Synfacts

Issue 08 · August 2019

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A113
SYNFORM ISSUE 2019/08 FREE ACCESS

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Synthesis of Natural Products and Potential Drugs
z0833
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0833
Synthesis of (+)-Longirabdiol, (–)-Longirabdolactone, and (–)-Effusin FREE ACCESS

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0834
Synthesis of a PDE10A Inhibitor

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0835
Synthesis of E2212

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0836
Synthesis of Taselisib

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0837
Synthesis of Taselisib

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0838
Syntheses of (±)-Rhodomolleins XX and XXII

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0839
Total Syntheses of (–)-Daphlongamine H and (–)-Isodaphlongamine H

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0840
Total Synthesis of Englerins A and B

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0841
Synthesis of (–)-7-Deacetoxyalcyonin Acetate FREE ACCESS

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0842
Synthesis of a Renin Inhibitor

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0843
Synthesis of a TAK-480 Fragment

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0844
Synthesis of TAK-063

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0845
Synthesis of (+)-Arborisidine

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0846
Synthesis of Dolutegravir

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0847
Synthesis of Dolutegravir

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0848
Synthesis of an Edoxaban Fragment

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0849
Synthesis of (+)-Principinol D

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0850
Synthesis of Tofogliflozin

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0851
Synthesis of BMS-986236

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Synthesis of Heterocycles
z0853
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0853
Synthesis of Two Azaborine Building Blocks FREE ACCESS

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0854
Phosphonium-Salt-Catalyzed Synthesis of Fused Aziridines by an Aza-Darzens Reaction

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0855
Chemoselective Demethylation of Methoxypyridines over Anisoles

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0856
Catalytic Azole Acylation with Acyl Fluorides

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0857
Acridone Synthesis by Double Amination of Dibromobenzophenones

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0858
Enantioselective Catalytic Aryl-Alkenylation To Give Dihydrobenzofurans

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0859
Synthesis of 1,2-Benzothiazine 1-Imines as New Heterocyclic Scaffolds

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0860
Selective C–H Alkenylation of Isoxazoles

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0861
Gold(III)-Catalyzed Synthesis of 4-Aminooxazoles

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0862
Synthesis of 1,4-Benzothiazines by Iodide-Catalyzed Alkene Sulfenoamination

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0863
Copper-Catalyzed Synthesis of 3,4-Dihydroquinazolines from Anthranils

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0864
Silver-Catalyzed Synthesis of Trifluoromethylated Triazines and Pyridines

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0865
Asymmetric Synthesis of Dihydrobenzofurans by an Organocatalytic [4+1] Cyclization

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0866
DBU-Mediated Synthesis of Bicyclic Heterocycles

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Synthesis of Materials and Unnatural Products
z0867
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0867
A Prefix to SuFEx

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0868
The Whole Kit and Caboodle: A Ferrocenyl Halogen Bonding Rotaxane for Electrochemical Bromide Sensing

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0869
It takes Strained Alkynes to make Polycyclic Aromatic Hydrocarbons

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0870
Forced into Antiaromaticity

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0871
Tetrahydroquinoline-Fused Fullerenes

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0872
(N-Phenylfluorenylidene)acridanes: Mechanochromic BAEs

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0873
Organocopper Cross-Coupling for Crowded Environments

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0874
Deep LUMO Level Diimide π-Electron Core

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0875
Renewing the Synthesis of Sterically Hindered Phenanthrenes

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0876
Studies of Polyarylether COFs

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0877
Cranking out Functionalized Helicenes

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0878
Unlocking a [2.2.2]Carbon Nanocage

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Metals in Synthesis
z0879
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0879
Diastereoselective [4+4] Cycloadditions FREE ACCESS

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0880
Asymmetric Copper-Catalyzed Hydroamination of Enamines

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0881
Iridium-Catalyzed Asymmetric Hydroalkynylation of Unactivated Alkenes FREE ACCESS

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0882
Nickel-Catalyzed Amination of Phenols

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0883
Mild Copper-Catalyzed N-Arylation of Sulfoximines

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0884
Enantioselective Synthesis of Chiral Homoallylic Tertiary Alcohols through Copper Catalysis

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0885
Dual Nickel/Photo-Catalyzed Esterification of Aryl Halides

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0886
Nickel-Catalyzed Cyano-Borrowing Reaction Affording β-Cyano Ketones

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0887
Cobalt-Catalyzed Aminocarbonylation of Alkyl Tosylates

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0888
Synthesis of Chiral β-Nitroamides

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0889
Enantioselective Synthesis of Tertiary α-Silyl Alcohols

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0890
The Catalytic Kulinkovich Reaction FREE ACCESS

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0891
Synthesis of Areneamides

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0892
Intermolecular [2+2] Carbonyl–Olefin Photocycloadditions Enabled by a Copper(I)–Norbornene Complex

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0893
Regioselective Palladium-Catalyzed C–H Iodination of Alkenes

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0894
Amide Enolate Surrogates in Asymmetric Allylation Reactions

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0895
Catalytic Preparation of Potassium Acyltrifluoroborates

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0896
Amination of Triaryl Phophates

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0897
Palladium-Catalyzed Dearomative Carboamination

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0898
Counterion-Controlled Cobalt-Catalyzed Addition of Cyclopropanols to Oxabyciclic Alkenes

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0899
Palladium-Catalyzed Enantioselective N‑Alkylation of Indoles

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0900
Decarboxylative Alkylation

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0901
Iodination/Cross-Coupling Cascade Reaction

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0902
Radical-Driven Deoxygenation of Secondary Alcohols: The Barton–McCombie Reaction FREE ACCESS

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0903
Nickel-Catalyzed Reaction of Umpolung Carbonyls and Alkyl Halides

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0904
Ligand-Controlled Selection of Diastereoisomers in Asymmetric 1,3-Dipolar Cycloaddition

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0905
Ruthenium-Catalyzed Transfer Hydrogenation of α-Acetamido Benzocyclic Ketones

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0906
Intramolecular Asymmetric Hydroamination of Allenes

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0907
Preparation of 2-Substituted Propenes

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0908
Nickel/Manganese Dual-Catalyzed Hydroalkylation of Olefins

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Polymer-Supported Synthesis
z0909
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0909
Ion-Exchange-Resin-Supported Hydrogen Fluoride for Fluorination Reactions FREE ACCESS

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0910
Michael Addition on a Squaramide-Decorated Covalent Organic Framework

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0911
Aqueous Flow Hydroxycarbonylation on an Amphiphilic Polymer-Supported Pd Complex

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0912
Transfer Hydrogenation of Aryl Ketones on Mesoporous Silica-Supported Nickel

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0913
Buchwald–Hartwig Amination on NHC-Pd Immobilized on Wang Resin

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0914
Couplings of Aryl Halides with Arylboronic Acids on Silica-Supported Nickel

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0915
Palladium-Catalyzed Dehydrogenative Aromatization of Cyclic Amines

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0916
Dehydrogenation of N-Heterocycles with Cobalt Nanocrystals on Carbon

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0917
Suzuki–Miyaura Coupling on Aluminosilicate-Encapsulated Palladium Nanoparticles

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0918
Benzylic C(sp³)–H Bond Oxidation Catalyzed by a Supported Manganese Complex

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0919
Alumina-Supported Copper Oxide Hydrogenation Catalyst

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0920
Hydroxylation of Alkyl Halides on an Aminopolystyrene-Supported Ionic Liquid

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0921
Nickel-Catalyzed Cross-Coupling of Aryl Chlorides with Organolithiums

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0922
Porous NiCo-Catalyzed Reduction of Nitroarenes with Ammonia Borane

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Organo- and Biocatalysis
z0923
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0923
Enzyme-Catalyzed Site-Selective C–H Amidation

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0924
Chiral Phosphine Catalyzed Asymmetric Staudinger–aza-Wittig Reaction

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0925
Photochemical Organocatalytic Borylation of Alkyl Halides and Sulfonates

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0926
Benzothiophene-Catalyzed Oxidative Coupling of 2-Naphthols

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0927
Benziodoxole-Catalyzed Anti-Markovnikov Hydroazidation of Olefins

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0928
Organocatalytic Enantioselective Dichlorination of Cyclic Styrenes

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0929
[4+2] Cycloaddition via NHC-Bound Aza-ortho-Quinone Methides

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0930
Diazaphospholene-Catalyzed Reductive Ireland–Claisen Rearrangement FREE ACCESS

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0931
Asymmetric Catalytic Transannular Morita–Baylis–Hillman Reaction

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0932
A Bifunctional Catalyst Permits Atroposelective Aromatization

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0933
Enantioselective Protonation of Disilyl Ketene Acetals with Water or Methanol

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0934
Thiazolium Salt Catalyzed Asymmetric Benzoin Reaction FREE ACCESS

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Chemistry in Medicine and Biology
z0935
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0935
A Mitochondria-Targeting Calcium Dye FREE ACCESS

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0936
Small-Molecule Inhibitors of CRISPR-Cas9

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0937
In Vivo Imaging of Glucose Uptake

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0938
Chemical Diversification of Pleuromutilin

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0939
Highly Selective Insulin-Degrading Enzyme Inhibitors

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0940
Selective α-Glycosidation of Sialic Acid

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0941
Short Synthesis of the 3-Deazaguanosine RNA Building Block

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0942
SCOTfluors: Small, Conjugatable, Orthogonal, and Tunable Fluorophores

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0943
Photoactivated Fluxional Fluorophore Enables Extended Time-Lapse Microscopy

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Peptide Chemistry
z0945
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0945
Organcatalytic Transamination for the Synthesis of α-Amino Acids FREE ACCESS

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0946
One-Pot Four-Component Strategy for Electrophilic Fluorination

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0947
Site-Selective Reduction of Cyclosporine A by Borane Catalysis

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0948
Palladium-Catalyzed β-C–H Arylation of N-Methylated Peptides

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0949
Synthesis of Rigidified Cyclic Peptides by Ring-Closing Metathesis

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0950
Azotide Ligands for Hetero-Diels–Alder Reactions FREE ACCESS

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0951
Synthesis of N-Terminal Cysteinyl Thioesters

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0952
Nickel-Catalyzed Synthesis of Amides from Methyl Esters

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0953
Pd-Catalyzed Arylation of α-Amino Esters with Diaryliodonium Triflates

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Flow Chemistry
z0955
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0955
Continuous-Flow Preparation of Alkynylzinc and its Subsequent Cross-Coupling Reaction

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0956
Continuous-Flow Electrochemical Oxidation with Hypervalent Iodine Reagents

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0957
Syntheses of Sulfilimines and Sulfoximines in a Flow System

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0958
Flow Synthesis of Vaborbactam

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0959
Flow Synthesis of Ceramide d-erythro-CER[NDS]

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0960
Synthesis of Sialic Acid Derivatives in a Continuous-Flow Enzymic Reactor

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0961
Cascade Oxidation over Contiguous Dual Catalyst Beds in Continuous Flow

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Erratum
0962
Iron-Catalyzed Synthesis of Fluoroalkylated 2H-Azirines from Alkynes

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0962
Continuous-Flow, Michaelis−Arbuzov Rearrangement

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