0057
Catalytic Asymmetric C–C Bond Formation by 1,4-Addition of Alkyl Nitriles
0058
Rhodium-Catalyzed Asymmetric Hydrogenation of 2-Pyridine Ketones
0059
Asymmetric Copper-Catalyzed Addition of ZnEt2 to Pentafulvenes
0060
Gold-Catalyzed Asymmetric Synthesis of Six-Membered Rings
0061
Tandem Asymmetric Hydrogen Transfer Oxidation/Aldol Condensation
0062
Palladium-Catalyzed Enantioselective Allylic Alkylation of Cyclopentanones
0063
Enantioselective Copper-Catalyzed Alkynyl-ation of Quinolinium Salts Generated In Situ
0064
Asymmetric Synthesis of γ-Lactones by Iridium Catalysis
0065
Vanadium-Catalyzed Asymmetric Cascade Reaction
0066
Diastereoselective Palladium-Catalyzed [5+2] Annulation Forming Dibenzo[b,d]azepines
0067
Lycorane Analogues by Palladium-Catalyzed Heck–Heck Cascade

Metal-Mediated Synthesis

z69
All PDFs of this category
0069
Organocopper-Promoted Cyclization of Conjugated Diene-ynes
0070
Asymmetric Arylation of Allylic Halides with Boronic Acids
0071
Diastereoselective α-Alkylation of α-Epoxy N-Sulfonyl Hydrazones
0072
Regioselective Ring Opening of Diisopropylsilylenes
0073
Silver Carbonate-Promoted ipso-Nitration of Carboxylic Acids
0074
Carbonylative Suzuki Coupling of Aryl Halides with Arylboronic Esters
0075
Zinc-Mediated Carboxylation of 2-Alkynyl Bromides
0076
Dihydroboration of Organonitriles
0077
Copper-Promoted Cycloaddition
0078
Copper-Catalyzed Reaction of Trifluoromethylketones with Aldehydes
0079
Copper-Catalyzed Oxyboration of Terminal Unactivated Alkenes
0080
Reverse Diastereocontrol in the Conjugate Addition of Cuprates
0081
Water Opens the Door to Organolithiums and Grignard Reagents
0082
Asymmetric Reduction of Ketimines by N-Heterocyclic Carbene Boranes
0083
Copper-Catalyzed Borylation/ortho-Cyanation Cascade

Organo- and Biocatalysis

z85
All PDFs of this category
0085
Highly Diastereoselective Triflimide-Catalyzed Mukaiyama Aldol Reaction
0086
Organocatalytic Asymmetric Passerini Reaction
0087
Asymmetric Dearomatizing Michael Addition of β-Naphthols
0088
Organocatalytic Diels–Alder Reaction to Access Norcamphor Scaffolds
0089
Aminothiourea-Catalyzed Asymmetric Synthesis of Spiroketals
0090
Enantioselective Biocatalytic Dealkylation of N-Benzylisoquinolines
0091
Enantioselective Organocatalytic Trichloromethylation with Chloroform

Polymer-Supported Synthesis

z93
All PDFs of this category
0093
Asymmetric Aldol Reaction by Dipeptide Nanotubes
0094
Selective Oxidation of Hydroquinones with Silica Gel-Supported Cerium(IV)
0095
Copper/DNA G-Quadruplex-Catalyzed Diels–Alder Reaction
0096
Polystyrene-Supported Imidazolidine-4-one–Copper Complexes for the Henry Reaction
0097
Cyclization of Propargylic Alcohols with Carbon Dioxide by Using Silver Nanoparticles
0098
Silica-Supported Oligomeric Benzylic Phosphates as Alkylating Reagents
0099
A Star Polymer-Supported Palladium–N-Heterocyclic Carbene Precatalyst
0100
Aerobic Oxidative Coupling of Alcohols on a Cobalt Nanocomposite Catalyst
0101
Flow Cycloisomerization of Ugi Adducts with Supported Gold Nanoparticles
0102
Oxidative Esterification of Aldehydes on Reduced Graphene Oxide-Supported Co3O4
0103
Desulfurative C–C Coupling Reactions with a Wool–Palladium Acetate Complex
0104
Reduction of Nitroarenes Catalyzed by Water-Soluble Gold Nanoparticles
0105
Suzuki–Miyaura Reaction on Nanosheet-Supported Palladium Nanoparticles
0106
Aerobic Oxidation of Alcohol by Using a Supported Copper Complex
0107
Synthesis of Disulfides and Diselenides Catalyzed by a Metal–Organic Framework
0108
N-Substituted Anilines by Tandem Oxidation Catalyzed by Gold–Palladium/Alumina