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Publication Date: 07 March 2025

letter > Small Molecules in Medicinal Chemistry

Garg, Aakriti; Bhattacharya, Bireswar; Samanta, Uttam; Singha, Subhankar; Ghosh, Dipanjan; Bhowmik, Subhendu; Jaisankar, Parasuraman; Gupta, Sreya: Phototriggered Migration of Indole-Based Cationic Fluorophore from Mitochondria to Nucleolus in Live Cells

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Sharma, Manisha; Leadbeater, Nicholas E.: Preparation of Symmetric and Nonsymmetric Imines from Primary Benzyl Amines by Means of an Oxidative Functionalization Reaction Using an Oxoammonium Salt Bearing the Nitrate Anion

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Jiang, Yuan-Xu; Liao, Li-Li; Ye, Jian-Heng; Yu, Da-Gang: Visible-Light-Driven Thiolate-Catalyzed Carboxylation of C(sp²)–H Bonds in Azines with Carbon Dioxide

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Publication Date: 06 March 2025

account > Small Molecules in Medicinal Chemistry

Purohit, Priyank; Bhatt, Akanksha; Mittal, Ravi Kumar: Ruthenium-Based Small-Molecule Complexes: A Promising Approach for Drug Discovery

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letter > Emerging Trends in Organic Chemistry: A Focus on India

Kumar, Prashant; Kant, Ruchir; Srivastava, Ajay Kumar: Iodine-Mediated Oxidative [3+2] Annulation of Quinoxalinones with Oxime Esters: An Approach toward Imidazo[1,2-a]quinoxalin-4(5H)-ones

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letter > Small Molecules in Medicinal Chemistry

Shaikh, Arbaz Sujat; Rathod, Mahipal Singh; Vemula, Divya; Makhal, Priyanka N.; Bhandhari, Vasundhara; Kaki, Venkata Rao: Metal-Free Amidation and Selenoamidation of 2-Methylquinolines with Secondary Amines Using Selenium Dioxide, and Antibacterial Evaluation of the Products

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Publication Date: 04 March 2025

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Cheng, Guang; Cai, Chenchen; Zhang, Xingxian; Qiu, Guanyinsheng; Li, Shaoyu: Catalyst-Free Radical Dearomatization of Phenols with Aryldiazonium Tetrafluoroborates and DABCO·(SO₂)₂

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Publication Date: 28 February 2025

letter > Emerging Trends in Organic Chemistry: A Focus on India

Malvi, Payal; Mistry, Dharti; Karunakar, Galla V.; Rajput, Diksha; Lenin, Dandamudi V.: Baylis–Hillman Adducts as a Valuable Source for Synthesis of Functionalized [4,4,4]-Propellone Dilactone Derivatives

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Publication Date: 24 February 2025

perspectives > Small Molecules in Medicinal Chemistry

Goel, Kapil Kumar; Singhal, Peeush; Marianesan, Arockia Babu; Pandey, Sarvesh Kumar; Kumar, Roshan; Singh, Thakur Gurjeet; Tyagi, Yogita; Gaidhane, Shilpa; Singh, Mahendra Pratap; Dwivedi, Ashish Ranjan: A Decade of Piperazine-Based Small Molecules Approved by U.S. FDA: Exploring the Medicinal Chemistry Impact of this Versatile Pharmacophore

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Publication Date: 21 February 2025

letter > Small Molecules in Medicinal Chemistry

Chaudhury, Subhabrata; Wetzel, Edward A.; Elmansy, Mohamed F.; Hanson, Alicia M.; Brown-Ford, Sandra; Gleason, Alexandra; Perera, K. L. Iresha Sampathi; Sem, Daniel S.; Donaldson, William A.: Analogues of the Potent and Selective ERβ Agonist trans-4-(4-Hydroxyphenyl)cyclohexanemethanol: Synthesis and Evaluation

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Desai, Bhargav; Bharodiya, Akshay; Seshathre, Shruti; Patel, Raj N.; Dholakiya, Bharatkumar; Satani, Piyushkumar; Kanchupalli, Vinaykumar; Naveen, Togati: Microwave-Assisted Copper-Catalyzed Electrophilic Amination of Arylboronic Acids: A Rapid Approach to Arylhydrazides

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Wang, Qing; Mei, Guangyao; Luo, Zi Jin; Sun, Xiaotong; Weng, Jianquan; Zhang, Guofu: Light-Induced Metal-Free Catalyzed C–H Alkylation of (Iso)Quinolines

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Publication Date: 19 February 2025

perspectives > 14th EuCheMS Organic Division Young Investigator Workshop

Cunningham, Laura: Supramolecular Chemistry: An Enabling Tool for Asymmetric Catalysis

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Publication Date: 18 February 2025

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Li, Xiaolan; Luo, Haiqing: Rhodium(III)-Catalyzed C–C Bond Formation by Direct C–H Activation

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letter > First-Row Transition-Metal Catalysis for Organic Synthesis

Dong, Haiyan; Ding, Xinrang; Wang, Chuan: Nickel-Catalyzed Cross-Electrophile [2+4] Annulation of Benzynes

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Shimose, Asuha; Nagashima, Yuki: Photoinduced Dearomative Multiple Functionalization of Quinolines to Construct Highly Substituted 3D Frameworks

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Publication Date: 13 February 2025

account > Small Molecules in Medicinal Chemistry

Tomohara, Keisuke; Nose, Takeru; Nambu, Hisanori: Straightforward Synthesis of Unnatural α,α-Disubstituted α-Amino Acid Derivatives Using Readily Accessible Building Blocks

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Yang, Xingheng; Zhang, Chi; Wang, Cheng-Qiang; Feng, Chao: Expedient Access to Structural Complexity via Radical β-Fragmentation of N–O Bonds

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Publication Date: 12 February 2025

account > Small Molecules in Medicinal Chemistry

Thaker, Aanal; Patel, Shrusti; Dey, Rajdeep; Shaw, Suman; Bhatt, Hardik; Patel, Bhumika; Chaube, Udit: Advancements in mTOR Inhibitors for Non-Small-Cell Lung Cancer: Mechanisms, Efficacy, and Future Perspectives

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Publication Date: 10 February 2025

letter

Zhu, Junmei; Zhang, Ting; Bi, Ruru: Gram-Scale Total Synthesis of Cordiachrome B

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