Synfacts

Issue 01 · January 2023

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SYNFORM ISSUE 2023/01 FREE ACCESS

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Synthesis of Natural Products
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0001
Total Synthesis of (±)-Daphgraciline FREE ACCESS

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0002
Synthesis of (+)-Dysiherbols A and D

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0003
Synthesis of (–)-Gedunin

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0004
Total Synthesis of (+)-Gilbertine

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0005
Total Synthesis of (±)-Psammaplysin A

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0006
Synthesis and Structural Revision of (±)-6,11-Epoxyisodaucane

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0007
Total Synthesis of Pagodane FREE ACCESS

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Synthesis of Heterocycles
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0009
Synthesis and Biological Activity of Bicyclic Nitroimidazole Derivatives

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0010
Synthesis and Characterization of Spiro-Tetrahydrotetrazines as Energetic Materials

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0011
Preparation of 4-Iodo-1-tosylpyrazoles via Iodocyclization of N-Propargyl-N′-tosylhydrazines

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0012
Rh(I)-Catalyzed Synthesis of 3-Substituted Oxindoles

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0013
One-Pot Synthesis of N-Aryl Tetrahydroquinolines

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0014
Iron-Catalyzed Stereo-Convergent Cyclization with E/Z-Mixed Internal Olefines

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0015
A Grignard-Free 1,2-Arylation of Isatins

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0016
Nickel-Catalyzed Synthesis of chiral N-Heterocycles via C(sp³)–H Activation of Formamides

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0017
An Aza-Baeyer–Villiger Reaction for Nitrogen Insertion into Cyclobutanones

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0018
Decarboxylative Asymmetric Allylic Alkylation for the Synthesis of α‑Difunctionalized Cyclic Sulfones

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0019
Multicomponent Reaction for the Synthesis of Quinoxalin-2-Thiones and Quinoxalines

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0020
Catalyst-Free Synthesis of CF₃-Containing 2-Pyrazolines via [3+2] Cycloadditions

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0021
Pd-Catalyzed Suzuki Coupling of Nitroarenes and Heteroarylboronate Esters

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Synthesis of Materials and Unnatural Products
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0023
Cyclopropane-fused Dehydro[10]annulene FREE ACCESS

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0024
Fused Heteroaromatics via Double C–F Activation

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0025
Large Arylene Vinylene Polymers Stitched by Rhodium

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0026
Linear Ladder-Type S,N-Heteroacenes

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0027
4-Organoselenyl Quinolines

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0028
A Cubic Electron Catcher

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0029
Phosphaalkene Metathesis to Tetraaryl Olefins

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0030
Cyclopolymerization towards Bicyclic Polyacetylenes

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0031
[1,4]Diazocine with Application as Chiral Ligand

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0032
From Vinyl Azides to Phenanthridines

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0033
Twisted Armchair-Edged Graphene Nanoribbons

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0034
Metal-Free Benzylic C–O Cyclization

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Metals in Synthesis
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0035
Selective Cyanation of Benzylic C(sp³)–H Bonds Using Photoelectrochemical Asymmetric Catalysis FREE ACCESS

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0036
The Kochi–Salomon [2+2] Photocycloaddition of Amine-Containing Dienes under Aqueous Conditions

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0037
Palladium-Catalyzed Cross-Coupling of Aryl Halides with Carboxylic Acids by Photoinduced Reductive Elimination FREE ACCESS

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0038
Rh(II)-Catalyzed Arylation/Allylation of Diazo Esters

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0039
Nickel-Catalyzed Dicarbofunctionalization of Olefins

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0040
Directed Addition of Nitroalkanes Across Unactivated Olefins via Palladium(II) Catalysis

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0041
Shining Blue Light on the Palladium-Catalyzed Carbo-iodination of Alkenes Leads to a Radical Mechanism

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0042
Palladium(0)-Catalyzed Carbonylative Formation of Acyl-DMAP Salts from Organotriflates

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0043
Synthesis of Spirocyclic and Bis-Indolinones via Palladium-Catalyzed Carbonylation Reactions

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0044
Regio- and Enantioselective Alkylation of Pyridinium Ions in C2 or C4 Position

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0045
Dual Iron/Photoredox-Catalyzed 1,2-Arylchlorination of Vinylboronic Esters via In Situ Generated Aryl Radicals

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0046
Nickel-Catalyzed Enantioselective Hydrocarbo- and Dicarbofunctionalization of Alkenes

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0047
Z-Selective Olefin Metathesis by Combining Grubbs II with a Photoisomerization Catalyst

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0048
Enantioselective Three-Component 1,2-Oxyalkylation of Conjugated Dienes under Copper Catalysis

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0049
Palladium(0) α-Arylation of Enones Using Aryltriflates via a Morita–Baylis–Hillman Approach

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0050
Nucleophilic Ring Opening of Arylcyclopropanes under Photoredox Catalysis

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0051
Ni/Photoredox-Catalyzed Ring-Opening/Alkylation of Aziridines

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0052
Regiodivergent Disilylation of Arylacetylenes Using Cobalt Catalysis in a One-Pot, Two-Step Fashion

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0053
Photocatalytic Decarboxylative C–H Alkylation of Pyridines Under Oxidant-Free Conditions

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0054
Synthesis of Fluorinated Chromanes via Palladium-Based Dyotropic Rearrangement

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0055
Stereospecific Cross-Coupling of Cyclopropyl Zincates under Dinuclear Palladium(I) Catalysis

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0056
Enantioselecitve Allylation/Retro-Claisen Cascade

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0057
Bimetallic-Catalyzed Asymmetric C2-Selective C–H Alkylation of Pyridines with 1,3-Dienes

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0058
Modular Synthesis of Esters Using Unactivated Alkyl Chlorides, CO, Alcohols and Rhodium Catalysis

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0059
The Murai Reaction: ortho-Directed Ruthenium-Catalyzed C–H Alkylation of Aromatic Ketones FREE ACCESS

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0060
Regioselective N-Allylation of Azoles Using Dual Palladium(0)–Organoboron Catalysis and Allyl Alcohols

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0061
Intramolecular Nucleopalladation/Carbonylation of Alcohol-Tethered Alkenes FREE ACCESS

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Polymer-Supported Synthesis
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0063
Z-Selective Semi-Hydrogenation of Alkynes by a Cobalt-Melamine Catalyst Supported on SiO₂

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0064
Aerobic Oxidation of Sulfides by Zr-Based Porphyrin MOFs Using HOOC-TEMPO Under Red LED Irradiation

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0065
Photocatalytic Reductive Dimerization of Aryl Bromides Using Water as a Reductant

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0066
Fluorination of Acyl Chlorides Promoted by a Single-Atom Cobalt Catalyst FREE ACCESS

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0067
Zn-Catalyzed Aerobic Oxidation of Alcohols Under Solvent-Free and Blue LED Irradiation Conditions

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0068
Synthesis of a Covalent Organic Framework through a Sunlight Photocatalytic Reaction

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0069
α-Alkylation of Ketones with Alcohols Using a MgO-Codeposited Mn Catalyst Supported on Al₂O₃

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0070
Suzuki–Miyaura Coupling by Pd Polyaniline Complex Under Batch and Flow Conditions

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0071
Suzuki–Miyaura Coupling of Nitrogen Heteroarenes by Pd-Ag Nanoclusters Decorated with Microcellulose

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0072
Synthesis of β-Keto Sulfones Using g-C₃N₄ Under Blue LED Irradiation

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0073
Hydroboration of Arylacetylenes by Ultrathin Imide-Linked Metal–Organic Framework Nanosheets

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Organo- and Biocatalysis
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0075
Vitamin B₂-Catalyzed Coupling of Sulfides and Alkenes

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0076
Phenothiazine Photocatalyst Permits Copper-Free Bromoalkylation of Thianthrenium Salts

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0077
Visible Light-Mediated β-Lactam Synthesis from Acryl Amide Precursors FREE ACCESS

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0078
Bridged Tetrahydrobenzo[b]azepines/oxepines through Organocatalytic Aza-Piancatelli/Michael Reactions

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0079
Stereoselective Multicomponent Synthesis of Alkaloid-Like Frameworks by Inverse Hydride Shuttle Catalysis

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0080
Engineered Methyl Transferases Enable Regioselective N-Methylation of Unsaturated Heterocycles

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0081
Enzymatic Amination and Amidation of Unactivated Csp³–H Sites

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0082
Bifunctional Pyridoxal-Catalyzed Direct Enantioselective Synthesis of β-Aminoalcohols

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0083
Organocatalytic Asymmetric Synthesis of SynVesT-1 and [¹⁸F]-SynVesT-1

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0084
Catalytic Asymmetric Tautomerization of α-Hydroxy Ketones

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Innovative Drug Discovery and Development
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0085
Photoaffinity Lipid Probes Decipher Docosahexanoic Acid Target FREE ACCESS

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0086
The Power of Symmetry: Disorazole Z Analogues via a Double Stille Cross-Coupling

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0087
Novel Dioxane- and Morpholino Nucleotide Analogues with Improved Off-Target Profiles in siRNAs FREE ACCESS

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0088
Scalable Synthesis of a Fluorinated Bicyclic Pyrrolidinol

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0090
Total Syntheses of Anthracimycin and Anthracimycin B

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0091
PROCID: A Proximity-Based Drug Target-ID System

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0092
Saxitoxin Structure–Activity Relationships Reveal Selective Inhibitors of Na_V1.7

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0093
T-Shaped Benzimidazole Platform for ER-Targeting Fluorophores

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0094
Antiproliferative Effect of a Hybrid of Two Bistetrahydroisoquinoline Alkaloids

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0095
Overcoming Antimicrobial Resistance: Rational Design of Rifamycin Antibiotics

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0096
From Soil to Bench: Total Synthesis of Tigilanol Tiglate

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0097
An Enantioenriched Synthesis of (S)-Ketamine FREE ACCESS

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Peptide Chemistry
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0099
Ynamide-Mediated Peptide Synthesis FREE ACCESS

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0100
Transfer Hydrogenation of α-Aryl Imino Esters for the Synthesis of α-Amino Acid Esters

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0101
Cu-Catalyzed N–H Insertion of α-Alkyl-α-Diazo-acetates to Form N-Protected α-Alkyl Amino Esters

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0102
Rh-Catalyzed Polyfluoroaryl Amino Acids Synthesis

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0103
Synthesis of Glycopeptides Linked by Disulfide

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0104
Rh-Catalyzed Three-Component Coupling Reaction to Form α,β-Tetrasubstituted Amino Acids

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0105
Enantioselective Synthesis of α-Amino Acid Derivatives

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0106
MgO-Mediated Synthesis of Fmoc-Protected Amino Acid Hydroxamates FREE ACCESS

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Flow Chemistry
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0107
Benzophenone-Photocatalytic C4-Alkylation of Pyridinium Salts from C–H Bonds in Continuous Flow

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0108
Flow-Type Switchable Oxidation to Form Carboxylic Acids and Aldehydes from Primary Alcohols

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Erratum
0109
Shortest Synthesis of Lysergol and its Binding to 5-HT_1/2Receptors

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