Synfacts

Issue 02 · February 2024

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A022
Zanda, Matteo: SYNFORM ISSUE 2024/02 FREE ACCESS

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Synthesis of Natural Products
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0111
Synthesis of (±)-Aleutianamine FREE ACCESS

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0112
Total Synthesis of (–)-Taxol

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0113
Total Synthesis of (+)-Discorhabdin V

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0114
Total Synthesis of (–)-Cyclopamine

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0115
Total Synthesis of (+)-Acremolactone B

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0116
Isolation and Bioinspired Synthesis of (+)-Orientanoid A

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0117
Synthesis of the Rubrolone Aglycon FREE ACCESS

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Synthesis of Heterocycles
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0119
Heteroarene Functionalization Using Solid Gas-MOF Reagents

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0120
Ring-Opening the Door to Amination: Nitrobenzene-Derived Azepines as Key Intermediates for N-Arylation

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0121
Skeletal Editing of Indoles and Pyrroles by LiHMDS Nitrogen Insertion Reaction FREE ACCESS

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0122
Efficient Access to Novel Vinyl Indomorphan Scaffolds

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0123
One-Pot Synthesis of Disubstituted Nicotinonitriles

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0124
Copper-Catalyzed Synthesis of Pyrozles from Sydnones and Sydnomines

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0125
Photoredox/Cobalt-Catalyzed Cascade Synthesis of 2,5-Disubstituted 1,3,4-Oxadiazoles

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0126
Radical-Mediated Synthesis of Isoquinolines

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0127
Bi-Catalyzed Trifluoromethylation Using CF₃SO₂Cl

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0128
Intramolecular Diels–Alder Cascade to Access 6- or 7-Aza-Indazoles

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0129
Metal-Controlled Regioselective Synthesis of Imidazoles and Pyrroles from 2H-Azirines

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0130
Palladium-Catalyzed Asymmetric C–H Functionalization Reactions

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0131
sp²–sp³ Coupling of Unprotected Halogenated Anilines with Grignard Reagents

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Synthesis of Materials and Unnatural Products
z0133
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0133
Conjugated [5]Cumulene Polymers from Propargylic Monomers FREE ACCESS

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0134
Tetrafluorenofulvalene: To Be Single or Double?

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0135
1,2-Azaborines via Ring-Opening Benzannulation

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0136
Ring Expansion Polymerization via Alkyne Metathesis

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0137
B₂,N₄-Doped Heptacene

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0138
Mild Aryne Generation from Triaryloxonium

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0139
Chiral Emissive Corral-Like Macrocycles

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0140
Facile Ipso-Nitration of Organosilanes

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0141
Tetrahedral Nanographene

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0142
Ring-Size Controlled Racemization

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0143
Phthalimides from Maleimides and Triethylamine

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0144
Anthracene with Continuous B–N Bonds

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Metals in Synthesis
z0145
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0145
Nickel-Catalyzed Hydrocyanation of Alkynes Using a Malononitrile as Transnitrilation Reagent FREE ACCESS

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0146
Asymmetric Intramolecular Oxyamination of Alkenes Enabled by a Chiral-at-Ruthenium Catalyst

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0147
Photoelectrocatalyzed Synthesis of Chiral Cyclobutanes FREE ACCESS

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0148
Synthesis of Atropoisomeric Dienes via Enantioselective Rhodium-Catalyzed Hydroarylative Cyclization

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0149
Synthesis of Functionalized Alkynes via Regioselective Ni-Catalyzed Hydroalkynylation

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0150
Photochemical Amination of Aryl Chlorides Using Werner Salt

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0151
Fe/Blue Light Catalyzed Electrophilic Aromatic Substitution of Acyl Nitrene Precursors

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0152
Rhodium/CPA Co-Catalyzed Multicomponent Synthesis of Chiral β-Amino Esters

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0153
A General Photochemical Protocol for Alkene Hydrofluoroalkylation under Iron and Thiol Catalysis

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0154
Stereoconvergent Synthesis of Z-Allylsilanes by Iron-Catalyzed 1,4-Hydrosilylation of Conjugated Dienes

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0155
Synthesis of Allylated Arenes via Ruthenium-Catalyzed Aromatic C–H Allylation

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0156
Synthesis of Chiral Alkynes via Ni-Catalyzed Cross-Electrophile Coupling

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0157
Hydroxylation of Free Amines Using a Palladium(CarboxPyridone) Catalytic System

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0158
Synthesis of δ-Lactams via Biomimetic Polycyclization Initiated by an Iridium Acylnitrenoid Transfer

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0159
Iridium-Catalyzed Terminal C(sp³)–H Amidation of Internal Alkenes via Olefin Chain Walking

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0160
Enantioconvergent Reductive Nickel Catalysis Enables Access to Chiral 2-Alkyl-Pyridines

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0161
Rhodium-Catalyzed Dynamic Kinetic Asymmetric Fluorination of Racemic Trichloroacetimidates

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0162
Enantioconvergent C(sp³)–C(sp²) Stille Cross-Coupling under Photoredox/Nickel Catalysis

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0163
Fluorolocatonization of Ene-Carboxylic Acid via Pd-Catalyzed Dyotropic Rearrangement

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0164
Hiyama Cross-Coupling of Aryl Chlorides with Aryl Trimethoxysilanes using Pd(NHC) Precatalysts

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0165
Mild Access to Aryl–Alkyl Ketones Enabled by Photoinduced Nickel Catalysis

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0166
An Electrochemical Approach to the Copper-Catalyzed Azidocyanation of Alkyl and Aryl Alkenes

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0167
Ruthenium-Catalyzed Intermediate Kinetic Resolution to Access Two Chiral Products

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0168
Photocatalyzed Synthesis of Tricyclic Aza-Arenes by Pyridyl Radical Trapping with Diynes and Dienes

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0169
Decarboxylative Difunctionalization of Alkenes Enabled by Nickel/Photoredox Catalysis

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0170
The Murahashi Reaction: Palladium-Catalyzed Cross-Coupling of Vinyl Halides with Organolithium Reagents FREE ACCESS

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Polymer-Supported Synthesis
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0171
Cross-Coupling Reactions Catalyzed by Regularly Spaced Copper Atom Pairs on Polymeric Carbon Nitride FREE ACCESS

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0172
C(sp³)–H Amination of Alkanes by Pd Nanoparticles on Gallium Nitrides

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0173
Cyclization of Propargylamines with CO₂ Catalyzed by a Ag₄ Nanocluster

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0174
A³ Coupling Catalyzed by a Tridentate Cu–NHC Nanocluster

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0175
N-Alkylation of Anilines with Primary Alcohols by MOF-Derived CoN_x Nanoparticles on N-Doped Carbon

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0176
Hydrodeoxygenation of Aromatic Ketones and Aldehydes, and Benzylic Alcohols Using Co/CoO_x

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0177
An Imidazolium-Functionalized Cage Catalyst for Site-Selective C(sp³)–H Chlorination of Amides

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0178
Borylation with an N-Heterocyclic Carbene-Borane and a CdS Photocatalyst

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0179
The Suzuki–Miyaura Coupling by a Reduced Polynuclear Palladium Complex Supported on Alumina

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0180
Transfer Hydrogenation of Azo Compounds with MeOH or EtOH by a Cobalt Single Atomic Catalyst

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0181
N-Arylation of Amides with Aryl Halides Catalyzed by a CuO Nanoplate

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Organo- and Biocatalysis
z0183
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0183
Enzymatic Hydrogen Atom Transfer Allows for Remote Stereocontrol Using Aza-arenes FREE ACCESS

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0184
Tuning Electron Donation Capacity Enables Regio-divergent NHC/Base-Catalyzed Aminolactone Synthesis

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0185
Enantioselective Construction of Bicyclo[2.1.1]hexane Bioisosteres

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0186
Enantioselective α-Arylation of β-Keto Amides with Arynes Enabled by Phase-Transfer Organocatalysis

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0187
Organocatalytic Highly Selective Nitroso-Diels–Alder Reaction of Conjugated Trienes

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0188
One-Pot Trifluorination/Cyclization Cascade Enabled by I(I)/I(III) Catalysis

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0189
Photocatalysis-Enabled Alkylation of C(sp³)–H Bonds with Sulfonylhydrazones

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0190
Organocatalytic Asymmetric Decarboxylative Protonation of Aminomalonic Acids

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0191
Stereoconvergent Biocatalysis – The Conversion of E/Z-Silyl Enol Ethers into Enantiopure α-Branched Ketones

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0192
Acid-Catalyzed Ring-Opening Olefination of Carbonyl Compounds Using Cyclic Ketals

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Innovative Drug Discovery and Development
z0193
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0193
Enantioselective Indole C3 Oxidation FREE ACCESS

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0194
Predicting Late-Stage C–H Borylations of Drug Molecules

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0195
Chiral Lithium Amide Improves Stereoselectivity and Yield of Tuberculosis Drug Bedaquiline

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0196
A Rh(III)-Catalyzed C–H Activation/[5+2] Annulation Sequence Allows Access to 1,2-Diazepinones

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0197
Cyclopropanation: Vitamin B12 as Photoredox Catalyst

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0198
Discovery of [¹¹C]MK-8056: A Selective mGluR₂ Negative Allosteric Modulator PET Tracer

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0199
Introducing Boronaphthoids as the New Boron-Containing Drug Chemotypes

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0200
One-Pot Hydrogenation Allows for Quick Accesses to Pharmaceuticals

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0201
Photochemical Synthesis of a Cubyl Derivative of Dapsone

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0202
Phosphine Catalysis of the Fluorination of Unactivated Tertiary Alkyl Chlorides under Mild Conditions

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0203
Regiodivergent Access to ortho-Functionalized Anilines via Photoexcitation of Aryl Azides

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0204
Radical Bicyclopentylation of Alcohols

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0205
Total Synthesis of Opioid Precursor (−)-Thebaine

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0206
Total Synthesis of Nimbolide and its Analogues

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0207
Photocatalyzed [2+2] Cycloadditions of 1,3,2-Dioxaboroles to Alkenes to Afford Cyclobutanes and 1,4-Dicarbonyls

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0208
Radical [4+1] Annulation Allows for Late-Stage Indole Synthesis

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0209
Stereodivergent Synthesis of 3,3′-Disubstituted Oxindoles by N-Heterocyclic Carbene/Nickel Catalysis

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Peptide Chemistry
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0211
Atom-Economical N-to-C Peptide Elongation FREE ACCESS

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0212
Three-Component Reaction of Diazoacetates, Sulfonamides, Imines to Form Unnatural Amino Acids

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0213
Regio-Selective Arylation Reaction for the Trp-Unit of Oligopeptides

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0214
Copper-Catalyzed Asymmetric Arylation to Synthesize β-Amino Ester Precursor

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0215
Electrochemical Arylation of Cysteine-Containing Peptides

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0216
Microwave-Assisted Transamidation of Boc-Activated Secondary Amides

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0217
Late-Stage C3_Ar Functionalization of Tyrosine and Tyrosine-Containing Peptides with Maleimides

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0218
Nucleophilic Hydrazide-Catalyzed Chlorination of Tyrosine-Containing Peptides

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0219
Synthesis of α-Quaternary Amino Esters via Intramolecular Rearrangement FREE ACCESS

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0220
Synthesis of N-Aryl Amino Acid Esters

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Flow Chemistry
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0221
Simmons–Smith Cyclopropanation in Flow

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0222
Continuous-Flow Chemoenzymatic Enantioselective Synthesis of Chiral α-Fluoromethyl Amines

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