Synfacts

Issue 03 · March 2023

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SYNFORM ISSUE 2023/03 FREE ACCESS

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Synthesis of Natural Products
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0213
Synthesis of (+)-Alterbrassicicene C FREE ACCESS

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0214
Synthesis of (+)-Candol A, (+)-Powerol A and (–)-Trachinol

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0215
Total Synthesis of (+)-Luminamicin

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0216
Synthesis of (–)-GA₁₈ Methyl Ester

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0217
Total Synthesis of (+)-Neobraclactone C

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0218
Total Synthesis of the Alkaloid (±)-Puberuline C

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0219
Total Synthesis of (+)-Maritimol FREE ACCESS

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Synthesis of Heterocycles
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0221
Dearomative Redox-Neutral Strategy for the Selective meta-Functionalization of Pyridines

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0222
Ni-Catalyzed Synthesis of 2-Heteroaryl Azetidines

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0223
Synthesis of Anilines from Boronic Acids FREE ACCESS

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0224
Rhodium-Catalyzed Cross-Coupling to Form Ketones

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0225
Gram-Scale Synthesis and Characterization of HAT

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0226
Selective Approach to 1,3-Oxazines via Controlled Amino-Diazidation and Amino-Iodoazidation of Alkenes

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0227
Synthesis of Imidazo[1,5-a]pyridines via Anomeric Stereoauxiliary Cleavage of d-Glucosamine

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0228
Bench-Stable Reagents for Introduction of Highly Lipophilic Thiofluoroalkyl Fragments

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0229
Perfluoroalcohol Solvent-Promoted Inverse Electron Demand Diels–Alder Reactions

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0230
Ring Expansion of Isoxazoles using Cu(I) Catalysis

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0231
Selective meta-Halogenation of Pyridines

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0232
[2+2] Cycloadditions to Access sp³-Rich Spirocycles FREE ACCESS

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0233
Synthesis of Pyrazolo[5,1-c][1,4]oxazine Derivatives from 2,2-Dichlorovinylacetophenones

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Synthesis of Materials and Unnatural Products
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0235
Trifunctional Lewis Pair Catalyzed Cyclopolymerization FREE ACCESS

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0236
Möbius Cyclophenylenes

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0237
BN-Doped Graphenoid Nanoribbons

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0238
2-Thioquinolines from Cascade Radical Cyclization

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0239
Dehydrofluorination of Phosphinines

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0240
Furan-Assisted Cyclization to Prepare Naphthalenophanes

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0241
Cu(I)-Catalyzed Cascade Synthesis of Benzo[b]fluorenes

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0242
A Large Planar N,S-Heterocycloarene

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0243
N→B-Bridged Quasi-[7]circulenes

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0244
Catalyst-Free Arene C–H Borylation

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0245
Lock the Fickle Macrocycle

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0246
Ring-Expansion from Tellurophenes to Telluropyrans

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Metals in Synthesis
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0247
Copper-Catalyzed Selective C–H Carboxylation of Alkenes with CO₂ FREE ACCESS

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0248
Wacker Oxidation of Methylenecyclobutanes to Cyclopentanones via a Semi-Pinacol-Rearrangement

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0249
Turning Carbocycles into N-Heterocycles by Cobalt-Catalyzed Nitrogen Atom Insertion FREE ACCESS

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0250
Gold-Catalyzed Thioamination of Terminal Alkynes with Sulfenamides

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0251
Cyclopropanols as a Source for Alkylation of 1-Arylpyrazole via Rhodium-Catalyzed C–H Activation

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0252
Palladium-Catalyzed Sequential Cyclization for Polycyclic Scaffold Synthesis

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0253
C3-Alkylation of Indoles via Ru-Catalyzed Transfer Hydrogenation and Borrowing Hydrogen Approaches

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0254
Atroposelective Iron-Catalyzed Coupling between Naphthols and Indoles

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0255
Synthesis of Aminobicyclo[3.1.1]heptanes by a Photoinduced Intermolecular [3σ+2σ] Cycloaddition

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0256
Ligand Control in the Synthesis of cis-and trans-1,3-Dienes Using Dual Nickel/Photoredox Catalysis

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0257
C(sp³)–H Allylation of Alkanes with in situ Formed Carbenes to Access Allylic Quaternary Carbon Centers

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0258
Indolo[2,3-b]indoles Syntheses via a Copper-Catalyzed Reaction Using (Aryl)(Mesityl)Iodonium Salts

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0259
Copper-Catalyzed Synthesis of Enantioenriched β^2,3,3-Amino Acids

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0260
Make Your Choice: Ligand-Dependent [2+2] and [4+2] Cycloaddition Reactions of 1,3-Dienes and Alkynes

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0261
Regioselective Alkene-Hydroamidation Using Dioxazolones and Isopropanol Under Rhodium Catalysis

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0262
Regioselective Hydroacylation of Alkenes via Triple Photoredox/Cobalt/NHC Catalysis

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0263
Lewis Acid-Promoted Asymmetric Dearomatization of Pyridines with Grignard Reagents under Cu(I) Catalysis

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0264
Desulfurization of Thioamides to Amines or Imines by Manganese-Catalyzed Hydrogenation

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0265
Asymmetric Tandem Copper- and Iridium-Catalyzed Reaction for the Construction of 1,3-Chiral Centers

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0266
A Three-Component Asymmetric Synthesis of 1,3-Diamines under Relay Amine and Palladium Catalysis

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0267
Photoinduced Nickel-Catalyzed Cross-Coupling of Aryl Bromides with Phthalimido Trifluoroethanol

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0268
Asymmetric Synthesis of Oxazoline-Spiroketals via Iridium-Catalyzed Domino Allylation/Spiroketalization

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0269
Synthesis of Esters via Manganese-Catalyzed Alkoxycarbonylation of Alkyl Chlorides

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0270
Asymmetric Intramolecular Reductive Coupling of Imines and Alkenes under Nickel Catalysis

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0271
Palladium-Catalyzed Enantioselective Allylic C–H Amination of Alkenes Induced by Blue Light

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0272
Novel Access to β‑Carboline-1-one Derivatives via Ru(II)-Catalyzed Annulation of Indole-2-Carboxamides

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0273
Access to Chiral Succinimides by Rhodium-Catalyzed Asymmetric Transfer Hydrogenation

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0274
Nickel-Catalyzed Synthesis of Polycyclic Imidazoles via Catalyst-Controlled endo-Selective Cyclization

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0275
Asymmetric Zirconium-Catalyzed Alkylalumination of Alkenes FREE ACCESS

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Polymer-Supported Synthesis
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0277
One-Pot Synthesis of Allyl- and Alkylamines through A³ Coupling with a Silica-Supported Ru/Cu-Bimetallic Catalyst

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0278
Synthesis of Cyclic Carbonates from Epoxides Using Silica-Supported Salophens and Salens

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0279
Cross-coupling of Cinnamyl Bromides and Alkyl Boronates Catalyzed by a Pd-Fe MOF FREE ACCESS

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0280
Conjugated Microporous Polymers as Photocatalysts for Hydroxylation of Phenylboronic Acids

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0281
[3+2] Cycloaddition of Cyanoarenes and NaN₃ with a Mesoporous Silica-Supported Lanthanum Complex

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0282
C–H Activation of 2-Arylbenzoxazinones by a Heterogeneous Magnetic Palladium Catalyst

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0283
Controllable Cyclization Reactions of Isonitriles Using a MOF-Based Palladium Catalyst

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0284
Switchable Perfluoroalkylation of Terminal Alkynes Promoted by Mesoporous Graphitic Carbon Nitride

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0285
Hydro(Deutero)dehalogenation of Aryl Bromides by Water as a Reductant and a Hydrogen Source

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0286
Friedel–Crafts Alkylation between Indoles or Pyrroles and β-Nitrostyrenes Using La(III)-Based MOF

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0287
Synthesis of Disulfides through Dehydrogenative Dimerization of Thiols Promoted by Zeolite ETS-10

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Organo- and Biocatalysis
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0289
Chiral Pyridoxal–Gold Rush in Asymmetric Carbonyl Catalysis FREE ACCESS

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0290
Sulfonium-Based EDA Complexes Grant Access to Electronically Diverse Aryl Radicals

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0291
Organocatalytic/Photochemical Approach to Regioselective Functionalization of Azines

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0292
Radical-Based 1,4-Difunctionalization of Two Electronically Differentiated Olefins

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0293
A Chemo-Enzymatic Dearomatization Cascade Approach to Enantioenriched Piperidines from Pyridines

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0294
Hydroalkylation of Olefins Mediated by Photochemically Generated NHC-Ligated Boryl Radicals

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0295
Photocatalytic Radical Addition to N-Sulfonyl Hydrazones as a C–H Alkylation Strategy

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0296
Organocatalysis Enables the Isotopic Labelling of Amino Acids

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0297
Organocatalytic Hydrophosphonylation Towards Enantioenriched Self-Recognizing Ureidophosphonates

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0298
Chiral Phosphoric Acid- and Photoredox-Catalyzed Enantioselective Giese Additions of α-Amino Radicals

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Innovative Drug Discovery and Development
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0299
Expanding the Toolbox of Cysteine-Reactive Probes

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0300
Structurally Guided Synthesis and Development of Novel Macrocyclic Antibiotics

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0301
High-Level Data Fusion Leads to the Discovery of a General Atropselective Iodination Catalyst

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0302
Raise the ALARM: An Enzyme-Controlled, Light-Activated RNA Modification Approach

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0303
Synthesis of an Improved Enterobactin–Muraymycin-Drug Conjugate Against Gram-Negative Bacteria

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0304
Small Molecule SST2 Agonist as a Potential Therapeutic for Acromegaly and Neuroendocrine Tumors

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0305
Discovery of Selective Inhibitor and Degrader of Mutant PI3Kα

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0306
Modular Total Synthesis of Antibacterial Nucleosides

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0307
Concise and Scalable Synthesis of Thalidomide FREE ACCESS

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0308
Development of Potent and Selective Dual Cyclin-Dependent Kinase 7 and 9 Inhibitors

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0309
Potent and Selective PARP7 Inhibitor, KMR-206, Regulates IFN-I Signaling

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0310
Harnessing Biocatalytic Cascades to Access Pharmaceutically Relevant Piperidines FREE ACCESS

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Peptide Chemistry
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0311
Cu-Catalyzed Introduction of Oxime Ethers into Peptides FREE ACCESS

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0312
Rh/Chiral Phosphoric Acid Cocatalyzed Synthesis of N-(Anthrancen-9-ylmethyl) Isoserines

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0313
Squaramide-Catalyzed Amino Acid Induced Tetrahydro-β-Carboline Synthesis

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0314
Visible-Light Photocatalysis for the Synthesis of Quaternary Alkynyl α‑Amino Esters

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0315
Photoinduced Coupling Reaction of Glycine Derivatives with N-Alkoxyphthalimides

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0316
Synthesis of Unnatural Amino Acids from Glycinates

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0317
Cu-Catalyzed Borylamination for the Synthesis β-Boryl-α-amino Esters

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0318
Chiral Aldehyde-Ni Dual-Catalyzed α-Propargylation to α-Amino Acids

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0319
One-Pot Synthesis of N-Methyl Dipeptides from Amino Acid-Derived Oxazolidinones FREE ACCESS

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Flow Chemistry
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0321
A Safe and Mild Protocol for the Synthesis of Dithiocarbamates under Continuous Flow Conditions

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